NO152128C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES

Info

Publication number
NO152128C
NO152128C NO802834A NO802834A NO152128C NO 152128 C NO152128 C NO 152128C NO 802834 A NO802834 A NO 802834A NO 802834 A NO802834 A NO 802834A NO 152128 C NO152128 C NO 152128C
Authority
NO
Norway
Prior art keywords
benzoylphenyl
acetamides
amino
preparation
therapeutic active
Prior art date
Application number
NO802834A
Other languages
Norwegian (no)
Other versions
NO152128B (en
NO802834L (en
Inventor
James Robert Shanklin Jr
Dwight Allan Shamblee
David Allen Walsh
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of NO802834L publication Critical patent/NO802834L/en
Publication of NO152128B publication Critical patent/NO152128B/en
Publication of NO152128C publication Critical patent/NO152128C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182Radicals derived from carboxylic acids
    • C07D295/185Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
NO802834A 1979-09-26 1980-09-25 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES NO152128C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7886079A 1979-09-26 1979-09-26

Publications (3)

Publication Number Publication Date
NO802834L NO802834L (en) 1981-03-27
NO152128B NO152128B (en) 1985-04-29
NO152128C true NO152128C (en) 1985-08-07

Family

ID=22146633

Family Applications (1)

Application Number Title Priority Date Filing Date
NO802834A NO152128C (en) 1979-09-26 1980-09-25 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-3-BENZOYLPHENYL ACETAMIDES

Country Status (36)

Country Link
JP (1) JPS5657751A (en)
KR (1) KR840000763B1 (en)
AT (1) AT374170B (en)
AU (1) AU532359B2 (en)
BE (1) BE885393A (en)
BR (1) BR8006042A (en)
CA (1) CA1128512A (en)
CH (1) CH646138A5 (en)
CS (1) CS227012B2 (en)
DE (1) DE3035688A1 (en)
DK (1) DK154136C (en)
EG (1) EG15020A (en)
ES (2) ES8200329A1 (en)
FI (1) FI72967C (en)
FR (1) FR2465710A1 (en)
GB (1) GB2059963B (en)
GR (1) GR70049B (en)
HK (1) HK59383A (en)
HU (1) HU183215B (en)
IE (1) IE50268B1 (en)
IL (1) IL60999A (en)
IN (3) IN151313B (en)
IT (1) IT1133823B (en)
KE (1) KE3307A (en)
LU (1) LU82797A1 (en)
MX (1) MX7159E (en)
NL (1) NL8005346A (en)
NO (1) NO152128C (en)
NZ (1) NZ195061A (en)
PH (1) PH22628A (en)
PL (1) PL128998B1 (en)
PT (1) PT71839B (en)
SE (1) SE448626B (en)
SG (1) SG42983G (en)
YU (3) YU41734B (en)
ZA (1) ZA805476B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them
US6066671A (en) * 1997-12-19 2000-05-23 Alcon Laboratories, Inc. Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides
US6646001B2 (en) 1997-12-19 2003-11-11 Alcon Manufacturing, Ltd. Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension
GB9727523D0 (en) 1997-12-31 1998-02-25 Pharmacia & Upjohn Spa Alpha-aminoamide derivatives useful as analgesic agents
AR030345A1 (en) * 2000-08-14 2003-08-20 Alcon Inc METHOD OF TREATMENT OF DISORDERS RELATED TO ANGIOGENESIS
IL160523A0 (en) 2001-09-03 2004-07-25 Newron Pharm Spa PHARMACEUTICAL COMPOSITION COMPRISING GABAPENTIN OR AN ANALOGUE THEREOF AND AN alpha-AMINOAMIDE AND ITS ANALGESIC USE
EP1438956A1 (en) 2003-01-16 2004-07-21 Newron Pharmaceuticals S.p.A. Alpha-aminoamide derivatives useful as antimigraine agents
CZ2009367A3 (en) * 2009-06-08 2010-06-16 Farmak, A.S. Process for preparing 2-amino-3-benzoylphenylacetamide (nepafenac) with minimum of by-products
CN112794809B (en) * 2019-11-14 2023-12-29 南京济群医药科技股份有限公司 Preparation method of high-purity nepafenac intermediate

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1226344A (en) * 1967-07-31 1971-03-24
CH577461A5 (en) * 1975-08-13 1976-07-15 Robins Co Inc A H
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
EG15020A (en) 1985-03-31
FR2465710B1 (en) 1984-10-12
KE3307A (en) 1983-08-19
JPS5657751A (en) 1981-05-20
FI803002A (en) 1981-03-27
IL60999A0 (en) 1980-11-30
LU82797A1 (en) 1982-05-10
GB2059963A (en) 1981-04-29
AU6211680A (en) 1981-04-02
PL128998B1 (en) 1984-03-31
AU532359B2 (en) 1983-09-29
BR8006042A (en) 1981-04-07
NZ195061A (en) 1984-04-27
YU73183A (en) 1983-12-31
SG42983G (en) 1985-01-11
PT71839A (en) 1980-10-01
FI72967C (en) 1987-08-10
KR840000763B1 (en) 1984-06-08
DE3035688A1 (en) 1981-04-16
CH646138A5 (en) 1984-11-15
IN156255B (en) 1985-06-08
ES495329A0 (en) 1981-10-16
GR70049B (en) 1982-07-26
IT8024948A0 (en) 1980-09-26
FR2465710A1 (en) 1981-03-27
HU183215B (en) 1984-04-28
ZA805476B (en) 1981-11-25
MX7159E (en) 1987-12-02
DK154136B (en) 1988-10-17
IL60999A (en) 1984-05-31
IN151313B (en) 1983-03-26
FI72967B (en) 1987-04-30
AT374170B (en) 1984-03-26
DK154136C (en) 1989-03-06
ES8200329A1 (en) 1981-10-16
CS227012B2 (en) 1984-04-16
JPH0141616B2 (en) 1989-09-06
YU43305B (en) 1989-06-30
NL8005346A (en) 1981-03-30
SE448626B (en) 1987-03-09
DE3035688C2 (en) 1990-05-17
KR830004210A (en) 1983-07-06
DK405780A (en) 1981-03-27
NO152128B (en) 1985-04-29
PT71839B (en) 1981-06-25
YU73083A (en) 1983-12-31
SE8006668L (en) 1981-03-27
IN156254B (en) 1985-06-08
YU41734B (en) 1987-12-31
ES503019A0 (en) 1982-05-01
HK59383A (en) 1983-12-02
IT1133823B (en) 1986-07-24
CA1128512A (en) 1982-07-27
GB2059963B (en) 1983-04-20
YU245080A (en) 1983-09-30
ES8204715A1 (en) 1982-05-01
ATA474580A (en) 1983-08-15
IE801946L (en) 1981-03-26
PL226919A1 (en) 1982-02-01
IE50268B1 (en) 1986-03-19
YU43306B (en) 1989-06-30
PH22628A (en) 1988-10-28
NO802834L (en) 1981-03-27
BE885393A (en) 1981-01-16

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