NO20063841L - Krystallinske polymorfer av en CXC-kjemokinreseptorligand - Google Patents

Krystallinske polymorfer av en CXC-kjemokinreseptorligand

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Publication number
NO20063841L
NO20063841L NO20063841A NO20063841A NO20063841L NO 20063841 L NO20063841 L NO 20063841L NO 20063841 A NO20063841 A NO 20063841A NO 20063841 A NO20063841 A NO 20063841A NO 20063841 L NO20063841 L NO 20063841L
Authority
NO
Norway
Prior art keywords
chemokine receptor
cxc chemokine
crystalline polymorphs
receptor ligand
methods
Prior art date
Application number
NO20063841A
Other languages
English (en)
Inventor
Michael Dwyer
Mengwei Hu
Younong Yu
Arthur G Taveras
Agnes Kim-Meade
Jianguo Yin
Xiaoyong Fu
Timothy Mcallister
Shuyi Zhang
Kevin Klopfer
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34837390&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20063841(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of NO20063841L publication Critical patent/NO20063841L/no

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Abstract

Den foreliggende oppfinnelse vedrører fire forskjellige krystallinske polymorfer av monohydrat av forbindelse A som har den følgende kjemiske stnikturformel (A). Disse fire polymorfe formene, her henvist til som formene I, II, III og IV, er aktive som CXC-kjemokinreseptorligander. Oppfinnelsen er videre rettet mot preparater, fremgangsmåter for behandling og fremgangsmåter for syntese av disse polymorfe formene.
NO20063841A 2004-01-30 2006-08-29 Krystallinske polymorfer av en CXC-kjemokinreseptorligand NO20063841L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54048704P 2004-01-30 2004-01-30
PCT/US2005/003414 WO2005075447A1 (en) 2004-01-30 2005-01-28 Crystalline polymorphs of a cxc-chemokine receptor ligand

Publications (1)

Publication Number Publication Date
NO20063841L true NO20063841L (no) 2006-10-27

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ID=34837390

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20063841A NO20063841L (no) 2004-01-30 2006-08-29 Krystallinske polymorfer av en CXC-kjemokinreseptorligand

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US (2) US20050192345A1 (no)
EP (1) EP1723131B1 (no)
JP (2) JP2007519751A (no)
KR (1) KR100883476B1 (no)
CN (1) CN1914187B (no)
AR (1) AR047739A1 (no)
AT (1) ATE478061T1 (no)
AU (1) AU2005210504B2 (no)
BR (1) BRPI0507329A (no)
CA (1) CA2554709C (no)
CO (1) CO5700731A2 (no)
DE (1) DE602005022986D1 (no)
EC (1) ECSP066733A (no)
ES (1) ES2349788T3 (no)
HK (1) HK1091496A1 (no)
IL (1) IL177033A0 (no)
MX (1) MXPA06008599A (no)
MY (1) MY144657A (no)
NO (1) NO20063841L (no)
NZ (1) NZ548499A (no)
PE (1) PE20051093A1 (no)
PL (1) PL380997A1 (no)
RU (1) RU2388756C2 (no)
TW (1) TW200536848A (no)
WO (1) WO2005075447A1 (no)
ZA (1) ZA200606295B (no)

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ES2655942T3 (es) 2011-09-02 2018-02-22 Novartis Ag Sal de colina de un compuesto anti-inflamatorio de ciclobutenodiona sustituida
US8865723B2 (en) 2012-10-25 2014-10-21 Tetra Discovery Partners Llc Selective PDE4 B inhibition and improvement in cognition in subjects with brain injury
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TWI734715B (zh) 2015-11-19 2021-08-01 美商卡默森屈有限公司 趨化因子受體調節劑
TWI724056B (zh) 2015-11-19 2021-04-11 美商卡默森屈有限公司 Ｃｘｃｒ２抑制劑
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DE602005022986D1 (de) 2010-09-30
ZA200606295B (en) 2008-02-27
ATE478061T1 (de) 2010-09-15
US20050192345A1 (en) 2005-09-01
IL177033A0 (en) 2006-12-10
MXPA06008599A (es) 2006-08-28
RU2006131050A (ru) 2008-03-10
US20080279822A1 (en) 2008-11-13
CN1914187A (zh) 2007-02-14
EP1723131A1 (en) 2006-11-22
CA2554709A1 (en) 2005-08-18
PE20051093A1 (es) 2006-01-16
ES2349788T3 (es) 2011-01-11
KR20060128981A (ko) 2006-12-14
CO5700731A2 (es) 2006-11-30
ECSP066733A (es) 2006-11-24
PL380997A1 (pl) 2007-04-16
BRPI0507329A (pt) 2007-07-03
CN1914187B (zh) 2012-01-25
HK1091496A1 (en) 2007-01-19
RU2388756C2 (ru) 2010-05-10
AU2005210504B2 (en) 2009-01-08
AU2005210504A1 (en) 2005-08-18
JP2011042692A (ja) 2011-03-03
AR047739A1 (es) 2006-02-15
US8207221B2 (en) 2012-06-26
JP2007519751A (ja) 2007-07-19
CA2554709C (en) 2011-11-15
NZ548499A (en) 2010-06-25
EP1723131B1 (en) 2010-08-18
MY144657A (en) 2011-10-31
TW200536848A (en) 2005-11-16
WO2005075447A1 (en) 2005-08-18
KR100883476B1 (ko) 2009-02-16

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