NO20070484L - Sammenspleisede pyrimidinderivater og sammensetninger derav som CXCR3 reseptormodulatorer, anvendbare ved forebygging og behandling av inflammatoriske og immunregulatoriske lidelser og sykdommer. - Google Patents
Sammenspleisede pyrimidinderivater og sammensetninger derav som CXCR3 reseptormodulatorer, anvendbare ved forebygging og behandling av inflammatoriske og immunregulatoriske lidelser og sykdommer.Info
- Publication number
- NO20070484L NO20070484L NO20070484A NO20070484A NO20070484L NO 20070484 L NO20070484 L NO 20070484L NO 20070484 A NO20070484 A NO 20070484A NO 20070484 A NO20070484 A NO 20070484A NO 20070484 L NO20070484 L NO 20070484L
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58390104P | 2004-06-28 | 2004-06-28 | |
PCT/US2005/023251 WO2006004915A1 (fr) | 2004-06-28 | 2005-06-28 | Derives de pyrimidine fusionnes et compositions sur leur base, utilises en tant que modulateurs du recepteur de cxcr3, utiles dans la prevention et le traitement de maladies et troubles inflammatoires ou immunoregulateurs |
Publications (1)
Publication Number | Publication Date |
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NO20070484L true NO20070484L (no) | 2007-03-26 |
Family
ID=35197976
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20070484A NO20070484L (no) | 2004-06-28 | 2007-01-25 | Sammenspleisede pyrimidinderivater og sammensetninger derav som CXCR3 reseptormodulatorer, anvendbare ved forebygging og behandling av inflammatoriske og immunregulatoriske lidelser og sykdommer. |
Country Status (19)
Country | Link |
---|---|
US (1) | US7939538B2 (fr) |
EP (1) | EP1771447A1 (fr) |
JP (1) | JP2008504301A (fr) |
KR (1) | KR20070045203A (fr) |
CN (1) | CN101006088A (fr) |
AR (1) | AR049558A1 (fr) |
AU (1) | AU2005260620A1 (fr) |
BR (1) | BRPI0512703A (fr) |
CA (1) | CA2572083A1 (fr) |
EA (1) | EA011439B1 (fr) |
EC (1) | ECSP077212A (fr) |
IL (1) | IL180327A0 (fr) |
MA (1) | MA28755B1 (fr) |
MX (1) | MX2007000051A (fr) |
NO (1) | NO20070484L (fr) |
TN (1) | TNSN06430A1 (fr) |
TW (1) | TW200611699A (fr) |
WO (1) | WO2006004915A1 (fr) |
ZA (1) | ZA200700752B (fr) |
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KR101129868B1 (ko) * | 2006-10-04 | 2012-04-12 | 화이자 프로덕츠 인코포레이티드 | 칼슘 수용체 길항제로서의 피리도[4,3-d]피리미딘-4(3H)-온 유도체 |
NZ581606A (en) * | 2007-05-03 | 2012-06-29 | Intermune Inc | Novel macrocyclic inhibitors of hepatitis c virus replication |
AP2009005057A0 (en) | 2007-05-10 | 2009-12-31 | Array Biopharma Inc | Novel peptide inhibitors of hepatitis c virus replication |
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EA201071034A1 (ru) * | 2008-04-15 | 2011-06-30 | Интермьюн, Инк. | Новые макроциклические ингибиторы репликаций вируса гепатита с |
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CN106456628A (zh) | 2014-03-19 | 2017-02-22 | 无限药品股份有限公司 | 用于治疗PI3K‑γ介导的障碍的杂环化合物 |
WO2016054491A1 (fr) | 2014-10-03 | 2016-04-07 | Infinity Pharmaceuticals, Inc. | Composés hétérocycliques et leurs utilisations |
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TW201815787A (zh) | 2016-09-23 | 2018-05-01 | 美商基利科學股份有限公司 | 磷脂醯肌醇3-激酶抑制劑 |
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US20040242498A1 (en) | 2003-02-27 | 2004-12-02 | Collins Tassie L. | CXCR3 antagonists |
US7271271B2 (en) * | 2004-06-28 | 2007-09-18 | Amgen Sf, Llc | Imidazolo-related compounds, compositions and methods for their use |
US7939538B2 (en) | 2004-06-28 | 2011-05-10 | Amgen Inc. | Compounds, compositions and methods for prevention and treatment of inflammatory and immunoregulatory disorders and diseases |
US7375102B2 (en) * | 2004-06-28 | 2008-05-20 | Amgen Sf, Llc | Tetrahydroquinazolin-4(3H)-one-related and tetrahydropyrido[2,3-D]pyrimidin-4(3H)-one-related compounds, compositions and methods for their use |
WO2006023381A1 (fr) * | 2004-08-16 | 2006-03-02 | Taigen Biotechnology | Composés de type pyrimidinone |
JP2008546843A (ja) * | 2005-06-27 | 2008-12-25 | アムゲン インコーポレイティッド | 抗炎症性アリールニトリル化合物 |
-
2005
- 2005-06-27 US US11/168,005 patent/US7939538B2/en not_active Expired - Fee Related
- 2005-06-28 CN CNA2005800277780A patent/CN101006088A/zh active Pending
- 2005-06-28 TW TW094121708A patent/TW200611699A/zh unknown
- 2005-06-28 AR ARP050102670A patent/AR049558A1/es not_active Application Discontinuation
- 2005-06-28 BR BRPI0512703-3A patent/BRPI0512703A/pt not_active IP Right Cessation
- 2005-06-28 EA EA200700169A patent/EA011439B1/ru not_active IP Right Cessation
- 2005-06-28 WO PCT/US2005/023251 patent/WO2006004915A1/fr active Application Filing
- 2005-06-28 KR KR1020077002012A patent/KR20070045203A/ko not_active Application Discontinuation
- 2005-06-28 AU AU2005260620A patent/AU2005260620A1/en not_active Abandoned
- 2005-06-28 JP JP2007518379A patent/JP2008504301A/ja active Pending
- 2005-06-28 ZA ZA200700752A patent/ZA200700752B/xx unknown
- 2005-06-28 MX MX2007000051A patent/MX2007000051A/es not_active Application Discontinuation
- 2005-06-28 EP EP05789126A patent/EP1771447A1/fr not_active Withdrawn
- 2005-06-28 CA CA002572083A patent/CA2572083A1/fr not_active Abandoned
-
2006
- 2006-12-25 IL IL180327A patent/IL180327A0/en unknown
- 2006-12-26 TN TNP2006000430A patent/TNSN06430A1/en unknown
-
2007
- 2007-01-25 NO NO20070484A patent/NO20070484L/no not_active Application Discontinuation
- 2007-01-29 MA MA29639A patent/MA28755B1/fr unknown
- 2007-01-29 EC EC2007007212A patent/ECSP077212A/es unknown
Also Published As
Publication number | Publication date |
---|---|
IL180327A0 (en) | 2007-07-04 |
MA28755B1 (fr) | 2007-07-02 |
MX2007000051A (es) | 2007-05-11 |
CA2572083A1 (fr) | 2006-01-12 |
BRPI0512703A (pt) | 2008-04-01 |
AR049558A1 (es) | 2006-08-16 |
US7939538B2 (en) | 2011-05-10 |
TNSN06430A1 (en) | 2008-02-22 |
CN101006088A (zh) | 2007-07-25 |
US20060069099A1 (en) | 2006-03-30 |
EA200700169A1 (ru) | 2007-08-31 |
WO2006004915A1 (fr) | 2006-01-12 |
ZA200700752B (en) | 2008-09-25 |
AU2005260620A1 (en) | 2006-01-12 |
KR20070045203A (ko) | 2007-05-02 |
JP2008504301A (ja) | 2008-02-14 |
ECSP077212A (es) | 2007-03-29 |
TW200611699A (en) | 2006-04-16 |
EA011439B1 (ru) | 2009-02-27 |
EP1771447A1 (fr) | 2007-04-11 |
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