NO20091485L - Sulfonylpyrazol og sulfonylpyrazolin karboksamidinderivater som 5-HT6 antagonister - Google Patents

Sulfonylpyrazol og sulfonylpyrazolin karboksamidinderivater som 5-HT6 antagonister

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Publication number
NO20091485L
NO20091485L NO20091485A NO20091485A NO20091485L NO 20091485 L NO20091485 L NO 20091485L NO 20091485 A NO20091485 A NO 20091485A NO 20091485 A NO20091485 A NO 20091485A NO 20091485 L NO20091485 L NO 20091485L
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NO
Norway
Prior art keywords
disorders
attention deficit
disorder
compounds
antagonists
Prior art date
Application number
NO20091485A
Other languages
English (en)
Norwegian (no)
Inventor
Hiskias G Keizer
Cornelis G Kruse
Wouter I Iwema Bakker
Martina A W Van Der Neut
Arnold Van Loevezijn
Jan Zorgdrager
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Publication of NO20091485L publication Critical patent/NO20091485L/no

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K9/1605—Excipients; Inactive ingredients
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NO20091485A 2006-09-22 2009-04-16 Sulfonylpyrazol og sulfonylpyrazolin karboksamidinderivater som 5-HT6 antagonister NO20091485L (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US84640606P 2006-09-22 2006-09-22
EP06121087 2006-09-22
US90286507P 2007-02-23 2007-02-23
EP07102965 2007-02-23
PCT/EP2007/059944 WO2008034863A2 (en) 2006-09-22 2007-09-20 Sulfonylpyrazoline carboxamidine derivatives as 5-ht6 antagonists

Publications (1)

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NO20091485L true NO20091485L (no) 2009-04-17

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AR062907A1 (es) 2006-09-22 2008-12-17 Solvay Pharm Bv Derivados de sulfonilpirazol y sulfonilpirazolincarboxamidina como antagonistas de 5-ht6
AR070898A1 (es) 2008-03-18 2010-05-12 Solvay Pharm Bv Derivados de arilsulfonil pirazolin carboxamidina como antagonistas de 5-ht6
AR079935A1 (es) 2010-01-29 2012-02-29 Abbott Healthcare Products Bv Sintesis de derivados de pirazolin carboxamidina sustituida
WO2013055386A2 (en) * 2011-10-03 2013-04-18 The University Of Utah Research Foundation Application of 5-ht6 receptor antagonists for the alleviation of cognitive deficits of down syndrome
FR2999574B1 (fr) * 2012-12-18 2014-12-05 Isochem Sa Procede de synthese des hydrazines endocycliques
ES2674476T3 (es) 2013-07-25 2018-07-02 Uniwersytet Jagiellonski Derivados de pirroloquinolina como antagonistas de 5-HT6, método de preparación y uso de los mismos
EP3109237A1 (en) * 2015-06-22 2016-12-28 AnaMar AB Novel 5-ht2 antagonists
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EP2069310A2 (en) 2009-06-17
WO2008034863A3 (en) 2008-05-08
EA200970310A1 (ru) 2009-10-30
IL197232A0 (en) 2009-12-24
KR20090060356A (ko) 2009-06-11
AR062907A1 (es) 2008-12-17
ATE537149T1 (de) 2011-12-15
US8722887B2 (en) 2014-05-13
SA07280510B1 (ar) 2012-02-07
KR101433745B1 (ko) 2014-08-25
PT2069310E (pt) 2012-02-28
CA2662484C (en) 2015-06-23
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IL197232A (en) 2015-11-30
JP2010504302A (ja) 2010-02-12
WO2008034863A2 (en) 2008-03-27
JP5225280B2 (ja) 2013-07-03
US20140303372A1 (en) 2014-10-09
CN101679279B (zh) 2013-11-13
MX2009003183A (es) 2009-04-03
SI2069310T1 (sl) 2012-02-29
US7728018B2 (en) 2010-06-01
US20080311179A1 (en) 2008-12-18
CY1112418T1 (el) 2015-12-09
HRP20120215T1 (hr) 2012-04-30
TWI428334B (zh) 2014-03-01
BRPI0716860A2 (pt) 2013-10-15
EP2069310B1 (en) 2011-12-14
TW200821299A (en) 2008-05-16
EA021543B1 (ru) 2015-07-30
AU2007298987A1 (en) 2008-03-27
DK2069310T3 (da) 2012-03-19
PL2069310T3 (pl) 2012-05-31
ES2377996T3 (es) 2012-04-04
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