NO863608L - Fremgangsmaate for fremstilling av benzimidazolderivater. - Google Patents

Fremgangsmaate for fremstilling av benzimidazolderivater.

Info

Publication number
NO863608L
NO863608L NO863608A NO863608A NO863608L NO 863608 L NO863608 L NO 863608L NO 863608 A NO863608 A NO 863608A NO 863608 A NO863608 A NO 863608A NO 863608 L NO863608 L NO 863608L
Authority
NO
Norway
Prior art keywords
preparing
procedure
benzimidazold
derivatives
benzimidazold derivatives
Prior art date
Application number
NO863608A
Other languages
English (en)
Other versions
NO863608D0 (no
NO167026C (no
NO167026B (no
Inventor
Philippe Manoury
Jean Binet
Gerard Defosse
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO863608D0 publication Critical patent/NO863608D0/no
Publication of NO863608L publication Critical patent/NO863608L/no
Publication of NO167026B publication Critical patent/NO167026B/no
Publication of NO167026C publication Critical patent/NO167026C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO863608A 1985-09-11 1986-09-10 Analogifremgangsmaate for fremstilling av terapeutisk aktive benzimidazolderivater NO167026C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8513453A FR2587029B1 (fr) 1985-09-11 1985-09-11 Derives de benzimidazole, leur preparation et leur application en therapeutique

Publications (4)

Publication Number Publication Date
NO863608D0 NO863608D0 (no) 1986-09-10
NO863608L true NO863608L (no) 1987-03-12
NO167026B NO167026B (no) 1991-06-17
NO167026C NO167026C (no) 1991-09-25

Family

ID=9322797

Family Applications (2)

Application Number Title Priority Date Filing Date
NO863608A NO167026C (no) 1985-09-11 1986-09-10 Analogifremgangsmaate for fremstilling av terapeutisk aktive benzimidazolderivater
NO2001017C NO2001017I1 (no) 1985-09-11 2001-10-15 Mizolastine

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2001017C NO2001017I1 (no) 1985-09-11 2001-10-15 Mizolastine

Country Status (25)

Country Link
US (2) US4820710A (no)
EP (1) EP0217700B1 (no)
JP (1) JPS6261979A (no)
KR (1) KR930001411B1 (no)
AR (1) AR243187A1 (no)
AT (1) ATE103603T1 (no)
AU (1) AU582894B2 (no)
CA (1) CA1272486A (no)
CS (1) CS357991A3 (no)
DE (2) DE3689748T2 (no)
DK (1) DK170594B1 (no)
ES (1) ES2001782A6 (no)
FI (1) FI87210C (no)
FR (1) FR2587029B1 (no)
GR (1) GR862318B (no)
HK (1) HK1005592A1 (no)
HU (1) HU196597B (no)
IE (1) IE61607B1 (no)
IL (1) IL79992A (no)
LU (1) LU90085I2 (no)
NL (1) NL970029I2 (no)
NO (2) NO167026C (no)
NZ (1) NZ217537A (no)
PT (1) PT83355B (no)
ZA (1) ZA866901B (no)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2618435B1 (fr) * 1987-07-23 1989-10-27 Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique
FR2637595B1 (fr) * 1988-10-11 1990-11-30 Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique
JPH02294758A (ja) * 1989-05-09 1990-12-05 Nec Corp 計算機使用時間管理方式
FR2658823B1 (fr) * 1990-02-27 1992-04-30 Adir Nouveaux derives d'aminomethylpiperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent .
FR2666582B1 (fr) * 1990-09-07 1994-09-02 Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique.
FR2693194B1 (fr) * 1992-07-03 1994-09-23 Synthelabo Dérivés d'alcanecarboxamide, leur préparation et leur application thérapeutique.
FR2745500B1 (fr) * 1996-03-04 1998-04-03 Synthelabo Formulations pharmaceutiques a liberation prolongee contenant de la mizolastine
JPH10101564A (ja) * 1996-09-27 1998-04-21 Mitsubishi Chem Corp 鼻炎予防及び／又は治療剤
CA2281927C (en) 1997-02-25 2004-01-27 Christopher J. Michejda Substituted benzimidazoles as non-nucleoside inhibitors of reverse transcriptase
FR2762214B1 (fr) * 1997-04-17 2000-10-06 Synthelabo Utilisation de la mizolastine pour la preparation d'un medicament destine au traitement de l'inflammation
EP0958820A1 (en) * 1998-05-19 1999-11-24 Sanofi-Synthelabo Use of an imidazol derivative for the manufacture of a medicament for treating auto-immunodiseases
ES2208098B1 (es) * 2002-10-02 2005-10-16 Ragactives, S.L. Procedimiento e intermedios para la obtencion de derivados de 1-(1h-bencimidazol-2-il)-4-(2-aminopirimidin) piperidina.
AR045955A1 (es) * 2003-09-30 2005-11-16 Janssen Pharmaceutica Nv Compuestos benzoimidazolicos
ES2245227B1 (es) * 2004-04-06 2007-03-01 Ragactives, S.L. Formas cristalinas de mizolastina, procedimientos para su obtencion y composiciones farmaceuticas que las contienen.
US8686009B2 (en) * 2009-06-25 2014-04-01 Alkermes Pharma Ireland Limited Prodrugs of NH-acidic compounds
AU2010266018B2 (en) 2009-06-25 2014-01-09 Alkermes Pharma Ireland Limited Heterocyclic compounds for the treatment of neurological and psychological disorders
CN102140076A (zh) * 2010-02-03 2011-08-03 辽宁本源制药有限公司 咪唑斯汀中间体的制备
WO2013088255A1 (en) 2011-12-15 2013-06-20 Alkermes Pharma Ireland Limited Prodrugs of secondary amine compounds
WO2019173230A1 (en) 2018-03-05 2019-09-12 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
JP7227398B2 (ja) * 2019-04-11 2023-02-21 帝人ファーマ株式会社 ベンズイミダゾール誘導体及びその使用
WO2023107705A1 (en) 2021-12-10 2023-06-15 Incyte Corporation Bicyclic amines as cdk12 inhibitors
CN116655596A (zh) * 2022-02-17 2023-08-29 济南同路医药科技发展有限公司 一种大粒径咪唑斯汀原料药制备方法
CN119707917B (zh) * 2024-12-24 2025-12-09 沈阳三九药业有限公司 一种咪唑斯汀中间体的制备方法
CN120441547B (zh) * 2025-05-06 2026-01-27 大连医科大学附属第二医院 一种脂肪酸酰胺水解酶（faah）抑制剂及其在疾病治疗中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4281005A (en) * 1979-03-05 1981-07-28 Merck & Co., Inc. Novel 2-pyridylimidazole compounds
US4556660A (en) * 1982-07-12 1985-12-03 Janssen Pharmaceutica N.V. N-(Bicyclic heterocyclyl)-4-piperidinamines
DE3484096D1 (de) * 1983-11-30 1991-03-14 Janssen Pharmaceutica Nv Bizyklisches heterozyklyl aufveisende n-(bizyklisches heterozyklyl-4-piperidinamine.
PH23995A (en) * 1984-01-09 1990-02-09 Janssen Pharmaceutica Nv 4((bicycle heterocyclyl)-methyl and hetero)piperidines
US4588722A (en) * 1984-01-09 1986-05-13 Janssen Pharmaceutica N.V. N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives

Also Published As

Publication number Publication date
ZA866901B (en) 1987-04-29
US4912219A (en) 1990-03-27
FI87210B (fi) 1992-08-31
IL79992A0 (en) 1986-12-31
KR930001411B1 (ko) 1993-02-27
DK170594B1 (da) 1995-11-06
NO2001017I1 (no) 2001-11-05
FI863661A0 (fi) 1986-09-10
JPH0460596B2 (no) 1992-09-28
AU582894B2 (en) 1989-04-13
EP0217700A1 (fr) 1987-04-08
DK431586D0 (da) 1986-09-10
HK1005592A1 (en) 1999-01-15
LU90085I2 (fr) 1997-09-25
FR2587029A1 (fr) 1987-03-13
KR870003100A (ko) 1987-04-15
ATE103603T1 (de) 1994-04-15
PT83355A (fr) 1986-10-01
DE19775081I2 (de) 2002-08-29
FR2587029B1 (fr) 1987-10-30
DE3689748D1 (de) 1994-05-05
ES2001782A6 (es) 1988-06-16
FI87210C (fi) 1992-12-10
IL79992A (en) 1990-07-12
FI863661L (fi) 1987-03-12
DE3689748T2 (de) 1994-08-11
CA1272486A (en) 1990-08-07
NO863608D0 (no) 1986-09-10
CS357991A3 (en) 1992-06-17
US4820710A (en) 1989-04-11
PT83355B (pt) 1989-05-12
NO167026C (no) 1991-09-25
AR243187A1 (es) 1993-07-30
GR862318B (en) 1987-01-19
IE61607B1 (en) 1994-11-16
JPS6261979A (ja) 1987-03-18
NL970029I2 (nl) 1998-04-01
HUT41771A (en) 1987-05-28
NZ217537A (en) 1988-11-29
DK431586A (da) 1987-03-12
AU6255286A (en) 1987-03-12
IE862416L (en) 1987-03-11
HU196597B (en) 1988-12-28
NL970029I1 (nl) 1997-10-01
NO167026B (no) 1991-06-17
EP0217700B1 (fr) 1994-03-30

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