MX7159E - PROCEDURE FOR THE PREPARATION OF 2-AMINO-3-BENZOIL PHENYLACETAMIDES AND CYCLIC APPROVALS - Google Patents

PROCEDURE FOR THE PREPARATION OF 2-AMINO-3-BENZOIL PHENYLACETAMIDES AND CYCLIC APPROVALS

Info

Publication number
MX7159E
MX7159E MX809050U MX905080U MX7159E MX 7159 E MX7159 E MX 7159E MX 809050 U MX809050 U MX 809050U MX 905080 U MX905080 U MX 905080U MX 7159 E MX7159 E MX 7159E
Authority
MX
Mexico
Prior art keywords
phenylacetamides
benzoil
approvals
cyclic
amino
Prior art date
Application number
MX809050U
Other languages
Spanish (es)
Inventor
James Robert Shanklin Jr
Dwight Allen Shamblee
David Allan Walsh
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of MX7159E publication Critical patent/MX7159E/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182Radicals derived from carboxylic acids
    • C07D295/185Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX809050U 1979-09-26 1980-09-25 PROCEDURE FOR THE PREPARATION OF 2-AMINO-3-BENZOIL PHENYLACETAMIDES AND CYCLIC APPROVALS MX7159E (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7886079A 1979-09-26 1979-09-26

Publications (1)

Publication Number Publication Date
MX7159E true MX7159E (en) 1987-12-02

Family

ID=22146633

Family Applications (1)

Application Number Title Priority Date Filing Date
MX809050U MX7159E (en) 1979-09-26 1980-09-25 PROCEDURE FOR THE PREPARATION OF 2-AMINO-3-BENZOIL PHENYLACETAMIDES AND CYCLIC APPROVALS

Country Status (36)

Country Link
JP (1) JPS5657751A (en)
KR (1) KR840000763B1 (en)
AT (1) AT374170B (en)
AU (1) AU532359B2 (en)
BE (1) BE885393A (en)
BR (1) BR8006042A (en)
CA (1) CA1128512A (en)
CH (1) CH646138A5 (en)
CS (1) CS227012B2 (en)
DE (1) DE3035688A1 (en)
DK (1) DK154136C (en)
EG (1) EG15020A (en)
ES (2) ES8200329A1 (en)
FI (1) FI72967C (en)
FR (1) FR2465710A1 (en)
GB (1) GB2059963B (en)
GR (1) GR70049B (en)
HK (1) HK59383A (en)
HU (1) HU183215B (en)
IE (1) IE50268B1 (en)
IL (1) IL60999A (en)
IN (3) IN151313B (en)
IT (1) IT1133823B (en)
KE (1) KE3307A (en)
LU (1) LU82797A1 (en)
MX (1) MX7159E (en)
NL (1) NL8005346A (en)
NO (1) NO152128C (en)
NZ (1) NZ195061A (en)
PH (1) PH22628A (en)
PL (1) PL128998B1 (en)
PT (1) PT71839B (en)
SE (1) SE448626B (en)
SG (1) SG42983G (en)
YU (3) YU41734B (en)
ZA (1) ZA805476B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them
US6646001B2 (en) 1997-12-19 2003-11-11 Alcon Manufacturing, Ltd. Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension
US6066671A (en) * 1997-12-19 2000-05-23 Alcon Laboratories, Inc. Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides
GB9727523D0 (en) * 1997-12-31 1998-02-25 Pharmacia & Upjohn Spa Alpha-aminoamide derivatives useful as analgesic agents
AR030345A1 (en) * 2000-08-14 2003-08-20 Alcon Inc METHOD OF TREATMENT OF DISORDERS RELATED TO ANGIOGENESIS
ES2253579T3 (en) 2001-09-03 2006-06-01 Newron Pharmaceuticals S.P.A. PHARMACEUTICAL COMPOSITION INCLUDING GABAPENTINA OR AN ANALOG OF HER AND AN ALPHA-AMINOAMIDE AND ITS ANALGESIC USE.
EP1438956A1 (en) 2003-01-16 2004-07-21 Newron Pharmaceuticals S.p.A. Alpha-aminoamide derivatives useful as antimigraine agents
CZ2009367A3 (en) * 2009-06-08 2010-06-16 Farmak, A.S. Process for preparing 2-amino-3-benzoylphenylacetamide (nepafenac) with minimum of by-products
CN112794809B (en) * 2019-11-14 2023-12-29 南京济群医药科技股份有限公司 Preparation method of high-purity nepafenac intermediate

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1226344A (en) * 1967-07-31 1971-03-24
SE400966B (en) * 1975-08-13 1978-04-17 Robins Co Inc A H PROCEDURE FOR PREPARING 2-AMINO-3- (OR 5-) BENZOYL-PHENYLETIC ACIDS
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
IL60999A0 (en) 1980-11-30
IN156254B (en) 1985-06-08
GB2059963B (en) 1983-04-20
FI72967B (en) 1987-04-30
IT8024948A0 (en) 1980-09-26
KR840000763B1 (en) 1984-06-08
PT71839A (en) 1980-10-01
DK154136B (en) 1988-10-17
AU532359B2 (en) 1983-09-29
DE3035688A1 (en) 1981-04-16
IE801946L (en) 1981-03-26
ES495329A0 (en) 1981-10-16
IN151313B (en) 1983-03-26
ZA805476B (en) 1981-11-25
DK154136C (en) 1989-03-06
PL128998B1 (en) 1984-03-31
BE885393A (en) 1981-01-16
NO802834L (en) 1981-03-27
YU73183A (en) 1983-12-31
HU183215B (en) 1984-04-28
YU73083A (en) 1983-12-31
PL226919A1 (en) 1982-02-01
NZ195061A (en) 1984-04-27
FI72967C (en) 1987-08-10
SE8006668L (en) 1981-03-27
FR2465710A1 (en) 1981-03-27
YU245080A (en) 1983-09-30
IT1133823B (en) 1986-07-24
AT374170B (en) 1984-03-26
SE448626B (en) 1987-03-09
PT71839B (en) 1981-06-25
ES8200329A1 (en) 1981-10-16
NO152128C (en) 1985-08-07
IN156255B (en) 1985-06-08
GR70049B (en) 1982-07-26
YU43306B (en) 1989-06-30
FR2465710B1 (en) 1984-10-12
LU82797A1 (en) 1982-05-10
NL8005346A (en) 1981-03-30
ES503019A0 (en) 1982-05-01
HK59383A (en) 1983-12-02
CS227012B2 (en) 1984-04-16
DE3035688C2 (en) 1990-05-17
KR830004210A (en) 1983-07-06
DK405780A (en) 1981-03-27
YU41734B (en) 1987-12-31
JPH0141616B2 (en) 1989-09-06
SG42983G (en) 1985-01-11
IE50268B1 (en) 1986-03-19
ATA474580A (en) 1983-08-15
YU43305B (en) 1989-06-30
IL60999A (en) 1984-05-31
EG15020A (en) 1985-03-31
BR8006042A (en) 1981-04-07
PH22628A (en) 1988-10-28
FI803002A (en) 1981-03-27
NO152128B (en) 1985-04-29
JPS5657751A (en) 1981-05-20
KE3307A (en) 1983-08-19
GB2059963A (en) 1981-04-29
ES8204715A1 (en) 1982-05-01
AU6211680A (en) 1981-04-02
CA1128512A (en) 1982-07-27
CH646138A5 (en) 1984-11-15

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