NO20083980L - 4-(3-benzoylaminofenyl)-6,7-dimetoksy-2-metylaminokinazolinderivat - Google Patents

4-(3-benzoylaminofenyl)-6,7-dimetoksy-2-metylaminokinazolinderivat

Info

Publication number
NO20083980L
NO20083980L NO20083980A NO20083980A NO20083980L NO 20083980 L NO20083980 L NO 20083980L NO 20083980 A NO20083980 A NO 20083980A NO 20083980 A NO20083980 A NO 20083980A NO 20083980 L NO20083980 L NO 20083980L
Authority
NO
Norway
Prior art keywords
metylaminokinazolinderivat
benzoylaminofenyl
dimethoxy
substituted
formula
Prior art date
Application number
NO20083980A
Other languages
English (en)
Other versions
NO332976B1 (no
Inventor
Kazuki Miyazaki
Kazutomi Kusano
Yasutaka Takase
Osamu Asano
Manabu Shirato
Hisashi Wakita
Naoto Ishi
Takao Saeki
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Publication of NO20083980L publication Critical patent/NO20083980L/no
Publication of NO332976B1 publication Critical patent/NO332976B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/84—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

En forbindelse representert ved formel (I) nedenfor, et salt derav eller et hydrat av hvilke som helst derav, som er i. stand til effektiv undertrykking av kløe ved atopisk sykdom og lignende [I formelen representerer R en hydroksyl, en Ci.6 alkoksygruppe som kan være substituert med en Ci-6 alkoksygruppe, eller en aminogruppe som kan være substituert med en Ci.6 alkylgruppe.]
NO20083980A 2006-02-21 2008-09-18 Kinazolinderivater samt farmasoytisk preparat NO332976B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US77462006P 2006-02-21 2006-02-21
JP2006043273 2006-02-21
PCT/JP2007/053066 WO2007097317A1 (ja) 2006-02-21 2007-02-20 ４－（３－ベンゾイルアミノフェニル）－６，７－ジメトキシ－２－メチルアミノキナゾリン誘導体

Publications (2)

Publication Number Publication Date
NO20083980L true NO20083980L (no) 2008-11-20
NO332976B1 NO332976B1 (no) 2013-02-11

Family

ID=41429386

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083980A NO332976B1 (no) 2006-02-21 2008-09-18 Kinazolinderivater samt farmasoytisk preparat

Country Status (11)

Country Link
US (1) US7939540B2 (no)
EP (1) EP1992622B1 (no)
CN (1) CN101389612B (no)
AU (1) AU2007218725B2 (no)
CA (1) CA2637573C (no)
MX (1) MX2008010774A (no)
NO (1) NO332976B1 (no)
PL (1) PL1992622T3 (no)
SA (1) SA07280059B1 (no)
WO (1) WO2007097317A1 (no)
ZA (1) ZA200805756B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007097317A1 (ja) 2006-02-21 2007-08-30 Eisai R & D Management Co., Ltd. ４－（３－ベンゾイルアミノフェニル）－６，７－ジメトキシ－２－メチルアミノキナゾリン誘導体
WO2008099887A1 (ja) * 2007-02-16 2008-08-21 Eisai R & D Management Co., Ltd. メチル ｎ－［３－（６，７－ジメトキシ－２－メチルアミノキナゾリン－４－イル）フェニル］テレフタラミックアシッドの結晶、非晶質体または塩
CN101687818B (zh) * 2007-02-19 2012-08-22 卫材R&D管理有限公司 甲基n-[3-(6,7-二甲氧基-2-甲氨基喹唑啉-4-基)苯基]对氨羰基苯甲酸的结晶、无定形物或盐
EP2189450B1 (en) 2007-08-17 2011-12-21 Eisai R&D Management Co., Ltd. Method for producing quinazoline derivative
JP5060561B2 (ja) 2007-08-17 2012-10-31 エーザイ・アール・アンド・ディー・マネジメント株式会社 新規外用剤
WO2014133020A1 (ja) * 2013-02-28 2014-09-04 エーザイ・アール・アンド・ディー・マネジメント株式会社 呼吸器疾患の予防治療剤
BR112018075202A2 (pt) * 2016-06-07 2019-03-19 Dermavant Sciences GmbH formulação tópica e método de tratamento de uma condição dermatológica em um sujeito
JP2021505621A (ja) 2017-12-07 2021-02-18 ダーマヴァント サイエンシーズ ゲーエムベーハー Ｐｄｅ−４阻害剤の局所軟膏製剤および皮膚状態の治療におけるそれらの使用

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2099112T3 (es) 1990-09-04 1997-05-16 Fujisawa Pharmaceutical Co Pomadas que contienen un compuesto triciclico.
US6115962A (en) * 1994-03-31 2000-09-12 Southpac Trust International, Inc. Sleeve for covering a flower pot
JP3466305B2 (ja) 1994-12-12 2003-11-10 久光製薬株式会社 溶解剤および該溶解剤を含有する外用製剤
AU4342997A (en) 1996-09-13 1998-04-02 Sugen, Inc. Use of quinazoline derivatives for the manufacture of a medicament in the reatment of hyperproliferative skin disorders
AR015966A1 (es) 1997-10-17 2001-05-30 Smithkline Beecham Corp Uso de un compuesto inhibidor de pde4 para la preparacion de un medicamento util para el tratamiento de prurito
JPH11209350A (ja) * 1998-01-26 1999-08-03 Eisai Co Ltd 含窒素複素環誘導体およびその医薬
JP3373838B2 (ja) 1999-10-25 2003-02-04 山之内製薬株式会社 ナフチリジン誘導体
AR029185A1 (es) * 1999-10-25 2003-06-18 Yamanouchi Pharma Co Ltd Derivado de naftiridina
NZ537308A (en) 2002-05-28 2009-09-25 Nycomed Gmbh Ophthalmological use of roflumilast for the treatment of diseases of the eye
US20040038958A1 (en) 2002-07-11 2004-02-26 Chris Rundfeldt Topical treatment of skin diseases
JP4387717B2 (ja) 2003-07-11 2009-12-24 株式会社資生堂 油中水型皮膚外用医薬品製剤
JP2005047909A (ja) 2003-07-17 2005-02-24 Santen Pharmaceut Co Ltd ピペリジン誘導体を有効成分とする掻痒治療剤
EP1647274A4 (en) * 2003-07-17 2008-12-10 Ono Pharmaceutical Co REMEDY AGAINST PRURIT COMPRISING A PIPERIDINE DERIVATIVE AS AN ACTIVE INGREDIENT
WO2005082865A1 (ja) * 2004-02-27 2005-09-09 Astellas Pharma Inc. 縮合二環性ピリミジン誘導体
JP2008137892A (ja) 2005-03-04 2008-06-19 Eisai Co Ltd 止痒剤
WO2007097317A1 (ja) 2006-02-21 2007-08-30 Eisai R & D Management Co., Ltd. ４－（３－ベンゾイルアミノフェニル）－６，７－ジメトキシ－２－メチルアミノキナゾリン誘導体
WO2008099887A1 (ja) 2007-02-16 2008-08-21 Eisai R & D Management Co., Ltd. メチル ｎ－［３－（６，７－ジメトキシ－２－メチルアミノキナゾリン－４－イル）フェニル］テレフタラミックアシッドの結晶、非晶質体または塩

Also Published As

Publication number Publication date
AU2007218725A1 (en) 2007-08-30
US7939540B2 (en) 2011-05-10
AU2007218725B2 (en) 2011-12-01
CN101389612B (zh) 2011-09-21
CA2637573A1 (en) 2007-08-30
ZA200805756B (en) 2009-04-29
CA2637573C (en) 2013-07-02
SA07280059B1 (ar) 2010-11-02
MX2008010774A (es) 2008-09-01
CN101389612A (zh) 2009-03-18
US20070299094A1 (en) 2007-12-27
WO2007097317A1 (ja) 2007-08-30
EP1992622B1 (en) 2011-07-27
NO332976B1 (no) 2013-02-11
PL1992622T3 (pl) 2012-01-31
EP1992622A4 (en) 2009-05-06
EP1992622A1 (en) 2008-11-19

Similar Documents

Publication Publication Date Title
NO20083980L (no) 4-(3-benzoylaminofenyl)-6,7-dimetoksy-2-metylaminokinazolinderivat
NO20076066L (no) Oksadiazolderivater som DGAT-inhibitorer
WO2006062984A3 (en) Inhibitors of protein kinases
NO20076059L (no) 2,4-Diamino-pyrimidiner anvendt som aurorainhibitorer
NO20076450L (no) Heterosykliske forbindelser som nikotinsyrereseptoragonister for behandling av dyslipidemi
NO20070933L (no) Indazoler anvendbare i behandling av kardiovaskulaere sykdommer
WO2008022286A3 (en) Small molecule inhibitors of kynurenine-3-monooxygenase
WO2009006389A3 (en) Pyrimidine derivatives useful as raf kinase inhibitors
NO20082673L (no) Nye 2-amino-imidazol-4-on forbindelser og deres anvendelse i fremstilling av et medikament som skal brukes til behandling av kognitiv svekkelse, Alzheimers sykdom, neurodegenerasjon og demens
NO20081315L (no) Benzokinazolinderivater og deres anvendelse ved behandling av benlidelser
WO2008011557A3 (en) Heteroaryl inhibitors of rho kinase
NO20084418L (no) Azolopyridin-3-on derivater som inhibitorer av endoteliallipase
EP2085389A4 (en) NOVEL 1,2-DIHYDROQUINOLINE DERIVATIVE COMPRISING AS SUBSTITUENTS A LOWER ALKYL-CARBONYLOXY GROUP (PHENYL-SUBSTITUTED OR HETEROCYCLIC SUBSTITUTED) AND A PHENYL GROUP LINKED BY AN ESTER
ATE536349T1 (de) In der 2-stellung durch phenyl substituierte 1h- benzimidazol-4-carbonsäureamide sind wirksame parp-inhibitoren
NO20072963L (no) 5-substituerte kinolin- og isokinolinderivater, fremgangsmate for deres fremstilling og deres anvendelse som betennelseshemmere
NO20073791L (no) Pyrazolylaminopyridinderivater anvendbare som kinaseinhibitorer
NO20074763L (no) (1,5-difenyl-1H-pyrazol-3-yl)oksadiazolderivater, fremgangsmate ved fremstilling derav og anvendelse av samme i terapi
WO2006103277A3 (en) 2 , 4 , 5-substituted piperidines as renin inhibitors
NO20070445L (no) Pyrimidinderivater.
WO2007109105A3 (en) Flavivirus inhibition by sultams and related compounds
WO2008057775A3 (en) Heterocyclic amide compounds useful as kinase inhibitors
WO2007032028A8 (en) Thiazolinones and oxazolinones and their use as ptp1b inhibitors
NO20074311L (no) Kinazolinderivat med tyrosinkinase-inhiberendeaktivitet
WO2007126900A3 (en) Antifungal agents
NO20073941L (no) Dihydroimidazotiazolderivater

Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees