NO950319L - Inhibitorer for c-AMP fosfodiesterase og TNF - Google Patents
Inhibitorer for c-AMP fosfodiesterase og TNFInfo
- Publication number
- NO950319L NO950319L NO950319A NO950319A NO950319L NO 950319 L NO950319 L NO 950319L NO 950319 A NO950319 A NO 950319A NO 950319 A NO950319 A NO 950319A NO 950319 L NO950319 L NO 950319L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- directed
- tnf
- inhibitors
- amp phosphodiesterase
- Prior art date
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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- C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C205/59—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms
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- C07C217/80—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings
- C07C217/82—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring
- C07C217/88—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring the oxygen atom of at least one of the etherified hydroxy groups being further bound to a carbon atom of a ring other than a six-membered aromatic ring
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- C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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- C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
- C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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- C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
- C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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- C07C311/22—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms
- C07C311/29—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
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- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
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- C07C2601/14—The ring being saturated
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- C07C2602/42—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing seven carbon atoms
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Applications Claiming Priority (9)
Application Number | Priority Date | Filing Date | Title |
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GB929216005A GB9216005D0 (en) | 1992-07-28 | 1992-07-28 | New compounds |
GB929215989A GB9215989D0 (en) | 1992-07-28 | 1992-07-28 | Novel compounds |
GB929216008A GB9216008D0 (en) | 1992-07-28 | 1992-07-28 | Novel compositions of matter |
GB929216006A GB9216006D0 (en) | 1992-07-28 | 1992-07-28 | New use |
GB929216764A GB9216764D0 (en) | 1992-08-07 | 1992-08-07 | Novel compounds |
GB939310633A GB9310633D0 (en) | 1993-05-21 | 1993-05-21 | New compositions of matter |
GB939310938A GB9310938D0 (en) | 1993-05-27 | 1993-05-27 | New compositions of matter |
GB939311281A GB9311281D0 (en) | 1993-06-01 | 1993-06-01 | Novel composition of matter |
GB939314847A GB9314847D0 (en) | 1993-07-16 | 1993-07-16 | New use |
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NO950319D0 NO950319D0 (no) | 1995-01-27 |
NO950319L true NO950319L (no) | 1995-03-27 |
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NO950319A NO950319L (no) | 1992-07-28 | 1995-01-27 | Inhibitorer for c-AMP fosfodiesterase og TNF |
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JP (1) | JP3775684B2 (da) |
AT (1) | ATE282025T1 (da) |
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DE (1) | DE69333688T2 (da) |
DK (1) | DK0652868T3 (da) |
ES (1) | ES2227519T3 (da) |
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IL (1) | IL106517A0 (da) |
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NO (1) | NO950319L (da) |
NZ (1) | NZ254881A (da) |
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Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9007762D0 (en) * | 1990-04-05 | 1990-06-06 | Beecham Group Plc | Novel compounds |
US5393788A (en) * | 1990-07-10 | 1995-02-28 | Smithkline Beecham Corporation | Phenylalkyl oxamides |
US5124455A (en) * | 1990-08-08 | 1992-06-23 | American Home Products Corporation | Oxime-carbamates and oxime-carbonates as bronchodilators and anti-inflammatory agents |
AU9030691A (en) * | 1990-11-06 | 1992-05-26 | Smithkline Beecham Corporation | Imidazolidinone compounds |
IE71647B1 (en) * | 1991-01-28 | 1997-02-26 | Rhone Poulenc Rorer Ltd | Benzamide derivatives |
-
1993
- 1993-07-28 PL PL93307265A patent/PL307265A1/xx unknown
- 1993-07-28 CZ CZ95147A patent/CZ14795A3/cs unknown
- 1993-07-28 NZ NZ254881A patent/NZ254881A/en unknown
- 1993-07-28 CA CA002140441A patent/CA2140441C/en not_active Expired - Lifetime
- 1993-07-28 JP JP50433094A patent/JP3775684B2/ja not_active Expired - Lifetime
- 1993-07-28 AT AT93917937T patent/ATE282025T1/de active
- 1993-07-28 EP EP93917937A patent/EP0652868B1/en not_active Expired - Lifetime
- 1993-07-28 IL IL10651793A patent/IL106517A0/xx unknown
- 1993-07-28 MX MX9304571A patent/MX9304571A/es unknown
- 1993-07-28 DK DK93917937T patent/DK0652868T3/da active
- 1993-07-28 DE DE69333688T patent/DE69333688T2/de not_active Expired - Lifetime
- 1993-07-28 WO PCT/GB1993/001597 patent/WO1994002465A1/en active IP Right Grant
- 1993-07-28 ES ES93917937T patent/ES2227519T3/es not_active Expired - Lifetime
- 1993-07-28 AU AU47176/93A patent/AU4717693A/en not_active Abandoned
- 1993-07-28 HU HU9500265A patent/HUT72656A/hu unknown
- 1993-07-28 PT PT93917937T patent/PT652868E/pt unknown
-
1995
- 1995-01-27 FI FI950375A patent/FI950375A0/fi unknown
- 1995-01-27 NO NO950319A patent/NO950319L/no unknown
Also Published As
Publication number | Publication date |
---|---|
ES2227519T3 (es) | 2005-04-01 |
AU4717693A (en) | 1994-02-14 |
NZ254881A (en) | 1996-09-25 |
PL307265A1 (en) | 1995-05-15 |
ATE282025T1 (de) | 2004-11-15 |
JP3775684B2 (ja) | 2006-05-17 |
FI950375A (fi) | 1995-01-27 |
JPH08503925A (ja) | 1996-04-30 |
HU9500265D0 (en) | 1995-03-28 |
DE69333688T2 (de) | 2005-11-03 |
HUT72656A (en) | 1996-05-28 |
NO950319D0 (no) | 1995-01-27 |
EP0652868A1 (en) | 1995-05-17 |
CA2140441A1 (en) | 1994-02-03 |
FI950375A0 (fi) | 1995-01-27 |
MX9304571A (es) | 1994-05-31 |
CA2140441C (en) | 2006-11-21 |
EP0652868B1 (en) | 2004-11-10 |
DK0652868T3 (da) | 2005-02-14 |
PT652868E (pt) | 2005-01-31 |
CZ14795A3 (en) | 1996-07-17 |
IL106517A0 (en) | 1994-08-26 |
DE69333688D1 (de) | 2004-12-16 |
WO1994002465A1 (en) | 1994-02-03 |
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