NO152128C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES - Google Patents
ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDESInfo
- Publication number
- NO152128C NO152128C NO802834A NO802834A NO152128C NO 152128 C NO152128 C NO 152128C NO 802834 A NO802834 A NO 802834A NO 802834 A NO802834 A NO 802834A NO 152128 C NO152128 C NO 152128C
- Authority
- NO
- Norway
- Prior art keywords
- benzoylphenyl
- acetamides
- amino
- preparation
- therapeutic active
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US7886079A | 1979-09-26 | 1979-09-26 |
Publications (3)
Publication Number | Publication Date |
---|---|
NO802834L NO802834L (en) | 1981-03-27 |
NO152128B NO152128B (en) | 1985-04-29 |
NO152128C true NO152128C (en) | 1985-08-07 |
Family
ID=22146633
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO802834A NO152128C (en) | 1979-09-26 | 1980-09-25 | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES |
Country Status (36)
Country | Link |
---|---|
JP (1) | JPS5657751A (en) |
KR (1) | KR840000763B1 (en) |
AT (1) | AT374170B (en) |
AU (1) | AU532359B2 (en) |
BE (1) | BE885393A (en) |
BR (1) | BR8006042A (en) |
CA (1) | CA1128512A (en) |
CH (1) | CH646138A5 (en) |
CS (1) | CS227012B2 (en) |
DE (1) | DE3035688A1 (en) |
DK (1) | DK154136C (en) |
EG (1) | EG15020A (en) |
ES (2) | ES8200329A1 (en) |
FI (1) | FI72967C (en) |
FR (1) | FR2465710A1 (en) |
GB (1) | GB2059963B (en) |
GR (1) | GR70049B (en) |
HK (1) | HK59383A (en) |
HU (1) | HU183215B (en) |
IE (1) | IE50268B1 (en) |
IL (1) | IL60999A (en) |
IN (3) | IN151313B (en) |
IT (1) | IT1133823B (en) |
KE (1) | KE3307A (en) |
LU (1) | LU82797A1 (en) |
MX (1) | MX7159E (en) |
NL (1) | NL8005346A (en) |
NO (1) | NO152128C (en) |
NZ (1) | NZ195061A (en) |
PH (1) | PH22628A (en) |
PL (1) | PL128998B1 (en) |
PT (1) | PT71839B (en) |
SE (1) | SE448626B (en) |
SG (1) | SG42983G (en) |
YU (3) | YU41734B (en) |
ZA (1) | ZA805476B (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL61945A (en) * | 1980-02-19 | 1984-09-30 | Robins Co Inc A H | 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them |
US6066671A (en) * | 1997-12-19 | 2000-05-23 | Alcon Laboratories, Inc. | Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides |
US6646001B2 (en) | 1997-12-19 | 2003-11-11 | Alcon Manufacturing, Ltd. | Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension |
GB9727523D0 (en) | 1997-12-31 | 1998-02-25 | Pharmacia & Upjohn Spa | Alpha-aminoamide derivatives useful as analgesic agents |
AR030345A1 (en) * | 2000-08-14 | 2003-08-20 | Alcon Inc | METHOD OF TREATMENT OF DISORDERS RELATED TO ANGIOGENESIS |
IL160523A0 (en) | 2001-09-03 | 2004-07-25 | Newron Pharm Spa | PHARMACEUTICAL COMPOSITION COMPRISING GABAPENTIN OR AN ANALOGUE THEREOF AND AN alpha-AMINOAMIDE AND ITS ANALGESIC USE |
EP1438956A1 (en) | 2003-01-16 | 2004-07-21 | Newron Pharmaceuticals S.p.A. | Alpha-aminoamide derivatives useful as antimigraine agents |
CZ2009367A3 (en) * | 2009-06-08 | 2010-06-16 | Farmak, A.S. | Process for preparing 2-amino-3-benzoylphenylacetamide (nepafenac) with minimum of by-products |
CN112794809B (en) * | 2019-11-14 | 2023-12-29 | 南京济群医药科技股份有限公司 | Preparation method of high-purity nepafenac intermediate |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1226344A (en) * | 1967-07-31 | 1971-03-24 | ||
CH577461A5 (en) * | 1975-08-13 | 1976-07-15 | Robins Co Inc A H | |
IL61945A (en) * | 1980-02-19 | 1984-09-30 | Robins Co Inc A H | 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them |
-
1980
- 1980-09-04 ZA ZA00805476A patent/ZA805476B/en unknown
- 1980-09-08 AU AU62116/80A patent/AU532359B2/en not_active Ceased
- 1980-09-08 IL IL60999A patent/IL60999A/en unknown
- 1980-09-11 CS CS806196A patent/CS227012B2/en unknown
- 1980-09-17 IE IE1946/80A patent/IE50268B1/en unknown
- 1980-09-20 EG EG80573A patent/EG15020A/en active
- 1980-09-22 DE DE19803035688 patent/DE3035688A1/en active Granted
- 1980-09-22 BR BR8006042A patent/BR8006042A/en unknown
- 1980-09-22 GR GR62936A patent/GR70049B/el unknown
- 1980-09-23 PH PH24613A patent/PH22628A/en unknown
- 1980-09-23 AT AT0474580A patent/AT374170B/en not_active IP Right Cessation
- 1980-09-24 FI FI803002A patent/FI72967C/en not_active IP Right Cessation
- 1980-09-24 LU LU82797A patent/LU82797A1/en unknown
- 1980-09-24 SE SE8006668A patent/SE448626B/en not_active IP Right Cessation
- 1980-09-25 CA CA361,068A patent/CA1128512A/en not_active Expired
- 1980-09-25 HU HU802347A patent/HU183215B/en not_active IP Right Cessation
- 1980-09-25 NL NL8005346A patent/NL8005346A/en not_active Application Discontinuation
- 1980-09-25 GB GB8030955A patent/GB2059963B/en not_active Expired
- 1980-09-25 YU YU2450/80A patent/YU41734B/en unknown
- 1980-09-25 PT PT71839A patent/PT71839B/en unknown
- 1980-09-25 MX MX809050U patent/MX7159E/en unknown
- 1980-09-25 DK DK405780A patent/DK154136C/en not_active IP Right Cessation
- 1980-09-25 KR KR1019800003740A patent/KR840000763B1/en active
- 1980-09-25 FR FR8020596A patent/FR2465710A1/en active Granted
- 1980-09-25 CH CH719180A patent/CH646138A5/en not_active IP Right Cessation
- 1980-09-25 NO NO802834A patent/NO152128C/en unknown
- 1980-09-25 ES ES495329A patent/ES8200329A1/en not_active Expired
- 1980-09-25 PL PL1980226919A patent/PL128998B1/en unknown
- 1980-09-25 BE BE0/202226A patent/BE885393A/en not_active IP Right Cessation
- 1980-09-26 IT IT24948/80A patent/IT1133823B/en active
- 1980-09-26 IN IN1092/CAL/80A patent/IN151313B/en unknown
- 1980-09-26 JP JP13415280A patent/JPS5657751A/en active Granted
- 1980-09-26 NZ NZ195061A patent/NZ195061A/en unknown
-
1981
- 1981-06-12 ES ES503019A patent/ES8204715A1/en not_active Expired
-
1982
- 1982-12-30 IN IN1508/CAL/82A patent/IN156254B/en unknown
- 1982-12-30 IN IN1509/CAL/82A patent/IN156255B/en unknown
-
1983
- 1983-03-28 YU YU730/83A patent/YU43305B/en unknown
- 1983-03-28 YU YU731/83A patent/YU43306B/en unknown
- 1983-07-19 SG SG42983A patent/SG42983G/en unknown
- 1983-07-21 KE KE3307A patent/KE3307A/en unknown
- 1983-11-24 HK HK593/83A patent/HK59383A/en unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO155055C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES. | |
NO800858L (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 4-AMINO-3-QUINOLINCARBOXYLIC ACID DERIVATIVES | |
NO151588C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE N2-ARYLSULPHONYL-L-ARGININAMIDE DERIVATIVES | |
NO151320C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRROLIDYLMETHYL-2-METOXY-4-AMINO-5-ISOPROPYL-SULPHONYL BENZAMIDES | |
NO150760C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE AMINOTIAZOLES. | |
NO803764L (en) | PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BASIC ETHERS | |
NO152213C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE SUBSTITUTED BENZAZEPINES | |
NO150360C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BRAND CAPACYLDIPEPTIDES | |
NO149312C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2- (2-TENOYLTIO) -PROPIONYLGYLINE | |
NO151201C (en) | PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ANTIGENDATIVE DERIVATIVES | |
NO814055L (en) | PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE THIENOPYRIDINO DERIVATIVES | |
NO151319C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BETA-MONO-FLUORMETHYL-BETA-ALANINE AND BETA-DIFLUORMETHYL-BETA-ALANINE COMPOUNDS | |
NO152007C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVITY 7BETA- (SYN-2-OXYYMINO-ARYLACETAMIDO) -3- (SULPHALKYLTETRAZOL-5-YL-THIOMETHYL) -CPHEM-4-CARBOXYL | |
NO151288C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE INDOLOKINOLIZINDINS | |
NO149737C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 1-AZAXANTHON-3-CARBOXYLIC ACIDS | |
NO151239C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-PHENYLIMINOIMIDAZOLIDINES | |
NO150916C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC ACTIVE PHENOXYPROPANOLAMINE DERIVATIVE | |
NO157976C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3-PHENOXY-1-AZETIDINCARBOXAMIDES. | |
NO781879L (en) | ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PYRIDOBENZODIAZEPINES | |
NO152128C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES | |
NO152787C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PHENYL-CHINOLIZIDINES. | |
NO148451C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE OXIMETERS | |
NO151008C (en) | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE NITROPHANES | |
NO153141C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 4-AZA-17-SUBSTITUTED-5ALFA-ANDROSTAN-3-ONER. | |
NO155842C (en) | ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-BETA-D-RIBOFURANOSYLSELENAZOLE-4-CARBOXAMIDES. |