NO326375B1 - Vedvarende frigivelsesformuleringer av oksymorfon samt fast doseringsform inneholdende slike. - Google Patents
Vedvarende frigivelsesformuleringer av oksymorfon samt fast doseringsform inneholdende slike. Download PDFInfo
- Publication number
- NO326375B1 NO326375B1 NO20031019A NO20031019A NO326375B1 NO 326375 B1 NO326375 B1 NO 326375B1 NO 20031019 A NO20031019 A NO 20031019A NO 20031019 A NO20031019 A NO 20031019A NO 326375 B1 NO326375 B1 NO 326375B1
- Authority
- NO
- Norway
- Prior art keywords
- sustained release
- release formulation
- oxymorphone
- delivery system
- amount
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Emergency Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Pain & Pain Management (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Rheumatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Dental Preparations (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30335701P | 2001-07-06 | 2001-07-06 | |
| US32935201P | 2001-10-15 | 2001-10-15 | |
| US32942601P | 2001-10-15 | 2001-10-15 | |
| PCT/US2002/021403 WO2003004033A1 (en) | 2001-07-06 | 2002-07-03 | Sustained release formulations of oxymorphone |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20031019D0 NO20031019D0 (no) | 2003-03-05 |
| NO20031019L NO20031019L (no) | 2003-05-05 |
| NO326375B1 true NO326375B1 (no) | 2008-11-17 |
Family
ID=27404938
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20031019A NO326375B1 (no) | 2001-07-06 | 2003-03-05 | Vedvarende frigivelsesformuleringer av oksymorfon samt fast doseringsform inneholdende slike. |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US20030129234A1 (de) |
| EP (2) | EP1404331B1 (de) |
| KR (1) | KR20030048026A (de) |
| AT (1) | ATE376832T1 (de) |
| BR (2) | BR0205722A (de) |
| DE (1) | DE60223254T2 (de) |
| DK (1) | DK1404331T3 (de) |
| ES (1) | ES2292775T3 (de) |
| HK (1) | HK1064921A1 (de) |
| NO (1) | NO326375B1 (de) |
| PL (2) | PL207748B1 (de) |
| WO (2) | WO2003004033A1 (de) |
Families Citing this family (67)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5478577A (en) * | 1993-11-23 | 1995-12-26 | Euroceltique, S.A. | Method of treating pain by administering 24 hour oral opioid formulations exhibiting rapid rate of initial rise of plasma drug level |
| WO2002100382A2 (en) * | 2001-06-08 | 2002-12-19 | Endo Pharmaceuticals, Inc. | Controlled release dosage forms using acrylic polymer, and process for making the same |
| KR20030048026A (ko) * | 2001-07-06 | 2003-06-18 | 펜웨스트 파머슈티칼즈 컴파니 | 옥시모르폰의 서방형 제제 |
| WO2003004031A1 (en) * | 2001-07-06 | 2003-01-16 | Endo Pharmaceuticals, Inc. | Parenteral administration of 6-hydroxy-oxymorphone for use as an analgesic |
| US8329216B2 (en) | 2001-07-06 | 2012-12-11 | Endo Pharmaceuticals Inc. | Oxymorphone controlled release formulations |
| US20030068375A1 (en) | 2001-08-06 | 2003-04-10 | Curtis Wright | Pharmaceutical formulation containing gelling agent |
| EP1429730A4 (de) * | 2001-09-26 | 2010-06-16 | Penwest Pharmaceuticals Compan | Opioid-formulierungen mit verringertem missbrauchspotenzial |
| US7776314B2 (en) | 2002-06-17 | 2010-08-17 | Grunenthal Gmbh | Abuse-proofed dosage system |
| US8840928B2 (en) | 2002-07-05 | 2014-09-23 | Collegium Pharmaceutical, Inc. | Tamper-resistant pharmaceutical compositions of opioids and other drugs |
| US8557291B2 (en) | 2002-07-05 | 2013-10-15 | Collegium Pharmaceutical, Inc. | Abuse-deterrent pharmaceutical compositions of opioids and other drugs |
| WO2004004693A1 (en) | 2002-07-05 | 2004-01-15 | Collgegium Pharmaceutical | Abuse-deterrent pharmaceutical compositions of opiods and other drugs |
| US10004729B2 (en) | 2002-07-05 | 2018-06-26 | Collegium Pharmaceutical, Inc. | Tamper-resistant pharmaceutical compositions of opioids and other drugs |
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| AU2002324624A1 (en) * | 2001-08-06 | 2003-02-24 | Euro-Celtique S.A. | Sequestered antagonist formulations |
| US7141250B2 (en) | 2001-08-06 | 2006-11-28 | Euro-Celtique S.A. | Pharmaceutical formulation containing bittering agent |
| IS7142A (is) * | 2001-08-06 | 2004-02-05 | Euroceltique S.A. | Lyfjasamsetningar, sem innihalda morfíngerandaefni, ásamt losanlegu en hömdu mótlyfi |
| US20030049272A1 (en) | 2001-08-30 | 2003-03-13 | Yatindra Joshi | Pharmaceutical composition which produces irritation |
| US20030059397A1 (en) | 2001-09-17 | 2003-03-27 | Lyn Hughes | Dosage forms |
| US20030068276A1 (en) | 2001-09-17 | 2003-04-10 | Lyn Hughes | Dosage forms |
| EP1429730A4 (de) * | 2001-09-26 | 2010-06-16 | Penwest Pharmaceuticals Compan | Opioid-formulierungen mit verringertem missbrauchspotenzial |
| JP2005508372A (ja) * | 2001-11-02 | 2005-03-31 | エラン コーポレーシヨン ピーエルシー | 薬剤組成物 |
| ATE374602T1 (de) * | 2001-12-21 | 2007-10-15 | Supernus Pharmaceuticals Inc | Orale kapselformulierung mit verbesserter physikalischer stabilität |
| US20030158264A1 (en) * | 2002-02-20 | 2003-08-21 | Ramachandran Radhakrishnan | Orally administrable pharmaceutical formulation comprising ephedrine hydrochloride and process for preparing the same |
| US7524515B2 (en) * | 2003-01-10 | 2009-04-28 | Mutual Pharmaceuticals, Inc. | Pharmaceutical safety dosage forms |
-
2002
- 2002-07-03 KR KR10-2003-7003334A patent/KR20030048026A/ko not_active Application Discontinuation
- 2002-07-03 DK DK02744835T patent/DK1404331T3/da active
- 2002-07-03 AT AT02744835T patent/ATE376832T1/de active
- 2002-07-03 US US10/190,383 patent/US20030129234A1/en not_active Abandoned
- 2002-07-03 BR BR0205722-0A patent/BR0205722A/pt not_active IP Right Cessation
- 2002-07-03 PL PL366430A patent/PL207748B1/pl unknown
- 2002-07-03 WO PCT/US2002/021403 patent/WO2003004033A1/en active IP Right Grant
- 2002-07-03 WO PCT/US2002/021354 patent/WO2003004029A1/en not_active Application Discontinuation
- 2002-07-03 PL PL367277A patent/PL208484B1/pl unknown
- 2002-07-03 EP EP02744835A patent/EP1404331B1/de not_active Expired - Lifetime
- 2002-07-03 EP EP02748085A patent/EP1404332A1/de not_active Withdrawn
- 2002-07-03 BR BRPI0210855-0A patent/BR0210855A/pt not_active IP Right Cessation
- 2002-07-03 ES ES02744835T patent/ES2292775T3/es not_active Expired - Lifetime
- 2002-07-03 US US10/189,932 patent/US7276250B2/en not_active Expired - Lifetime
- 2002-07-03 DE DE60223254T patent/DE60223254T2/de not_active Expired - Lifetime
-
2003
- 2003-03-05 NO NO20031019A patent/NO326375B1/no not_active IP Right Cessation
-
2004
- 2004-09-23 HK HK04107358A patent/HK1064921A1/xx not_active IP Right Cessation
-
2007
- 2007-08-13 US US11/891,775 patent/US20080050431A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| ATE376832T1 (de) | 2007-11-15 |
| PL208484B1 (pl) | 2011-05-31 |
| US20030129234A1 (en) | 2003-07-10 |
| DE60223254T2 (de) | 2008-08-14 |
| WO2003004029A1 (en) | 2003-01-16 |
| US7276250B2 (en) | 2007-10-02 |
| KR20030048026A (ko) | 2003-06-18 |
| DE60223254D1 (de) | 2007-12-13 |
| EP1404332A1 (de) | 2004-04-07 |
| EP1404331B1 (de) | 2007-10-31 |
| PL367277A1 (en) | 2005-02-21 |
| US20080050431A1 (en) | 2008-02-28 |
| WO2003004033A1 (en) | 2003-01-16 |
| BR0205722A (pt) | 2005-04-05 |
| US20030129230A1 (en) | 2003-07-10 |
| PL207748B1 (pl) | 2011-01-31 |
| DK1404331T3 (da) | 2008-01-28 |
| BR0210855A (pt) | 2006-10-24 |
| NO20031019L (no) | 2003-05-05 |
| HK1064921A1 (en) | 2005-02-08 |
| PL366430A1 (en) | 2005-01-24 |
| ES2292775T3 (es) | 2008-03-16 |
| NO20031019D0 (no) | 2003-03-05 |
| EP1404331A1 (de) | 2004-04-07 |
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