NO301689B1 - Kontraseptivt preparat i form av en forpakning - Google Patents
Kontraseptivt preparat i form av en forpakning Download PDFInfo
- Publication number
- NO301689B1 NO301689B1 NO884230A NO884230A NO301689B1 NO 301689 B1 NO301689 B1 NO 301689B1 NO 884230 A NO884230 A NO 884230A NO 884230 A NO884230 A NO 884230A NO 301689 B1 NO301689 B1 NO 301689B1
- Authority
- NO
- Norway
- Prior art keywords
- progestin
- estrogen
- unit doses
- packaging according
- estradiol
- Prior art date
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- 238000002360 preparation method Methods 0.000 title claims description 34
- 239000003433 contraceptive agent Substances 0.000 title abstract description 9
- 230000002254 contraceptive effect Effects 0.000 title abstract description 9
- RJKFOVLPORLFTN-LEKSSAKUSA-N Progesterone Chemical class C1CC2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](C(=O)C)[C@@]1(C)CC2 RJKFOVLPORLFTN-LEKSSAKUSA-N 0.000 claims abstract description 116
- 239000000262 estrogen Substances 0.000 claims abstract description 93
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- 239000000583 progesterone congener Substances 0.000 claims abstract description 83
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- VIKNJXKGJWUCNN-XGXHKTLJSA-N norethisterone Chemical compound O=C1CC[C@@H]2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 VIKNJXKGJWUCNN-XGXHKTLJSA-N 0.000 claims description 41
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- 238000004806 packaging method and process Methods 0.000 claims description 28
- BFPYWIDHMRZLRN-SLHNCBLASA-N Ethinyl estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 BFPYWIDHMRZLRN-SLHNCBLASA-N 0.000 claims description 24
- 239000000186 progesterone Substances 0.000 claims description 22
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- BFPYWIDHMRZLRN-UHFFFAOYSA-N 17alpha-ethynyl estradiol Natural products OC1=CC=C2C3CCC(C)(C(CC4)(O)C#C)C4C3CCC2=C1 BFPYWIDHMRZLRN-UHFFFAOYSA-N 0.000 claims description 21
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- KIQQMECNKUGGKA-NMYWJIRASA-N norgestimate Chemical compound O/N=C/1CC[C@@H]2[C@H]3CC[C@](CC)([C@](CC4)(OC(C)=O)C#C)[C@@H]4[C@@H]3CCC2=C\1 KIQQMECNKUGGKA-NMYWJIRASA-N 0.000 claims description 13
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- JKKFKPJIXZFSSB-UHFFFAOYSA-N 1,3,5(10)-estratrien-17-one 3-sulfate Natural products OS(=O)(=O)OC1=CC=C2C3CCC(C)(C(CC4)=O)C4C3CCC2=C1 JKKFKPJIXZFSSB-UHFFFAOYSA-N 0.000 claims description 10
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- CHNXZKVNWQUJIB-CEGNMAFCSA-N ethisterone Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 CHNXZKVNWQUJIB-CEGNMAFCSA-N 0.000 claims description 4
- -1 norgeistrienon Chemical compound 0.000 claims description 4
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- 229910052623 talc Inorganic materials 0.000 description 1
- 230000001960 triggered effect Effects 0.000 description 1
- 239000011782 vitamin Substances 0.000 description 1
- 229940088594 vitamin Drugs 0.000 description 1
- 229930003231 vitamin Natural products 0.000 description 1
- 235000013343 vitamin Nutrition 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/24—Follicle-stimulating hormone [FSH]; Chorionic gonadotropins, e.g. HCG; Luteinising hormone [LH]; Thyroid-stimulating hormone [TSH]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CA 547744 CA1332228C (en) | 1987-09-24 | 1987-09-24 | Formulation and method for estrogen replacement therapy |
| CA000547743A CA1332227C (en) | 1987-09-24 | 1987-09-24 | Oral contraceptive formulation |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO884230D0 NO884230D0 (no) | 1988-09-23 |
| NO884230L NO884230L (no) | 1989-03-28 |
| NO301689B1 true NO301689B1 (no) | 1997-12-01 |
Family
ID=25671520
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO884230A NO301689B1 (no) | 1987-09-24 | 1988-09-23 | Kontraseptivt preparat i form av en forpakning |
Country Status (13)
| Country | Link |
|---|---|
| EP (2) | EP0309263B1 (ko) |
| JP (2) | JP3314207B2 (ko) |
| KR (1) | KR0170764B1 (ko) |
| CN (1) | CN1042296C (ko) |
| AT (1) | ATE209919T1 (ko) |
| AU (2) | AU630334B2 (ko) |
| DE (2) | DE3888269T2 (ko) |
| DK (1) | DK174071B1 (ko) |
| ES (2) | ES2061672T3 (ko) |
| FI (1) | FI101601B (ko) |
| HU (1) | HU214598B (ko) |
| NO (1) | NO301689B1 (ko) |
| NZ (1) | NZ226316A (ko) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3738620A1 (de) * | 1987-11-13 | 1989-05-24 | Luderschmidt Christoph | Verwendung von ethisterone zur topischen behandlung von akne oder androgenetischer alopezie |
| AU8166191A (en) * | 1990-08-10 | 1992-02-13 | Ortho Pharmaceutical Corporation | Method for treatment of bone wasting diseases |
| DE4104385C1 (ko) * | 1991-02-09 | 1992-08-13 | Marika Dr.Med. 6509 Framersheim De Ehrlich | |
| US5340586A (en) * | 1991-04-12 | 1994-08-23 | University Of Southern California | Methods and formulations for use in treating oophorectomized women |
| CA2152780A1 (en) * | 1992-12-28 | 1994-07-07 | Robert F. Casper | Transdermal hormone replacement therapy |
| WO1994016709A2 (en) * | 1993-01-19 | 1994-08-04 | Endorecherche Inc. | Therapeutic uses and delivery systems of dehydroepiandrosterone |
| NL9301562A (nl) * | 1993-09-09 | 1995-04-03 | Saturnus Ag | Preparaat voor substitutietherapie. |
| DE4344462C2 (de) * | 1993-12-22 | 1996-02-01 | Schering Ag | Zusammensetzung für die Empfängnisverhütung |
| DE4405591C1 (de) * | 1994-02-22 | 1995-07-20 | Hesch Rolf Dieter Prof Dr Med | Mittel zur postmenopausalen Hormonsubstitution |
| DE4405590C1 (de) * | 1994-02-22 | 1995-07-20 | Hesch Rolf Dieter Prof Dr Med | Mittel zur postmenopausalen Hormonbehandlung |
| US5612317A (en) * | 1994-08-04 | 1997-03-18 | Holick; Michael F. | Method for delivering estrogen |
| WO1998004268A1 (en) * | 1996-07-26 | 1998-02-05 | American Home Products Corporation | Oral contraceptive |
| FR2754179B1 (fr) * | 1996-10-08 | 1998-12-24 | Theramex | Nouvelle composition hormononale et son utilisation |
| WO2001030355A1 (fr) | 1999-10-25 | 2001-05-03 | Laboratoire Theramex | Medicament contraceptif a base d'un progestatif et d'un estrogene et son mode de preparation |
| EP1007052B1 (en) * | 1997-08-27 | 2004-10-13 | Ortho-McNeil Pharmaceutical, Inc. | Combinations of endometrial sparing progestins and endometrial atrophizing progestins with estrogens, in oral contraception |
| DE19739916C2 (de) * | 1997-09-11 | 2001-09-13 | Hesch Rolf Dieter | Verwendung einer Kombination aus einem Gestagen und einem Estrogen zur kontinuierlichen Ovulationshemmung und ggf. gleichzeitigen Behandlung und/oder Prophylaxe von Tumoren der Brustdrüsen |
| DE19831263A1 (de) * | 1998-07-11 | 2000-01-13 | Lohmann Therapie Syst Lts | Darreichungsform |
| DE19911799A1 (de) * | 1999-03-17 | 2000-09-28 | Lohmann Therapie Syst Lts | Sammelpackung zur Entnahme von befüllten Beuteln in vorgebener Reihenfolge |
| AU2005201151B2 (en) * | 1999-03-30 | 2008-01-10 | Jencap Research Ltd | Low dose estrogen interrupted hormone replacement therapy |
| CA2267743C (en) | 1999-03-30 | 2011-07-26 | Robert F. Casper | Low dose estrogen interrupted hormone replacement therapy |
| DE19934433A1 (de) | 1999-07-22 | 2001-01-25 | Merck Patent Gmbh | N-(Indolcarbonyl-)piperazinderivate |
| MXPA02002186A (es) * | 1999-08-31 | 2002-09-02 | Jenapharm Gmbh | Mesoprogestinas (moduladores del receptor de progesterona) como un componente de los anticonceptivos femeninos. |
| WO2001030356A1 (fr) | 1999-10-25 | 2001-05-03 | Laboratoire Theramex | Composition hormonale a base d'un progestatif et d'un estrogene et son utilisation |
| US20010034340A1 (en) * | 2000-03-20 | 2001-10-25 | American Home Products Corporation | Hormone replacement therapy |
| JP2005519961A (ja) * | 2002-03-11 | 2005-07-07 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 継続的スルファターゼ阻害プロゲストゲンホルモン補充療法 |
| UA82851C2 (en) * | 2002-08-28 | 2008-05-26 | Estrogen replacement regimen in menopausal women | |
| HUP0301981A2 (hu) * | 2003-06-30 | 2005-04-28 | Richter Gedeon Vegyészeti Gyár Rt. | Tiszta d-(17alfa)-13-etil-17-hidroxi-18,19-dinor-pregn-4-én-20-in-3-on-3E- és 3Z-oxim izomerek, valamint eljárás az izomer keverékek és a tiszta izomerek előállítására |
| US7816546B2 (en) | 2003-06-30 | 2010-10-19 | Richter Gedeon Vegyeszeti Gyar Rt. | Process for the synthesis of high purity d-(17α)-13-ethyl-17-hydroxy-18,19-dinorpregn-4-ene-20-yn-3-one-oxime |
| EP1535618A1 (en) * | 2003-11-26 | 2005-06-01 | Schering Aktiengesellschaft | Pharmaceutical preparation for continuous hormonal treatment over a period of longer than 21-28 days comprising two estrogen and/or progestin compositions |
| DE102004023984A1 (de) * | 2004-05-14 | 2005-12-08 | Hf Arzneimittelforschung Gmbh | Filmförmiges, oral zu verabreichendes Arzneimittel, enthaltend Estriol |
| JP5288796B2 (ja) * | 2004-07-07 | 2013-09-11 | ワイス・エルエルシー | 周期的プロゲスチンレジメン及びキット |
| CA2830984C (en) * | 2011-03-25 | 2020-02-11 | Universite Laval | Inhibitors of 17.beta.-hsd1, 17.beta.-hsd3 and 17.beta.-hsd10. |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3568828A (en) * | 1967-03-01 | 1971-03-09 | Squibb & Sons Inc | Modified sequential oral contraceptive |
| US3836651A (en) * | 1972-02-22 | 1974-09-17 | Biolog Concepts Inc | Novel oral contraceptive combination |
| DE2645307A1 (de) * | 1976-10-05 | 1978-04-06 | Schering Ag | Neue mittel und neue methoden zur behandlung klimakterischer ausfallerscheinungen |
| US4291028A (en) * | 1977-12-30 | 1981-09-22 | Nichols Vorys | Follicular phase estrogen or progestin with physiologic estrogen/progestin luteal phase replacement drug delivery system |
| US4292315A (en) * | 1977-12-30 | 1981-09-29 | Nichols Vorys | Follicular phase estrogen or progestin with physiologic estrogen/progestin luteal phase replacement drug delivery system |
| US4425339A (en) * | 1981-04-09 | 1984-01-10 | Syntex (U.S.A.) Inc. | Treatment of menopausal symptoms |
| AU581486B2 (en) * | 1985-12-30 | 1989-02-23 | Warner-Lambert Company | Graduated estrogen contraceptive |
| FR2589735A1 (fr) * | 1985-11-07 | 1987-05-15 | Beillon Xavier | Compositions anticonceptionnelles contenant un oestrogene et un progestatif |
| IE61236B1 (en) * | 1986-07-15 | 1994-10-19 | American Home Prod | Combination dosage form for pre-menopausal women |
-
1988
- 1988-09-23 DE DE3888269T patent/DE3888269T2/de not_active Expired - Lifetime
- 1988-09-23 NZ NZ226316A patent/NZ226316A/xx unknown
- 1988-09-23 AT AT93107794T patent/ATE209919T1/de not_active IP Right Cessation
- 1988-09-23 AU AU22760/88A patent/AU630334B2/en not_active Expired
- 1988-09-23 ES ES88308840T patent/ES2061672T3/es not_active Expired - Lifetime
- 1988-09-23 NO NO884230A patent/NO301689B1/no not_active IP Right Cessation
- 1988-09-23 EP EP88308840A patent/EP0309263B1/en not_active Expired - Lifetime
- 1988-09-23 ES ES93107794T patent/ES2169030T3/es not_active Expired - Lifetime
- 1988-09-23 DK DK198805296A patent/DK174071B1/da not_active IP Right Cessation
- 1988-09-23 EP EP93107794A patent/EP0559240B1/en not_active Expired - Lifetime
- 1988-09-23 FI FI884378A patent/FI101601B/fi not_active IP Right Cessation
- 1988-09-23 HU HU884989A patent/HU214598B/hu unknown
- 1988-09-23 DE DE3856508T patent/DE3856508T2/de not_active Expired - Lifetime
- 1988-09-24 JP JP23956688A patent/JP3314207B2/ja not_active Expired - Lifetime
- 1988-09-24 KR KR1019880012403A patent/KR0170764B1/ko not_active IP Right Cessation
- 1988-09-24 CN CN88107593A patent/CN1042296C/zh not_active Expired - Lifetime
-
1992
- 1992-12-24 AU AU30448/92A patent/AU3044892A/en not_active Abandoned
-
1998
- 1998-10-28 JP JP34482398A patent/JP3208482B2/ja not_active Expired - Lifetime
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK1K | Patent expired |