NO327207B1 - Forbindelser som er spesifikke overfor adenosin-A1, A2A og A3-reseptor samt anvendelse derav for fremstilling av medikamenter og fremgangsmate for fremstilling av forbindelsene - Google Patents
Forbindelser som er spesifikke overfor adenosin-A1, A2A og A3-reseptor samt anvendelse derav for fremstilling av medikamenter og fremgangsmate for fremstilling av forbindelsene Download PDFInfo
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- NO327207B1 NO327207B1 NO20032482A NO20032482A NO327207B1 NO 327207 B1 NO327207 B1 NO 327207B1 NO 20032482 A NO20032482 A NO 20032482A NO 20032482 A NO20032482 A NO 20032482A NO 327207 B1 NO327207 B1 NO 327207B1
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US09/728,616 US7160890B2 (en) | 1999-12-02 | 2000-12-01 | Compounds specific to adenosine A3 receptor and uses thereof |
US09/728,607 US6664252B2 (en) | 1999-12-02 | 2000-12-01 | 4-aminopyrrolo[2,3-d]pyrimidine compounds specific to adenosine A2a receptor and uses thereof |
US09/728,316 US6680322B2 (en) | 1999-12-02 | 2000-12-01 | Compounds specific to adenosine A1 receptors and uses thereof |
PCT/US2001/045280 WO2002057267A1 (en) | 2000-12-01 | 2001-11-30 | Compounds specific to adenosine a1, a2a, and a3 receptor and uses thereof |
Publications (3)
Publication Number | Publication Date |
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NO20032482D0 NO20032482D0 (no) | 2003-06-02 |
NO20032482L NO20032482L (no) | 2003-07-28 |
NO327207B1 true NO327207B1 (no) | 2009-05-11 |
Family
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NO20032482A NO327207B1 (no) | 2000-12-01 | 2003-06-02 | Forbindelser som er spesifikke overfor adenosin-A1, A2A og A3-reseptor samt anvendelse derav for fremstilling av medikamenter og fremgangsmate for fremstilling av forbindelsene |
Country Status (20)
Country | Link |
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EP (1) | EP1347980A4 (ru) |
JP (1) | JP4579497B2 (ru) |
CN (1) | CN1263757C (ru) |
AP (1) | AP1893A (ru) |
AU (1) | AU2002248151B2 (ru) |
BR (1) | BR0115847A (ru) |
CA (1) | CA2430577A1 (ru) |
CZ (1) | CZ20031831A3 (ru) |
EA (1) | EA007254B1 (ru) |
HU (1) | HUP0400692A3 (ru) |
IL (1) | IL155962A0 (ru) |
ME (1) | MEP35308A (ru) |
MX (1) | MXPA03004717A (ru) |
NO (1) | NO327207B1 (ru) |
NZ (1) | NZ525885A (ru) |
OA (1) | OA13295A (ru) |
PL (1) | PL363245A1 (ru) |
WO (1) | WO2002057267A1 (ru) |
YU (1) | YU42703A (ru) |
ZA (1) | ZA200303729B (ru) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
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US5090531A (en) * | 1990-01-10 | 1992-02-25 | Lord Corporation | Electrophoretic fluid differential |
PL204628B1 (pl) | 1998-06-02 | 2010-01-29 | Osi Pharmaceuticals | Pochodna pirolo[2,3d]pirymidyny, jej zastosowanie i sposoby wytwarzania tej pochodnej i preparaty farmaceutyczne |
US6680324B2 (en) | 2000-12-01 | 2004-01-20 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A1 receptors and uses thereof |
DE10148883A1 (de) * | 2001-10-04 | 2003-04-10 | Merck Patent Gmbh | Pyrimidinderivate |
EP1450811B1 (en) * | 2001-11-30 | 2009-10-21 | OSI Pharmaceuticals, Inc. | Compounds specific to adenosine A1 and A3 receptors and uses thereof |
EP2198867A1 (en) * | 2001-12-07 | 2010-06-23 | Vertex Pharmaceuticals, Inc. | Pyrimidine-based compounds useful as GSK-3 inhibitors |
CA2471059C (en) | 2001-12-20 | 2011-04-26 | Osi Pharmaceuticals, Inc. | Pyrimidine a2b selective antagonist compounds, their synthesis and use |
US20030229067A1 (en) | 2001-12-20 | 2003-12-11 | Arlindo Castelhano | Pyrrolopyrimidine A2b selective antagonist compounds, their synthesis and use |
CA2502429A1 (en) * | 2002-10-31 | 2004-05-21 | Amgen Inc. | Antiinflammation agents |
HUP0203976A3 (en) * | 2002-11-15 | 2004-08-30 | Sanofi Aventis | Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them |
MY179032A (en) | 2004-10-25 | 2020-10-26 | Cancer Research Tech Ltd | Ortho-condensed pyridine and pyrimidine derivatives (e.g.purines) as protein kinase inhibitors |
UY29177A1 (es) | 2004-10-25 | 2006-05-31 | Astex Therapeutics Ltd | Derivados sustituidos de purina, purinona y deazapurina, composiciones que los contienen métodos para su preparación y sus usos |
EP3421471B1 (en) | 2006-04-25 | 2021-05-26 | Astex Therapeutics Limited | Purine and deazapurine derivatives as pharmaceutical compounds |
US20070260203A1 (en) * | 2006-05-04 | 2007-11-08 | Allergan, Inc. | Vasoactive agent intraocular implant |
TW200808819A (en) * | 2006-06-19 | 2008-02-16 | Solvay Pharm Gmbh | Use of adenosine A1 antagonists in radiocontrast media induced nephrophaty |
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NO20032482L (no) | 2003-07-28 |
CA2430577A1 (en) | 2002-07-25 |
BR0115847A (pt) | 2004-02-25 |
HUP0400692A3 (en) | 2007-09-28 |
MXPA03004717A (es) | 2004-06-30 |
IL155962A0 (en) | 2003-12-23 |
MEP35308A (en) | 2011-02-10 |
OA13295A (en) | 2007-04-13 |
AP2003002807A0 (en) | 2003-06-30 |
NO20032482D0 (no) | 2003-06-02 |
CN1489590A (zh) | 2004-04-14 |
PL363245A1 (en) | 2004-11-15 |
HUP0400692A2 (hu) | 2004-07-28 |
EP1347980A4 (en) | 2005-02-09 |
NZ525885A (en) | 2005-01-28 |
CN1263757C (zh) | 2006-07-12 |
AU2002248151B2 (en) | 2008-02-21 |
JP2004517896A (ja) | 2004-06-17 |
EA007254B1 (ru) | 2006-08-25 |
JP4579497B2 (ja) | 2010-11-10 |
CZ20031831A3 (cs) | 2004-05-12 |
WO2002057267A1 (en) | 2002-07-25 |
ZA200303729B (en) | 2004-05-14 |
EA200300628A1 (ru) | 2003-12-25 |
EP1347980A1 (en) | 2003-10-01 |
AP1893A (en) | 2008-09-23 |
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