NO20065122L - 1,1'-(1,2-etyndiyl)bis-benzenderivater som PTP 1-B-hemmere - Google Patents

1,1'-(1,2-etyndiyl)bis-benzenderivater som PTP 1-B-hemmere

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Publication number
NO20065122L
NO20065122L NO20065122A NO20065122A NO20065122L NO 20065122 L NO20065122 L NO 20065122L NO 20065122 A NO20065122 A NO 20065122A NO 20065122 A NO20065122 A NO 20065122A NO 20065122 L NO20065122 L NO 20065122L
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NO
Norway
Prior art keywords
ptp
ethynthyl
inhibitors
bis
benzene derivatives
Prior art date
Application number
NO20065122A
Other languages
English (en)
Norwegian (no)
Inventor
Agnes Bombrun
Dominique Swinnen
Jerome Gonzalez
Catherine Jorand-Lebrun
Patrick Gerber
Original Assignee
Applied Research Systems
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Filing date
Publication date
Application filed by Applied Research Systems filed Critical Applied Research Systems
Publication of NO20065122L publication Critical patent/NO20065122L/no

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NO20065122A 2004-04-07 2006-11-07 1,1'-(1,2-etyndiyl)bis-benzenderivater som PTP 1-B-hemmere NO20065122L (no)

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EP1904048B1 (fr) * 2005-07-15 2011-11-23 Merck Serono SA Inhibiteurs glepp-1 dans le traitement de troubles autoimmunes et/ou inflammatoires
AU2015210454B2 (en) * 2005-12-23 2016-10-27 Ariad Pharmaceuticals, Inc. Bicyclic heteroaryl compounds
SI2495016T1 (sl) 2005-12-23 2020-04-30 Ariad Pharmaceuticals, Inc. Biciklične heteroarilne spojine
KR20090010186A (ko) * 2006-04-13 2009-01-29 주식회사 뉴로테크 살리실산 유도체 화합물 및 이를 포함하는 약학 조성물
EA200870514A1 (ru) * 2006-05-08 2009-04-28 Ариад Фармасьютикалз, Инк. Ацетиленовые гетероарильные соединения
KR101441365B1 (ko) 2006-05-08 2014-09-18 어리어드 파마슈티칼스, 인코포레이티드 모노시클릭 헤테로아릴 화합물
US8853392B2 (en) 2007-06-03 2014-10-07 Vanderbilt University Benzamide mGluR5 positive allosteric modulators and methods of making and using same
JP2009108036A (ja) * 2007-09-28 2009-05-21 Fujifilm Corp 新規アセチレン化合物、その製造方法、それを構成単位として含むポリマー、該化合物及び／又は該ポリマーを含む組成物、該組成物を硬化させてなる硬化物
WO2009120783A1 (fr) * 2008-03-25 2009-10-01 The Johns Hopkins University Inhibiteurs à haute affinité de protéase ns3/4a du virus de l'hépatite c
WO2010056311A1 (fr) 2008-11-12 2010-05-20 Ariad Pharmaceuticals, Inc. Pyrazinopyrazines et dérivés utiles comme inhibiteurs de kinases
WO2010059913A2 (fr) * 2008-11-20 2010-05-27 Dr. Reddy's Laboratories Ltd. Préparation de rasagiline et de ses sels
WO2013029555A1 (fr) * 2011-09-01 2013-03-07 天津医科大学附属肿瘤医院 Dérivés de lavendustine a, leur procédé de préparation et leur utilisation
CA3022250A1 (fr) 2012-12-12 2014-06-12 Ariad Pharmaceuticals, Inc. Formes cristallines de 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperaz in-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide mono hydrochloride
WO2015155738A2 (fr) 2014-04-09 2015-10-15 Christopher Rudd Utilisation d'inhibiteurs ou d'activateurs de gsk -3 qui modulent l'expression de pd -1 ou de t-bet pour moduler l'immunité due aux lymphocytes t
WO2016001452A1 (fr) 2014-07-04 2016-01-07 Universität Zürich Composés, destinés plus particulièrement à être utilisés dans le traitement d'une maladie ou d'une pathologie pour laquelle un inhibiteur du bromodomaine est indiqué
CN110291383B (zh) * 2017-02-23 2021-12-28 株式会社Ihi Oh自由基检测探测器、oh自由基测定装置以及oh自由基测定方法
WO2020040831A1 (fr) 2018-08-20 2020-02-27 Perlara Pbc Méthodes pour traiter des troubles congénitaux de la glycosylation
US20230365945A1 (en) 2020-09-18 2023-11-16 Iucf-Hyu (Industry-University Cooperation Foundation Hanyang University) Ptpsigma-fc fusion protein and pharmaceutical composition comprising same

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WO2005097773A1 (fr) 2005-10-20
AR048465A1 (es) 2006-04-26
IL178425A (en) 2012-02-29
EP1756081A1 (fr) 2007-02-28
BRPI0508790A (pt) 2007-09-04
CN1997638B (zh) 2011-07-06
JP2007532514A (ja) 2007-11-15
JP5043645B2 (ja) 2012-10-10
KR20070008675A (ko) 2007-01-17
MXPA06011678A (es) 2007-01-23
CN1997638A (zh) 2007-07-11
CA2560648C (fr) 2013-01-22
HK1102597A1 (en) 2007-11-30
EA011930B1 (ru) 2009-06-30
AU2005231980A1 (en) 2005-10-20
EA200601869A1 (ru) 2007-04-27
KR101194968B1 (ko) 2012-10-25
CA2560648A1 (fr) 2005-10-20
IL178425A0 (en) 2007-02-11
UA85405C2 (ru) 2009-01-26
US20090029903A1 (en) 2009-01-29
US7947851B2 (en) 2011-05-24
AU2005231980B2 (en) 2011-09-08

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