MX9306552A - Pirazolo[4,3-c]piridinas, procedimiento para su preparacion y su utilizacion como inhibidores de la reabsorcion de serotonina. - Google Patents

Pirazolo[4,3-c]piridinas, procedimiento para su preparacion y su utilizacion como inhibidores de la reabsorcion de serotonina.

Info

Publication number
MX9306552A
MX9306552A MX9306552A MX9306552A MX9306552A MX 9306552 A MX9306552 A MX 9306552A MX 9306552 A MX9306552 A MX 9306552A MX 9306552 A MX9306552 A MX 9306552A MX 9306552 A MX9306552 A MX 9306552A
Authority
MX
Mexico
Prior art keywords
loweralkyl
piridines
pirazolo
procedure
preparation
Prior art date
Application number
MX9306552A
Other languages
English (en)
Inventor
Gregory Shutske
Kevin J Kapples
John Dick Tomer
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of MX9306552A publication Critical patent/MX9306552A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Silver Salt Photography Or Processing Solution Therefor (AREA)
  • Other Investigation Or Analysis Of Materials By Electrical Means (AREA)

Abstract

Este invento se refiere a un procedimiento para preparar compuestos y a composiciones farmacéuticas, así como a su uso como inhibidores de la reabsorción de serotonina.
MX9306552A 1992-10-22 1993-10-21 Pirazolo[4,3-c]piridinas, procedimiento para su preparacion y su utilizacion como inhibidores de la reabsorcion de serotonina. MX9306552A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/964,690 US5264576A (en) 1992-10-22 1992-10-22 Pyrazolo[4,3-c]pyridines which are intermediates

Publications (1)

Publication Number Publication Date
MX9306552A true MX9306552A (es) 1994-06-30

Family

ID=25508857

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9306552A MX9306552A (es) 1992-10-22 1993-10-21 Pirazolo[4,3-c]piridinas, procedimiento para su preparacion y su utilizacion como inhibidores de la reabsorcion de serotonina.

Country Status (18)

Country Link
US (4) US5264576A (es)
EP (1) EP0594001B1 (es)
JP (1) JP2656211B2 (es)
KR (1) KR100295026B1 (es)
CN (1) CN1049658C (es)
AT (1) ATE195522T1 (es)
AU (1) AU671305B2 (es)
CA (1) CA2108941A1 (es)
DE (1) DE69329231T2 (es)
DK (1) DK0594001T3 (es)
ES (1) ES2152237T3 (es)
FI (1) FI103890B1 (es)
GR (1) GR3034819T3 (es)
MX (1) MX9306552A (es)
NO (1) NO300374B1 (es)
NZ (1) NZ250003A (es)
PT (1) PT594001E (es)
TW (1) TW252114B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5300498A (en) * 1993-06-04 1994-04-05 Hoechst-Roussel Pharmaceuticals Incorporated 6-piperazinyl-1H-pyrazolo[3,4-b]pyridine-3-carboxylic acids, esters, amides and related compounds
US5618824A (en) * 1994-03-09 1997-04-08 Merrell Pharmaceuticals Inc. Treatment of obsessive-compulsive disorders with 5-HT2 antagonists
US5565413A (en) * 1994-12-06 1996-10-15 Zeneca Limited Substituted pyridyl phenyl ketone herbicides
US6635633B2 (en) 2000-08-14 2003-10-21 Ortho-Pharmaceutical, Inc. Substituted pyrazoles
RU2317988C2 (ru) 2000-08-14 2008-02-27 Орто-Макнейл Фармасьютикал, Инк. Замещенные пиразолы, фармацевтическая композиция на их основе, применение фармацевтической композиции и способ ингибирования активности катепсина s
US7332494B2 (en) 2000-08-14 2008-02-19 Janssen Pharmaceutica, N.V. Method for treating allergies using substituted pyrazoles
AU2001281255B2 (en) 2000-08-14 2006-07-20 Ortho-Mcneil Pharmaceutical, Inc. Substituted pyrazoles
US20050101587A9 (en) * 2000-08-14 2005-05-12 Butler Christopher R. Method for treating allergies using substituted pyrazoles
US20070117785A1 (en) * 2000-08-14 2007-05-24 Butler Christopher R Substituted pyrazoles and methods of treatment with substituted pyrazoles
WO2002020002A2 (en) 2000-09-06 2002-03-14 Ortho Mcneil Pharmaceutical, Inc. A method for treating allergies
EP1510516A4 (en) * 2002-05-31 2005-11-02 Eisai Co Ltd PYRAZOL COMPOUND AND MEDICAL COMPOSITION CONTAINING THEM
EP2328895B1 (en) * 2008-09-16 2013-03-27 Proximagen Limited Pyrazolo[4,3-c]pyridine compounds and their use as inhibitors of SSAO
CN102558174B (zh) * 2011-08-23 2014-03-19 天津市斯芬克司药物研发有限公司 一种全新吡唑并[4,3-c]吡啶化合物的发明及其合成方法
MX2014014828A (es) 2012-06-27 2015-02-12 Hoffmann La Roche Compuestos de 5-azaindazol y metodos de uso.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3994890A (en) * 1974-01-31 1976-11-30 Chugai Seiyaku Kabushiki Kaisha 1-Aminoalkyl, 3-phenyl indazoles
JPS5944314B2 (ja) * 1975-01-15 1984-10-29 中外製薬株式会社 インダゾ−ル誘導体の製法
JPS5936627B2 (ja) * 1975-07-25 1984-09-05 中外製薬株式会社 インダゾ−ル誘導体の製法
DK27383A (da) * 1982-02-17 1983-08-18 Lepetit Spa Fremgangsmaade til fremstilling af pyrazol(4,3-c)pyridiner
JPH0615542B2 (ja) * 1986-07-22 1994-03-02 吉富製薬株式会社 ピラゾロピリジン化合物
EP0338087A4 (en) * 1987-10-13 1991-07-24 Yoshitomi Pharmaceutical Industries, Ltd. Fused pyrazole compounds, process for their preparation, and their medicinal use
DK181190D0 (da) * 1990-07-30 1990-07-30 Lundbeck & Co As H 3-aryl-indol- eller 3-aryl-indazolderivater
EP0494774A1 (en) * 1991-01-11 1992-07-15 MERCK SHARP & DOHME LTD. Indazole-substituted fivemembered heteroaromatic compounds
GB9216783D0 (en) * 1992-08-07 1992-09-23 Ici Plc Heterocyclic derivatives
US5300478A (en) * 1993-01-28 1994-04-05 Zeneca Limited Substituted fused pyrazolo compounds

Also Published As

Publication number Publication date
DE69329231D1 (de) 2000-09-21
DK0594001T3 (da) 2000-10-30
FI934621A0 (fi) 1993-10-20
KR100295026B1 (ko) 2001-09-17
US5428169A (en) 1995-06-27
ATE195522T1 (de) 2000-09-15
FI103890B (fi) 1999-10-15
US5296491A (en) 1994-03-22
EP0594001B1 (en) 2000-08-16
ES2152237T3 (es) 2001-02-01
EP0594001A1 (en) 1994-04-27
US5380847A (en) 1995-01-10
CN1049658C (zh) 2000-02-23
FI103890B1 (fi) 1999-10-15
AU4912893A (en) 1994-05-05
JPH06192257A (ja) 1994-07-12
FI934621A (fi) 1994-04-23
TW252114B (es) 1995-07-21
US5264576A (en) 1993-11-23
CA2108941A1 (en) 1994-04-23
CN1099033A (zh) 1995-02-22
NZ250003A (en) 1996-03-26
AU671305B2 (en) 1996-08-22
NO933784D0 (no) 1993-10-21
NO933784L (no) 1994-04-25
KR940009185A (ko) 1994-05-20
JP2656211B2 (ja) 1997-09-24
DE69329231T2 (de) 2001-03-29
GR3034819T3 (en) 2001-02-28
NO300374B1 (no) 1997-05-20
PT594001E (pt) 2001-01-31

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Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees