AT374170B - METHOD FOR PRODUCING NEW 2-AMINO-3 -BENZOYL-PHENYL ACETAMIDE DERIVATIVES - Google Patents
METHOD FOR PRODUCING NEW 2-AMINO-3 -BENZOYL-PHENYL ACETAMIDE DERIVATIVESInfo
- Publication number
- AT374170B AT374170B AT0474580A AT474580A AT374170B AT 374170 B AT374170 B AT 374170B AT 0474580 A AT0474580 A AT 0474580A AT 474580 A AT474580 A AT 474580A AT 374170 B AT374170 B AT 374170B
- Authority
- AT
- Austria
- Prior art keywords
- benzoyl
- amino
- producing new
- phenyl acetamide
- acetamide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AT538481A AT379740B (en) | 1979-09-26 | 1981-12-16 | METHOD FOR REDUCING INFLAMMATION AND PAIN OR FOR INHIBITING THE THROMBOZYTE AGGREGATION IN A LIVING ANIMAL BODY |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US7886079A | 1979-09-26 | 1979-09-26 |
Publications (2)
Publication Number | Publication Date |
---|---|
ATA474580A ATA474580A (en) | 1983-08-15 |
AT374170B true AT374170B (en) | 1984-03-26 |
Family
ID=22146633
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT0474580A AT374170B (en) | 1979-09-26 | 1980-09-23 | METHOD FOR PRODUCING NEW 2-AMINO-3 -BENZOYL-PHENYL ACETAMIDE DERIVATIVES |
Country Status (36)
Country | Link |
---|---|
JP (1) | JPS5657751A (en) |
KR (1) | KR840000763B1 (en) |
AT (1) | AT374170B (en) |
AU (1) | AU532359B2 (en) |
BE (1) | BE885393A (en) |
BR (1) | BR8006042A (en) |
CA (1) | CA1128512A (en) |
CH (1) | CH646138A5 (en) |
CS (1) | CS227012B2 (en) |
DE (1) | DE3035688A1 (en) |
DK (1) | DK154136C (en) |
EG (1) | EG15020A (en) |
ES (2) | ES8200329A1 (en) |
FI (1) | FI72967C (en) |
FR (1) | FR2465710A1 (en) |
GB (1) | GB2059963B (en) |
GR (1) | GR70049B (en) |
HK (1) | HK59383A (en) |
HU (1) | HU183215B (en) |
IE (1) | IE50268B1 (en) |
IL (1) | IL60999A (en) |
IN (3) | IN151313B (en) |
IT (1) | IT1133823B (en) |
KE (1) | KE3307A (en) |
LU (1) | LU82797A1 (en) |
MX (1) | MX7159E (en) |
NL (1) | NL8005346A (en) |
NO (1) | NO152128C (en) |
NZ (1) | NZ195061A (en) |
PH (1) | PH22628A (en) |
PL (1) | PL128998B1 (en) |
PT (1) | PT71839B (en) |
SE (1) | SE448626B (en) |
SG (1) | SG42983G (en) |
YU (3) | YU41734B (en) |
ZA (1) | ZA805476B (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL61945A (en) * | 1980-02-19 | 1984-09-30 | Robins Co Inc A H | 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them |
US6066671A (en) * | 1997-12-19 | 2000-05-23 | Alcon Laboratories, Inc. | Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides |
US6646001B2 (en) | 1997-12-19 | 2003-11-11 | Alcon Manufacturing, Ltd. | Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension |
GB9727523D0 (en) * | 1997-12-31 | 1998-02-25 | Pharmacia & Upjohn Spa | Alpha-aminoamide derivatives useful as analgesic agents |
AR030345A1 (en) * | 2000-08-14 | 2003-08-20 | Alcon Inc | METHOD OF TREATMENT OF DISORDERS RELATED TO ANGIOGENESIS |
MXPA04002009A (en) | 2001-09-03 | 2004-07-08 | Newron Pharm Spa | Pharmaceutical composition comprising gabapentin or an analogue thereof and an $g(a)-aminoamide and its analgesic use. |
EP1438956A1 (en) | 2003-01-16 | 2004-07-21 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful as antimigraine agents |
CZ2009367A3 (en) * | 2009-06-08 | 2010-06-16 | Farmak, A.S. | Process for preparing 2-amino-3-benzoylphenylacetamide (nepafenac) with minimum of by-products |
CN112794809B (en) * | 2019-11-14 | 2023-12-29 | 南京济群医药科技股份有限公司 | Preparation method of high-purity nepafenac intermediate |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1226344A (en) * | 1967-07-31 | 1971-03-24 | ||
SE400966B (en) * | 1975-08-13 | 1978-04-17 | Robins Co Inc A H | PROCEDURE FOR PREPARING 2-AMINO-3- (OR 5-) BENZOYL-PHENYLETIC ACIDS |
IL61945A (en) * | 1980-02-19 | 1984-09-30 | Robins Co Inc A H | 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them |
-
1980
- 1980-09-04 ZA ZA00805476A patent/ZA805476B/en unknown
- 1980-09-08 AU AU62116/80A patent/AU532359B2/en not_active Ceased
- 1980-09-08 IL IL60999A patent/IL60999A/en unknown
- 1980-09-11 CS CS806196A patent/CS227012B2/en unknown
- 1980-09-17 IE IE1946/80A patent/IE50268B1/en unknown
- 1980-09-20 EG EG80573A patent/EG15020A/en active
- 1980-09-22 GR GR62936A patent/GR70049B/el unknown
- 1980-09-22 BR BR8006042A patent/BR8006042A/en unknown
- 1980-09-22 DE DE19803035688 patent/DE3035688A1/en active Granted
- 1980-09-23 AT AT0474580A patent/AT374170B/en not_active IP Right Cessation
- 1980-09-23 PH PH24613A patent/PH22628A/en unknown
- 1980-09-24 LU LU82797A patent/LU82797A1/en unknown
- 1980-09-24 FI FI803002A patent/FI72967C/en not_active IP Right Cessation
- 1980-09-24 SE SE8006668A patent/SE448626B/en not_active IP Right Cessation
- 1980-09-25 PL PL1980226919A patent/PL128998B1/en unknown
- 1980-09-25 HU HU802347A patent/HU183215B/en not_active IP Right Cessation
- 1980-09-25 NO NO802834A patent/NO152128C/en unknown
- 1980-09-25 KR KR1019800003740A patent/KR840000763B1/en active
- 1980-09-25 YU YU2450/80A patent/YU41734B/en unknown
- 1980-09-25 CH CH719180A patent/CH646138A5/en not_active IP Right Cessation
- 1980-09-25 FR FR8020596A patent/FR2465710A1/en active Granted
- 1980-09-25 GB GB8030955A patent/GB2059963B/en not_active Expired
- 1980-09-25 NL NL8005346A patent/NL8005346A/en not_active Application Discontinuation
- 1980-09-25 MX MX809050U patent/MX7159E/en unknown
- 1980-09-25 PT PT71839A patent/PT71839B/en unknown
- 1980-09-25 DK DK405780A patent/DK154136C/en not_active IP Right Cessation
- 1980-09-25 ES ES495329A patent/ES8200329A1/en not_active Expired
- 1980-09-25 BE BE0/202226A patent/BE885393A/en not_active IP Right Cessation
- 1980-09-25 CA CA361,068A patent/CA1128512A/en not_active Expired
- 1980-09-26 NZ NZ195061A patent/NZ195061A/en unknown
- 1980-09-26 IT IT24948/80A patent/IT1133823B/en active
- 1980-09-26 JP JP13415280A patent/JPS5657751A/en active Granted
- 1980-09-26 IN IN1092/CAL/80A patent/IN151313B/en unknown
-
1981
- 1981-06-12 ES ES503019A patent/ES8204715A1/en not_active Expired
-
1982
- 1982-12-30 IN IN1509/CAL/82A patent/IN156255B/en unknown
- 1982-12-30 IN IN1508/CAL/82A patent/IN156254B/en unknown
-
1983
- 1983-03-28 YU YU731/83A patent/YU43306B/en unknown
- 1983-03-28 YU YU730/83A patent/YU43305B/en unknown
- 1983-07-19 SG SG42983A patent/SG42983G/en unknown
- 1983-07-21 KE KE3307A patent/KE3307A/en unknown
- 1983-11-24 HK HK593/83A patent/HK59383A/en unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ELJ | Ceased due to non-payment of the annual fee |