NO940927L - Kondenserte tricykliske nitrogenholdige heterocykler som substans-P-reseptor-antagonister - Google Patents

Kondenserte tricykliske nitrogenholdige heterocykler som substans-P-reseptor-antagonister

Info

Publication number
NO940927L
NO940927L NO940927A NO940927A NO940927L NO 940927 L NO940927 L NO 940927L NO 940927 A NO940927 A NO 940927A NO 940927 A NO940927 A NO 940927A NO 940927 L NO940927 L NO 940927L
Authority
NO
Norway
Prior art keywords
pct
substance
receptor antagonists
containing heterocycles
condensed tricyclic
Prior art date
Application number
NO940927A
Other languages
English (en)
Norwegian (no)
Other versions
NO940927D0 (no
Inventor
Iii John Adams Lowe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO940927D0 publication Critical patent/NO940927D0/no
Publication of NO940927L publication Critical patent/NO940927L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO940927A 1991-09-26 1994-03-15 Kondenserte tricykliske nitrogenholdige heterocykler som substans-P-reseptor-antagonister NO940927L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76648891A 1991-09-26 1991-09-26
PCT/US1992/006819 WO1993006099A1 (en) 1991-09-16 1992-08-20 Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists

Publications (2)

Publication Number Publication Date
NO940927D0 NO940927D0 (no) 1994-03-15
NO940927L true NO940927L (no) 1994-03-15

Family

ID=25076576

Family Applications (1)

Application Number Title Priority Date Filing Date
NO940927A NO940927L (no) 1991-09-26 1994-03-15 Kondenserte tricykliske nitrogenholdige heterocykler som substans-P-reseptor-antagonister

Country Status (19)

Country Link
US (1) US5527808A (de)
EP (1) EP0607164B1 (de)
JP (1) JP2535134B2 (de)
CN (1) CN1071168A (de)
AT (1) ATE216996T1 (de)
AU (1) AU2481292A (de)
BR (1) BR9206500A (de)
CA (1) CA2118704C (de)
CZ (1) CZ59394A3 (de)
DE (1) DE69232588T2 (de)
DK (1) DK0607164T3 (de)
ES (1) ES2174836T3 (de)
FI (1) FI941212L (de)
HU (1) HU9400728D0 (de)
MX (1) MX9205242A (de)
NO (1) NO940927L (de)
PT (1) PT100901A (de)
WO (1) WO1993006099A1 (de)
ZA (1) ZA927370B (de)

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FR2700472B1 (fr) 1993-01-19 1995-02-17 Rhone Poulenc Rorer Sa Association synergisante ayant un effet antagoniste des récepteurs NK1 et NK2.
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
EP0653208A3 (de) * 1993-11-17 1995-10-11 Pfizer Substanz P Antagonisten zur Behandlung oder Verhütung des sonnenbrandes.
EP0659409A3 (de) * 1993-11-23 1995-08-09 Pfizer Substanz P Antagonisten zur Hemmung der Angiogenese.
EP0655246A1 (de) * 1993-11-30 1995-05-31 Pfizer Inc. Substanz P Antagonisten zur Behandlung von durch Helicobacter Pylori oder andere spirale Urease-positive Gram-negative Bakterien verursachten Krankheiten
IL116249A (en) * 1994-12-12 2003-07-06 Pfizer Nk-1 receptor antagonists for the treatment of neuronal damage and stroke
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2728265A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p dans une composition pharmaceutique
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FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
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US8691825B2 (en) 2009-04-01 2014-04-08 Merck Sharp & Dohme Corp. Inhibitors of AKT activity
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BR112013028813B1 (pt) * 2011-08-27 2020-10-20 Wockhardt Limited derivados de 1,6-diazabiciclo[3,2,1]octan-7-ona e composições farmacêuticas que os compreendem
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US3506673A (en) * 1968-03-29 1970-04-14 Aldrich Chem Co Inc 2-(4'halo)-benzhydryl-3-quinuclidinols
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JP2514137B2 (ja) * 1990-07-23 1996-07-10 フアイザー・インコーポレイテツド キヌクリジン誘導体

Also Published As

Publication number Publication date
NO940927D0 (no) 1994-03-15
DK0607164T3 (da) 2002-06-17
ATE216996T1 (de) 2002-05-15
CN1071168A (zh) 1993-04-21
HU9400728D0 (en) 1994-06-28
PT100901A (pt) 1994-02-28
US5527808A (en) 1996-06-18
ES2174836T3 (es) 2002-11-16
JP2535134B2 (ja) 1996-09-18
EP0607164B1 (de) 2002-05-02
DE69232588D1 (de) 2002-06-06
ZA927370B (en) 1994-03-25
CZ59394A3 (en) 1994-11-16
BR9206500A (pt) 1995-10-03
JPH06507179A (ja) 1994-08-11
AU2481292A (en) 1993-04-27
MX9205242A (es) 1993-03-01
WO1993006099A1 (en) 1993-04-01
FI941212A0 (fi) 1994-03-15
FI941212A7 (fi) 1994-03-15
DE69232588T2 (de) 2002-08-22
CA2118704C (en) 1997-01-21
CA2118704A1 (en) 1993-04-01
FI941212L (fi) 1994-03-15
EP0607164A1 (de) 1994-07-27

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