NO802834L - PROCEDURE FOR THE PREPARATION OF 2-AMINO-3-BENZOYL-PHENYL ACETAMIDES - Google Patents
PROCEDURE FOR THE PREPARATION OF 2-AMINO-3-BENZOYL-PHENYL ACETAMIDESInfo
- Publication number
- NO802834L NO802834L NO802834A NO802834A NO802834L NO 802834 L NO802834 L NO 802834L NO 802834 A NO802834 A NO 802834A NO 802834 A NO802834 A NO 802834A NO 802834 L NO802834 L NO 802834L
- Authority
- NO
- Norway
- Prior art keywords
- benzoyl
- amino
- procedure
- preparation
- phenyl acetamides
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US7886079A | 1979-09-26 | 1979-09-26 |
Publications (3)
Publication Number | Publication Date |
---|---|
NO802834L true NO802834L (en) | 1981-03-27 |
NO152128B NO152128B (en) | 1985-04-29 |
NO152128C NO152128C (en) | 1985-08-07 |
Family
ID=22146633
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO802834A NO152128C (en) | 1979-09-26 | 1980-09-25 | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES |
Country Status (36)
Country | Link |
---|---|
JP (1) | JPS5657751A (en) |
KR (1) | KR840000763B1 (en) |
AT (1) | AT374170B (en) |
AU (1) | AU532359B2 (en) |
BE (1) | BE885393A (en) |
BR (1) | BR8006042A (en) |
CA (1) | CA1128512A (en) |
CH (1) | CH646138A5 (en) |
CS (1) | CS227012B2 (en) |
DE (1) | DE3035688A1 (en) |
DK (1) | DK154136C (en) |
EG (1) | EG15020A (en) |
ES (2) | ES495329A0 (en) |
FI (1) | FI72967C (en) |
FR (1) | FR2465710A1 (en) |
GB (1) | GB2059963B (en) |
GR (1) | GR70049B (en) |
HK (1) | HK59383A (en) |
HU (1) | HU183215B (en) |
IE (1) | IE50268B1 (en) |
IL (1) | IL60999A (en) |
IN (3) | IN151313B (en) |
IT (1) | IT1133823B (en) |
KE (1) | KE3307A (en) |
LU (1) | LU82797A1 (en) |
MX (1) | MX7159E (en) |
NL (1) | NL8005346A (en) |
NO (1) | NO152128C (en) |
NZ (1) | NZ195061A (en) |
PH (1) | PH22628A (en) |
PL (1) | PL128998B1 (en) |
PT (1) | PT71839B (en) |
SE (1) | SE448626B (en) |
SG (1) | SG42983G (en) |
YU (3) | YU41734B (en) |
ZA (1) | ZA805476B (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL61945A (en) * | 1980-02-19 | 1984-09-30 | Robins Co Inc A H | 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them |
US6646001B2 (en) | 1997-12-19 | 2003-11-11 | Alcon Manufacturing, Ltd. | Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension |
US6066671A (en) * | 1997-12-19 | 2000-05-23 | Alcon Laboratories, Inc. | Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides |
GB9727523D0 (en) * | 1997-12-31 | 1998-02-25 | Pharmacia & Upjohn Spa | Alpha-aminoamide derivatives useful as analgesic agents |
AR030345A1 (en) * | 2000-08-14 | 2003-08-20 | Alcon Inc | METHOD OF TREATMENT OF DISORDERS RELATED TO ANGIOGENESIS |
PT1423168E (en) | 2001-09-03 | 2006-05-31 | Newron Pharm Spa | PHARMACEUTICAL COMPOSITION WHICH UNDERSTAND GABAPENTINE OR ITS ANALOGUE AND AN X-AMINOAMIDE AND ITS USE AS ANALGESIC |
EP1438956A1 (en) | 2003-01-16 | 2004-07-21 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful as antimigraine agents |
CZ301776B6 (en) * | 2009-06-08 | 2010-06-16 | Farmak, A.S. | Process for preparing 2-amino-3-benzoylphenylacetamide (nepafenac) with minimum by-products |
CN112794809B (en) * | 2019-11-14 | 2023-12-29 | 南京济群医药科技股份有限公司 | Preparation method of high-purity nepafenac intermediate |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1226344A (en) * | 1967-07-31 | 1971-03-24 | ||
SE400966B (en) * | 1975-08-13 | 1978-04-17 | Robins Co Inc A H | PROCEDURE FOR PREPARING 2-AMINO-3- (OR 5-) BENZOYL-PHENYLETIC ACIDS |
IL61945A (en) * | 1980-02-19 | 1984-09-30 | Robins Co Inc A H | 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them |
-
1980
- 1980-09-04 ZA ZA00805476A patent/ZA805476B/en unknown
- 1980-09-08 IL IL60999A patent/IL60999A/en unknown
- 1980-09-08 AU AU62116/80A patent/AU532359B2/en not_active Ceased
- 1980-09-11 CS CS806196A patent/CS227012B2/en unknown
- 1980-09-17 IE IE1946/80A patent/IE50268B1/en unknown
- 1980-09-20 EG EG80573A patent/EG15020A/en active
- 1980-09-22 GR GR62936A patent/GR70049B/el unknown
- 1980-09-22 DE DE19803035688 patent/DE3035688A1/en active Granted
- 1980-09-22 BR BR8006042A patent/BR8006042A/en unknown
- 1980-09-23 AT AT0474580A patent/AT374170B/en not_active IP Right Cessation
- 1980-09-23 PH PH24613A patent/PH22628A/en unknown
- 1980-09-24 LU LU82797A patent/LU82797A1/en unknown
- 1980-09-24 FI FI803002A patent/FI72967C/en not_active IP Right Cessation
- 1980-09-24 SE SE8006668A patent/SE448626B/en not_active IP Right Cessation
- 1980-09-25 GB GB8030955A patent/GB2059963B/en not_active Expired
- 1980-09-25 YU YU2450/80A patent/YU41734B/en unknown
- 1980-09-25 KR KR1019800003740A patent/KR840000763B1/en active
- 1980-09-25 CA CA361,068A patent/CA1128512A/en not_active Expired
- 1980-09-25 PL PL1980226919A patent/PL128998B1/en unknown
- 1980-09-25 PT PT71839A patent/PT71839B/en unknown
- 1980-09-25 DK DK405780A patent/DK154136C/en not_active IP Right Cessation
- 1980-09-25 HU HU802347A patent/HU183215B/en not_active IP Right Cessation
- 1980-09-25 ES ES495329A patent/ES495329A0/en active Granted
- 1980-09-25 NO NO802834A patent/NO152128C/en unknown
- 1980-09-25 NL NL8005346A patent/NL8005346A/en not_active Application Discontinuation
- 1980-09-25 FR FR8020596A patent/FR2465710A1/en active Granted
- 1980-09-25 MX MX809050U patent/MX7159E/en unknown
- 1980-09-25 BE BE0/202226A patent/BE885393A/en not_active IP Right Cessation
- 1980-09-25 CH CH719180A patent/CH646138A5/en not_active IP Right Cessation
- 1980-09-26 IT IT24948/80A patent/IT1133823B/en active
- 1980-09-26 NZ NZ195061A patent/NZ195061A/en unknown
- 1980-09-26 IN IN1092/CAL/80A patent/IN151313B/en unknown
- 1980-09-26 JP JP13415280A patent/JPS5657751A/en active Granted
-
1981
- 1981-06-12 ES ES503019A patent/ES503019A0/en active Granted
-
1982
- 1982-12-30 IN IN1509/CAL/82A patent/IN156255B/en unknown
- 1982-12-30 IN IN1508/CAL/82A patent/IN156254B/en unknown
-
1983
- 1983-03-28 YU YU731/83A patent/YU43306B/en unknown
- 1983-03-28 YU YU730/83A patent/YU43305B/en unknown
- 1983-07-19 SG SG42983A patent/SG42983G/en unknown
- 1983-07-21 KE KE3307A patent/KE3307A/en unknown
- 1983-11-24 HK HK593/83A patent/HK59383A/en unknown
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