NO933784L - Pyrazolo(4,3-c)pyridiner, en fremgangsmåte for fremstilling av dem og deres anvendelse som hemmere av reopptak av serotonin - Google Patents

Pyrazolo(4,3-c)pyridiner, en fremgangsmåte for fremstilling av dem og deres anvendelse som hemmere av reopptak av serotonin

Info

Publication number
NO933784L
NO933784L NO933784A NO933784A NO933784L NO 933784 L NO933784 L NO 933784L NO 933784 A NO933784 A NO 933784A NO 933784 A NO933784 A NO 933784A NO 933784 L NO933784 L NO 933784L
Authority
NO
Norway
Prior art keywords
loweralkyl
serotonin reuptake
chem
hydrogen
inhibitors
Prior art date
Application number
NO933784A
Other languages
English (en)
Other versions
NO933784D0 (no
NO300374B1 (no
Inventor
Gregory M Shutske
Kevin J Kapples
Iv John D Tomer
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of NO933784D0 publication Critical patent/NO933784D0/no
Publication of NO933784L publication Critical patent/NO933784L/no
Publication of NO300374B1 publication Critical patent/NO300374B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other Investigation Or Analysis Of Materials By Electrical Means (AREA)
  • Silver Salt Photography Or Processing Solution Therefor (AREA)
NO933784A 1992-10-22 1993-10-21 Pyrazolo£4,3-c|pyridiner, farmasöytiske sammensetninger inneholdende disse og deres anvendelse til fremstilling av hemmere av reopptak av serotonin NO300374B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/964,690 US5264576A (en) 1992-10-22 1992-10-22 Pyrazolo[4,3-c]pyridines which are intermediates

Publications (3)

Publication Number Publication Date
NO933784D0 NO933784D0 (no) 1993-10-21
NO933784L true NO933784L (no) 1994-04-25
NO300374B1 NO300374B1 (no) 1997-05-20

Family

ID=25508857

Family Applications (1)

Application Number Title Priority Date Filing Date
NO933784A NO300374B1 (no) 1992-10-22 1993-10-21 Pyrazolo£4,3-c|pyridiner, farmasöytiske sammensetninger inneholdende disse og deres anvendelse til fremstilling av hemmere av reopptak av serotonin

Country Status (18)

Country Link
US (4) US5264576A (no)
EP (1) EP0594001B1 (no)
JP (1) JP2656211B2 (no)
KR (1) KR100295026B1 (no)
CN (1) CN1049658C (no)
AT (1) ATE195522T1 (no)
AU (1) AU671305B2 (no)
CA (1) CA2108941A1 (no)
DE (1) DE69329231T2 (no)
DK (1) DK0594001T3 (no)
ES (1) ES2152237T3 (no)
FI (1) FI103890B (no)
GR (1) GR3034819T3 (no)
MX (1) MX9306552A (no)
NO (1) NO300374B1 (no)
NZ (1) NZ250003A (no)
PT (1) PT594001E (no)
TW (1) TW252114B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5300498A (en) * 1993-06-04 1994-04-05 Hoechst-Roussel Pharmaceuticals Incorporated 6-piperazinyl-1H-pyrazolo[3,4-b]pyridine-3-carboxylic acids, esters, amides and related compounds
US5618824A (en) * 1994-03-09 1997-04-08 Merrell Pharmaceuticals Inc. Treatment of obsessive-compulsive disorders with 5-HT2 antagonists
US5565413A (en) * 1994-12-06 1996-10-15 Zeneca Limited Substituted pyridyl phenyl ketone herbicides
US20070117785A1 (en) * 2000-08-14 2007-05-24 Butler Christopher R Substituted pyrazoles and methods of treatment with substituted pyrazoles
DE60118004T2 (de) 2000-08-14 2006-11-16 Ortho-Mcneil Pharmaceutical, Inc. Substituierte pyrazole
US7589202B2 (en) 2000-08-14 2009-09-15 Ortho Mcneil Pharmaceutical, Inc. Substituted pyrazoles
US20050101587A9 (en) * 2000-08-14 2005-05-12 Butler Christopher R. Method for treating allergies using substituted pyrazoles
US7332494B2 (en) 2000-08-14 2008-02-19 Janssen Pharmaceutica, N.V. Method for treating allergies using substituted pyrazoles
JP4911864B2 (ja) * 2000-08-14 2012-04-04 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド 置換ピラゾール
RU2003106192A (ru) 2000-09-06 2004-07-27 Орто-Макнейл Фармасьютикал, Инк. (Us) Способ лечения аллергий
WO2003101968A1 (fr) * 2002-05-31 2003-12-11 Eisai Co., Ltd. Compose de pyrazole et composition medicinale le contenant
EP2328895B1 (en) * 2008-09-16 2013-03-27 Proximagen Limited Pyrazolo[4,3-c]pyridine compounds and their use as inhibitors of SSAO
CN102558174B (zh) * 2011-08-23 2014-03-19 天津市斯芬克司药物研发有限公司 一种全新吡唑并[4,3-c]吡啶化合物的发明及其合成方法
JP6242885B2 (ja) 2012-06-27 2017-12-06 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ５−アザインダゾール化合物及び使用方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3994890A (en) * 1974-01-31 1976-11-30 Chugai Seiyaku Kabushiki Kaisha 1-Aminoalkyl, 3-phenyl indazoles
JPS5944314B2 (ja) * 1975-01-15 1984-10-29 中外製薬株式会社 インダゾ−ル誘導体の製法
JPS5936627B2 (ja) * 1975-07-25 1984-09-05 中外製薬株式会社 インダゾ−ル誘導体の製法
DK27383A (da) * 1982-02-17 1983-08-18 Lepetit Spa Fremgangsmaade til fremstilling af pyrazol(4,3-c)pyridiner
JPH0615542B2 (ja) * 1986-07-22 1994-03-02 吉富製薬株式会社 ピラゾロピリジン化合物
EP0338087A4 (en) * 1987-10-13 1991-07-24 Yoshitomi Pharmaceutical Industries, Ltd. Fused pyrazole compounds, process for their preparation, and their medicinal use
DK181190D0 (da) * 1990-07-30 1990-07-30 Lundbeck & Co As H 3-aryl-indol- eller 3-aryl-indazolderivater
EP0494774A1 (en) * 1991-01-11 1992-07-15 MERCK SHARP & DOHME LTD. Indazole-substituted fivemembered heteroaromatic compounds
GB9216783D0 (en) * 1992-08-07 1992-09-23 Ici Plc Heterocyclic derivatives
US5300478A (en) * 1993-01-28 1994-04-05 Zeneca Limited Substituted fused pyrazolo compounds

Also Published As

Publication number Publication date
FI934621A0 (fi) 1993-10-20
NO933784D0 (no) 1993-10-21
CA2108941A1 (en) 1994-04-23
US5296491A (en) 1994-03-22
FI934621A (fi) 1994-04-23
TW252114B (no) 1995-07-21
PT594001E (pt) 2001-01-31
US5428169A (en) 1995-06-27
MX9306552A (es) 1994-06-30
AU4912893A (en) 1994-05-05
NZ250003A (en) 1996-03-26
FI103890B1 (fi) 1999-10-15
CN1049658C (zh) 2000-02-23
FI103890B (fi) 1999-10-15
EP0594001B1 (en) 2000-08-16
ES2152237T3 (es) 2001-02-01
US5264576A (en) 1993-11-23
US5380847A (en) 1995-01-10
AU671305B2 (en) 1996-08-22
JPH06192257A (ja) 1994-07-12
DK0594001T3 (da) 2000-10-30
DE69329231D1 (de) 2000-09-21
GR3034819T3 (en) 2001-02-28
JP2656211B2 (ja) 1997-09-24
KR940009185A (ko) 1994-05-20
NO300374B1 (no) 1997-05-20
KR100295026B1 (ko) 2001-09-17
CN1099033A (zh) 1995-02-22
ATE195522T1 (de) 2000-09-15
DE69329231T2 (de) 2001-03-29
EP0594001A1 (en) 1994-04-27

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Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees

Free format text: LAPSED IN APRIL 2001