NO315651B1 - Benzopyraner, farmasöytiske preparater inneholdende disse og deres anvendelse som terapeutiske midler - Google Patents
Benzopyraner, farmasöytiske preparater inneholdende disse og deres anvendelse som terapeutiske midler Download PDFInfo
- Publication number
- NO315651B1 NO315651B1 NO19965260A NO965260A NO315651B1 NO 315651 B1 NO315651 B1 NO 315651B1 NO 19965260 A NO19965260 A NO 19965260A NO 965260 A NO965260 A NO 965260A NO 315651 B1 NO315651 B1 NO 315651B1
- Authority
- NO
- Norway
- Prior art keywords
- acetyl
- benzopyran
- dimethyl
- dihydro
- pharmaceutically acceptable
- Prior art date
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
- C07D311/68—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with nitrogen atoms directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrane Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9411632A GB9411632D0 (en) | 1994-06-10 | 1994-06-10 | Novel treatment |
| GB9411798A GB9411798D0 (en) | 1994-06-13 | 1994-06-13 | Novel treatment |
| PCT/EP1995/002076 WO1995034545A1 (en) | 1994-06-10 | 1995-05-31 | Benzopyrans and their use as therapeutic agents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO965260D0 NO965260D0 (no) | 1996-12-09 |
| NO965260L NO965260L (no) | 1997-02-06 |
| NO315651B1 true NO315651B1 (no) | 2003-10-06 |
Family
ID=26305044
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19965260A NO315651B1 (no) | 1994-06-10 | 1996-12-09 | Benzopyraner, farmasöytiske preparater inneholdende disse og deres anvendelse som terapeutiske midler |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US5760074A (pt) |
| EP (2) | EP0764157B1 (pt) |
| JP (2) | JP3575767B2 (pt) |
| KR (1) | KR100397721B1 (pt) |
| CN (2) | CN1234702C (pt) |
| AP (1) | AP714A (pt) |
| AT (2) | ATE211469T1 (pt) |
| AU (1) | AU701060B2 (pt) |
| BG (1) | BG63339B1 (pt) |
| BR (1) | BR9507980A (pt) |
| CA (1) | CA2192480C (pt) |
| CY (1) | CY2508B1 (pt) |
| CZ (1) | CZ286081B6 (pt) |
| DE (2) | DE69531801T2 (pt) |
| DK (2) | DK0764157T3 (pt) |
| ES (2) | ES2170798T3 (pt) |
| FI (1) | FI120686B (pt) |
| HK (2) | HK1001286A1 (pt) |
| HU (1) | HUT76136A (pt) |
| NO (1) | NO315651B1 (pt) |
| NZ (1) | NZ287872A (pt) |
| OA (1) | OA10593A (pt) |
| PL (1) | PL188134B1 (pt) |
| PT (2) | PT764157E (pt) |
| RO (1) | RO113463B1 (pt) |
| SG (1) | SG67930A1 (pt) |
| SI (2) | SI0764157T1 (pt) |
| SK (1) | SK281456B6 (pt) |
| WO (1) | WO1995034545A1 (pt) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20010021780A1 (en) * | 1992-12-11 | 2001-09-13 | Smithkline Beecham P.L.C. | Pharmaceutical composition containing bicyclic type compounds |
| GB9411635D0 (en) * | 1994-06-10 | 1994-08-03 | Smithkline Beecham Plc | Novel treatment |
| US6492415B2 (en) * | 1996-09-18 | 2002-12-10 | Smithkline Beecham P.L.C. | Use of benzopyranols to treat neurological disorders |
| GB9619492D0 (en) * | 1996-09-18 | 1996-10-30 | Smithkline Beecham Plc | Novel treatment |
| GB9726543D0 (en) * | 1997-12-16 | 1998-02-11 | Smithkline Beecham Plc | Novel compositions |
| GB9813949D0 (en) * | 1998-06-29 | 1998-08-26 | Smithkline Beecham Plc | Novel compounds |
| GB0028697D0 (en) * | 2000-11-23 | 2001-01-10 | S P A | Novel process |
| ZA200708445B (en) * | 2005-04-04 | 2009-03-25 | Takeda Pharmaceutical | Preventive or remedy for depression or anxiety neurosis |
| US20130281524A1 (en) * | 2008-06-05 | 2013-10-24 | Peter Blower | Novel treatments |
| EP2296646A2 (en) * | 2008-06-05 | 2011-03-23 | Minster Research Limited | Novel treatments |
| MX2012006352A (es) * | 2009-12-03 | 2012-06-27 | Proximagen Ltd | Tratamiento de alodinia e hiperalgesia. |
| CA2782631A1 (en) | 2009-12-03 | 2011-06-09 | Proximagen Ltd | Treatment of infectious diseases |
| AU2013285164A1 (en) | 2012-07-03 | 2015-01-22 | Proximagen Limited | Pro-drug compounds |
| GB201304814D0 (en) * | 2013-03-15 | 2013-05-01 | Proximagen Ltd | Pro-drug compounds |
| GB201322932D0 (en) * | 2013-12-23 | 2014-02-12 | Proximagen Ltd | Pro-drug compounds |
| GB201322934D0 (en) | 2013-12-23 | 2014-02-12 | Proximagen Ltd | Prodrug compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3479726D1 (de) * | 1983-05-18 | 1989-10-19 | Beecham Group Plc | Benzopyran derivatives. |
| GB9112721D0 (en) * | 1991-06-13 | 1991-07-31 | Smithkline Beecham Plc | Novel treatment |
| EP0673373A1 (en) * | 1992-12-11 | 1995-09-27 | Smithkline Beecham Plc | Bicyclic compounds with pharmaceutical activity |
| EP0673374B1 (en) * | 1992-12-11 | 2000-03-01 | Smithkline Beecham Plc | Pharmaceutical composition containing bicyclic type compounds |
| US5536718A (en) * | 1995-01-17 | 1996-07-16 | American Cyanamid Company | Tricyclic benzazepine vasopressin antagonists |
-
1995
- 1995-05-31 ES ES95921798T patent/ES2170798T3/es not_active Expired - Lifetime
- 1995-05-31 AT AT95921798T patent/ATE211469T1/de active
- 1995-05-31 NZ NZ287872A patent/NZ287872A/en not_active IP Right Cessation
- 1995-05-31 RO RO96-02326A patent/RO113463B1/ro unknown
- 1995-05-31 BR BR9507980A patent/BR9507980A/pt not_active IP Right Cessation
- 1995-05-31 SK SK1587-96A patent/SK281456B6/sk not_active IP Right Cessation
- 1995-05-31 PL PL95317579A patent/PL188134B1/pl unknown
- 1995-05-31 AT AT01200801T patent/ATE250052T1/de active
- 1995-05-31 PT PT95921798T patent/PT764157E/pt unknown
- 1995-05-31 AP APAP/P/1996/000889A patent/AP714A/en active
- 1995-05-31 JP JP50155696A patent/JP3575767B2/ja not_active Expired - Lifetime
- 1995-05-31 CA CA002192480A patent/CA2192480C/en not_active Expired - Lifetime
- 1995-05-31 AU AU26727/95A patent/AU701060B2/en not_active Expired
- 1995-05-31 DE DE69531801T patent/DE69531801T2/de not_active Expired - Lifetime
- 1995-05-31 CZ CZ19963617A patent/CZ286081B6/cs not_active IP Right Cessation
- 1995-05-31 EP EP95921798A patent/EP0764157B1/en not_active Expired - Lifetime
- 1995-05-31 CN CNB01124366XA patent/CN1234702C/zh not_active Expired - Lifetime
- 1995-05-31 KR KR1019960707048A patent/KR100397721B1/ko active IP Right Grant
- 1995-05-31 WO PCT/EP1995/002076 patent/WO1995034545A1/en active IP Right Grant
- 1995-05-31 EP EP01200801A patent/EP1114821B1/en not_active Expired - Lifetime
- 1995-05-31 PT PT01200801T patent/PT1114821E/pt unknown
- 1995-05-31 DK DK95921798T patent/DK0764157T3/da active
- 1995-05-31 SI SI9530579T patent/SI0764157T1/xx unknown
- 1995-05-31 ES ES01200801T patent/ES2207590T3/es not_active Expired - Lifetime
- 1995-05-31 HU HU9603415A patent/HUT76136A/hu not_active Application Discontinuation
- 1995-05-31 DK DK01200801T patent/DK1114821T3/da active
- 1995-05-31 SI SI9530691T patent/SI1114821T1/xx unknown
- 1995-05-31 SG SG1996008495A patent/SG67930A1/en unknown
- 1995-05-31 CN CNB951944134A patent/CN1174975C/zh not_active Expired - Lifetime
- 1995-05-31 DE DE69524871T patent/DE69524871T2/de not_active Expired - Lifetime
- 1995-06-02 US US08/460,151 patent/US5760074A/en not_active Expired - Lifetime
-
1996
- 1996-12-09 NO NO19965260A patent/NO315651B1/no not_active IP Right Cessation
- 1996-12-10 FI FI964936A patent/FI120686B/fi not_active IP Right Cessation
- 1996-12-10 OA OA60933A patent/OA10593A/en unknown
- 1996-12-10 BG BG101040A patent/BG63339B1/bg unknown
-
1998
- 1998-01-08 HK HK98100154A patent/HK1001286A1/xx not_active IP Right Cessation
-
2002
- 2002-01-10 HK HK02100192.4A patent/HK1039115B/zh not_active IP Right Cessation
-
2003
- 2003-01-23 JP JP2003014984A patent/JP2003238554A/ja active Pending
-
2005
- 2005-03-15 CY CY0500017A patent/CY2508B1/xx unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK1K | Patent expired |