NO20062549L - Substituerte arylpyrazoler anti-paresittmidlert - Google Patents

Substituerte arylpyrazoler anti-paresittmidlert

Info

Publication number
NO20062549L
NO20062549L NO20062549A NO20062549A NO20062549L NO 20062549 L NO20062549 L NO 20062549L NO 20062549 A NO20062549 A NO 20062549A NO 20062549 A NO20062549 A NO 20062549A NO 20062549 L NO20062549 L NO 20062549L
Authority
NO
Norway
Prior art keywords
paresite
agent
substituted arylpyrazoles
arylpyrazoles
substituted
Prior art date
Application number
NO20062549A
Other languages
English (en)
Inventor
Nigel Derek Arthur Walshe
David Morris Gethin
Nathan Anthony Logan Chubb
Denis Billen
Kim Thomas Hall
Lee Richard Roberts
Original Assignee
Zoetis Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zoetis Llc filed Critical Zoetis Llc
Publication of NO20062549L publication Critical patent/NO20062549L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C07D231/40—Acylated on said nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Det beskrives 1 -aryl-4-syklopropylpyrazoler hvor der er minst ett fluor festet til syklopropylringen, materialer som omfatter slike forbindelser, fremgangsmåter for deres syntese og anvendelse av slike midler som anti-parasittmidler.
NO20062549A 2003-12-18 2006-06-02 Substituerte arylpyrazoler anti-paresittmidlert NO20062549L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0329314.9A GB0329314D0 (en) 2003-12-18 2003-12-18 Substituted arylpyrazoles
PCT/IB2004/004193 WO2005060749A1 (en) 2003-12-18 2004-12-15 Substituted arylpyrazoles as parasiticidal agents

Publications (1)

Publication Number Publication Date
NO20062549L true NO20062549L (no) 2006-06-27

Family

ID=30471290

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20062549A NO20062549L (no) 2003-12-18 2006-06-02 Substituerte arylpyrazoler anti-paresittmidlert

Country Status (33)

Country Link
US (1) US7435753B2 (no)
EP (1) EP1705989B8 (no)
JP (2) JP4805164B2 (no)
KR (1) KR100815637B1 (no)
CN (1) CN100377645C (no)
AR (1) AR046942A1 (no)
AT (1) ATE413809T1 (no)
AU (1) AU2004304717B2 (no)
BR (1) BRPI0417810B8 (no)
CA (1) CA2549479C (no)
CY (1) CY1108649T1 (no)
DE (1) DE602004017782D1 (no)
DK (1) DK1705989T3 (no)
EA (1) EA010740B1 (no)
ES (1) ES2315724T3 (no)
GB (1) GB0329314D0 (no)
HK (1) HK1096824A1 (no)
IL (1) IL175992A0 (no)
IS (1) IS8492A (no)
MA (1) MA28269A1 (no)
MX (1) MXPA06007006A (no)
NO (1) NO20062549L (no)
NZ (1) NZ547565A (no)
PL (1) PL1705989T3 (no)
PT (1) PT1705989E (no)
RS (1) RS51111B (no)
SI (1) SI1705989T1 (no)
TN (1) TNSN06187A1 (no)
TW (1) TW200526605A (no)
UA (1) UA83397C2 (no)
UY (1) UY28670A1 (no)
WO (1) WO2005060749A1 (no)
ZA (1) ZA200604715B (no)

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US7514464B2 (en) * 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
US20080176865A1 (en) * 2005-06-15 2008-07-24 Pfizer Limited Substituted arylpyrazoles
US20080146643A1 (en) * 2005-06-15 2008-06-19 Pfizer Limited Combination
US20070149464A1 (en) * 2005-06-15 2007-06-28 Pfizer Inc. Combination
ATE456557T1 (de) * 2005-06-15 2010-02-15 Pfizer Ltd Substituierte arylpyrazole zur verwendung gegen parasiten
US7645786B2 (en) * 2005-06-15 2010-01-12 Pfizer Inc. Substituted arylpyrazoles
CA2630849C (en) * 2005-12-14 2013-05-14 Makhteshim Chemical Works Ltd. Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
FR2928919B1 (fr) * 2008-03-19 2011-07-29 Rhodia Operations Procede de preparation de l'acide difluoroacetique et de ses sels
US20110190365A1 (en) 2008-08-14 2011-08-04 Bayer Crop Science Ag Insecticidal 4-phenyl-1H-pyrazoles
EP2184273A1 (de) 2008-11-05 2010-05-12 Bayer CropScience AG Halogen-substituierte Verbindungen als Pestizide
CN102356070B (zh) * 2009-03-16 2014-07-16 巴斯夫欧洲公司 制备吡唑衍生物的方法
EP2253617A1 (de) 2009-05-20 2010-11-24 Bayer CropScience AG Halogen-substituierte Verbindungen als Pestizide
US20110129574A1 (en) * 2009-11-30 2011-06-02 Pathak Chandrashekhar P Methods and compositions for filling fleshy fruits and vegetables
EP2556060A1 (en) 2010-04-08 2013-02-13 Ah Usa 42 Llc Substituted 3,5- diphenyl-isoxazoline derivatives as insecticides and acaricides
JP2012046486A (ja) * 2010-07-30 2012-03-08 Sumitomo Chemical Co Ltd 動物外部寄生虫防除剤
KR101508862B1 (ko) 2010-08-05 2015-04-07 조에티스 엘엘씨 구충제로서 이속사졸린 유도체
WO2012038851A1 (en) 2010-09-24 2012-03-29 Pfizer Inc. Isoxazoline oximes as antiparasitic agents
FR2972452B1 (fr) 2011-03-09 2013-03-15 Rhodia Operations Procede de preparation du difluoroacetonitrile et de ses derives
HUE029810T2 (en) 2011-03-10 2017-03-28 Zoetis Services Llc Spirocyclic isoxazole derivatives as antiparasitic agents
CN103562190A (zh) 2011-03-22 2014-02-05 佐蒂斯有限责任公司 作为抗寄生虫药的异噁唑啉衍生物
US9133172B2 (en) 2012-02-03 2015-09-15 Zoetis Services Llc Dihydrofuran azetidine derivatives as antiparasitic agents
US9073912B2 (en) 2012-05-09 2015-07-07 Zoetis Services Llc Azetidine derivatives as antiparasitic agents
US20150297565A1 (en) 2012-12-12 2015-10-22 Zoetis Services Llc Phenylpyrazole injectable compositions

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Also Published As

Publication number Publication date
MXPA06007006A (es) 2006-08-31
BRPI0417810A (pt) 2007-04-10
CN1893825A (zh) 2007-01-10
IS8492A (is) 2006-05-31
PL1705989T3 (pl) 2009-04-30
UA83397C2 (uk) 2008-07-10
KR100815637B1 (ko) 2008-03-20
CA2549479A1 (en) 2005-07-07
JP4805164B2 (ja) 2011-11-02
NZ547565A (en) 2009-07-31
UY28670A1 (es) 2005-07-29
BRPI0417810B8 (pt) 2021-05-25
ZA200604715B (en) 2007-03-28
JP2008174563A (ja) 2008-07-31
EP1705989B8 (en) 2009-03-25
HK1096824A1 (en) 2007-06-15
US20050148649A1 (en) 2005-07-07
ES2315724T3 (es) 2009-04-01
CN100377645C (zh) 2008-04-02
DE602004017782D1 (de) 2008-12-24
KR20060101777A (ko) 2006-09-26
AU2004304717B2 (en) 2010-11-18
JP2007514735A (ja) 2007-06-07
WO2005060749A1 (en) 2005-07-07
IL175992A0 (en) 2006-10-05
CA2549479C (en) 2009-08-18
US7435753B2 (en) 2008-10-14
AU2004304717A1 (en) 2005-07-07
EA010740B1 (ru) 2008-10-30
AR046942A1 (es) 2006-01-04
ATE413809T1 (de) 2008-11-15
EP1705989B1 (en) 2008-11-12
TW200526605A (en) 2005-08-16
TNSN06187A1 (fr) 2007-11-15
MA28269A1 (fr) 2006-11-01
CY1108649T1 (el) 2014-04-09
EP1705989A1 (en) 2006-10-04
DK1705989T3 (da) 2009-01-19
RS51111B (sr) 2010-10-31
SI1705989T1 (sl) 2009-02-28
GB0329314D0 (en) 2004-01-21
BRPI0417810B1 (pt) 2018-11-21
PT1705989E (pt) 2009-01-20
EA200600979A1 (ru) 2006-10-27

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CHAD Change of the owner's name or address (par. 44 patent law, par. patentforskriften)

Owner name: ZOETIS LLC, US

FC2A Withdrawal, rejection or dismissal of laid open patent application