NO324693B1 - 2-acetamidoacetamidderivater, anvendelse av slike forbindelser til fremstilling av preparater for behandling av sykdommer samt preparater omfattende slike forbindelser - Google Patents

2-acetamidoacetamidderivater, anvendelse av slike forbindelser til fremstilling av preparater for behandling av sykdommer samt preparater omfattende slike forbindelser Download PDF

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Publication number
NO324693B1
NO324693B1 NO20025405A NO20025405A NO324693B1 NO 324693 B1 NO324693 B1 NO 324693B1 NO 20025405 A NO20025405 A NO 20025405A NO 20025405 A NO20025405 A NO 20025405A NO 324693 B1 NO324693 B1 NO 324693B1
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NO
Norway
Prior art keywords
alkyl
phenyl
group
substituted
methyl
Prior art date
Application number
NO20025405A
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English (en)
Norwegian (no)
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NO20025405D0 (no
NO20025405L (no
Inventor
Scott F Sneddon
John L Kane
Bradford H Hirth
Fred Vinick
Shuang Qiao
Sharon R Nahill
John M Williams
Hans-Peter Biemann
Andrew Janjigian
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Genzyme Corp
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Publication of NO20025405D0 publication Critical patent/NO20025405D0/no
Publication of NO20025405L publication Critical patent/NO20025405L/no
Publication of NO324693B1 publication Critical patent/NO324693B1/no

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
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    • A61P21/04Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
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    • A61P37/02Immunomodulators
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    • A61P5/14Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

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NO20025405A 2000-05-12 2002-11-11 2-acetamidoacetamidderivater, anvendelse av slike forbindelser til fremstilling av preparater for behandling av sykdommer samt preparater omfattende slike forbindelser NO324693B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20378400P 2000-05-12 2000-05-12
US20521300P 2000-05-18 2000-05-18
PCT/US2001/015027 WO2001087849A2 (en) 2000-05-12 2001-05-10 Modulators of tnf- alpha signaling

Publications (3)

Publication Number Publication Date
NO20025405D0 NO20025405D0 (no) 2002-11-11
NO20025405L NO20025405L (no) 2003-01-09
NO324693B1 true NO324693B1 (no) 2007-12-03

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NO20025405A NO324693B1 (no) 2000-05-12 2002-11-11 2-acetamidoacetamidderivater, anvendelse av slike forbindelser til fremstilling av preparater for behandling av sykdommer samt preparater omfattende slike forbindelser

Country Status (13)

Country Link
US (5) US6969728B2 (zh)
EP (1) EP1294699B1 (zh)
JP (3) JP4960565B2 (zh)
KR (1) KR100840816B1 (zh)
CN (1) CN100494182C (zh)
AU (2) AU2001259691B2 (zh)
BR (1) BR0111158A (zh)
CA (3) CA2781858C (zh)
HK (1) HK1051186A1 (zh)
IL (2) IL152450A0 (zh)
MX (1) MXPA02010993A (zh)
NO (1) NO324693B1 (zh)
WO (1) WO2001087849A2 (zh)

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US7034031B2 (en) 2006-04-25
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US9579325B2 (en) 2017-02-28
US6969728B2 (en) 2005-11-29
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