NO20050801L - Prodrug av protonpumpe inhibitorer - Google Patents

Prodrug av protonpumpe inhibitorer

Info

Publication number
NO20050801L
NO20050801L NO20050801A NO20050801A NO20050801L NO 20050801 L NO20050801 L NO 20050801L NO 20050801 A NO20050801 A NO 20050801A NO 20050801 A NO20050801 A NO 20050801A NO 20050801 L NO20050801 L NO 20050801L
Authority
NO
Norway
Prior art keywords
proton pump
pump inhibitors
prodrug
prodrugs
bioavailability
Prior art date
Application number
NO20050801A
Other languages
English (en)
Norwegian (no)
Inventor
George Sachs
Jai Moo Shin
Michael E Garst
Original Assignee
Univ California
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ California filed Critical Univ California
Publication of NO20050801L publication Critical patent/NO20050801L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/04—Drugs for disorders of the respiratory system for throat disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
NO20050801A 2002-07-19 2005-02-15 Prodrug av protonpumpe inhibitorer NO20050801L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39745902P 2002-07-19 2002-07-19
PCT/US2003/022419 WO2004009583A2 (fr) 2002-07-19 2003-07-15 Promedicaments des inhibiteurs de la pompe a protons

Publications (1)

Publication Number Publication Date
NO20050801L true NO20050801L (no) 2005-02-15

Family

ID=30771064

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20050801A NO20050801L (no) 2002-07-19 2005-02-15 Prodrug av protonpumpe inhibitorer

Country Status (23)

Country Link
US (3) US6897227B2 (fr)
EP (1) EP1556371B1 (fr)
JP (1) JP4463103B2 (fr)
KR (2) KR100788778B1 (fr)
AT (1) ATE323695T1 (fr)
AU (1) AU2003259154B2 (fr)
BR (1) BR0312802A (fr)
CA (1) CA2492718C (fr)
CO (1) CO5690576A2 (fr)
DE (1) DE60304726T2 (fr)
DK (1) DK1556371T3 (fr)
ES (1) ES2263028T3 (fr)
HK (1) HK1079207A1 (fr)
IL (1) IL166371A0 (fr)
MX (1) MXPA05000657A (fr)
NO (1) NO20050801L (fr)
NZ (1) NZ538221A (fr)
PL (1) PL375255A1 (fr)
PT (1) PT1556371E (fr)
RU (1) RU2292342C2 (fr)
TW (1) TW200502231A (fr)
WO (1) WO2004009583A2 (fr)
ZA (1) ZA200501116B (fr)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6852739B1 (en) * 1999-02-26 2005-02-08 Nitromed Inc. Methods using proton pump inhibitors and nitric oxide donors
CA2493618A1 (fr) * 2002-08-01 2004-02-12 Nitromed, Inc. Inhibiteurs nitroses de la pompe a protons, compositions et procedes d'utilisation
BRPI0412590A (pt) * 2003-07-15 2006-09-19 Allergan Inc processo para preparação de pró-drogas isomericamente puras de inibidores de bomba de próton
US20050075371A1 (en) * 2003-10-03 2005-04-07 Allergan, Inc. Methods and compositions for the oral administration of prodrugs of proton pump inhibitors
US20060241037A1 (en) * 2003-10-03 2006-10-26 Allergan Inc. Compositions comprising trefoil factor family peptides and/or mucoadhesives and proton pump ihhibitor prodrugs
EP1715861A2 (fr) * 2004-02-18 2006-11-02 Allergan, Inc. Methodes et compositions d'administration de promedicaments d'inhibiteurs de la pompe a protons
US20070161679A1 (en) * 2004-02-18 2007-07-12 Allergan, Inc. Method and compositions for the intravenous administration of compounds related to proton pump inhibitors
BRPI0507796A (pt) * 2004-03-11 2007-07-17 Allergan Inc métodos e composições para o tratamento de condições relacionadas com a secreção de ácido gástrico
DK1740571T3 (da) 2004-04-28 2009-11-02 Hetero Drugs Ltd Fremgangsmåde til fremstilling af pyridinylmethyl-1H-benzimidazolforbindelser i enantiomerisk beriget form eller som enkelte enantiomerer
WO2007073301A1 (fr) * 2005-12-23 2007-06-28 Astrazeneca Ab Derives du benzoimidazole en tant que promedicaments d'inhibiteurs de la pompe a protons
WO2007081871A1 (fr) * 2006-01-10 2007-07-19 Allergan, Inc. Procedes et compositions de sels therapeutiques
NZ572007A (en) * 2006-05-09 2010-12-24 Astrazeneca Ab Parenteral formulation comprising proton pump inhibitor sterilized in its final container by ionizing radiation
US20070293543A1 (en) * 2006-06-19 2007-12-20 Edward Lee THRESHOLD BLOOD OMEPRAZOLE CONCENTRATION IS 50 NG/ML FOR THE MAINTENANCE OF INTRAGASTRIC pH OF AT LEAST 4.0 AFTER ORAL DOSING WITH CMA-OMEPRAZOLE, AGN 201904-Z
US20100317689A1 (en) * 2006-09-19 2010-12-16 Garst Michael E Prodrugs of proton pump inhibitors including the 1h-imidazo[4,5-b] pyridine moiety
US20100113524A1 (en) * 2006-09-19 2010-05-06 Garst Michael E Prodrugs of proton pump inhibitors including the (1h-pyrrol-1-yl)-1h-benzimidazole moiety
WO2009044976A1 (fr) * 2007-10-05 2009-04-09 Lg Electronics Inc. Dispositif d'affichage à plasma
KR20090035195A (ko) * 2007-10-05 2009-04-09 엘지전자 주식회사 플라즈마 디스플레이 장치
KR100895333B1 (ko) * 2007-11-01 2009-05-07 엘지전자 주식회사 플라즈마 디스플레이 패널의 구동 방법 및 그를 이용한플라즈마 디스플레이 장치
EP2627178B1 (fr) 2010-10-11 2018-05-02 Merck Sharp & Dohme Corp. Composés de type quinazolinone convenant comme antagonistes de crth2
AU2011349524B2 (en) 2010-12-23 2016-06-02 Merck Sharp & Dohme Corp. Quinoxalines and aza-quinoxalines as CRTH2 receptor modulators
EP2661265B1 (fr) 2010-12-23 2017-03-08 Merck Sharp & Dohme Corp. Quinoléines et aza-quinoléines en tant que modulateurs de l'activité du récepteur crth2
CN107405338A (zh) * 2015-01-09 2017-11-28 加州大学评议会 用于治疗胃肠道感染的组合物和方法
CN108997177A (zh) * 2018-09-04 2018-12-14 邵阳学院 一种微波促进n-苯磺酰基硝基苯胺类化合物合成的方法

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US430042A (en) * 1890-06-10 Valve
SE416649B (sv) * 1974-05-16 1981-01-26 Haessle Ab Forfarande for framstellning av foreningar som paverkar magsyrasekretionen
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
JPS6150978A (ja) * 1984-08-16 1986-03-13 Takeda Chem Ind Ltd ピリジン誘導体およびその製造法
IL76839A (en) * 1984-10-31 1988-08-31 Byk Gulden Lomberg Chem Fab Picoline derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
SE8505112D0 (sv) * 1985-10-29 1985-10-29 Haessle Ab Novel pharmacological compounds
US4758597A (en) * 1987-05-15 1988-07-19 University Patents, Inc. Carenadiol and derivatives
US4965269A (en) * 1989-12-20 1990-10-23 Ab Hassle Therapeutically active chloro substituted benzimidazoles
US5045522A (en) * 1990-03-27 1991-09-03 Phillips Petroleum Company Absorption composition comprising zinc titanate for removal of hydrogen sulfide from fluid streams
ES2140391T3 (es) * 1990-06-20 2000-03-01 Astra Ab Derivados de dialcoxi-piridinil-bencimidazol, procedimiento para su preparacion y su uso farmaceutico.
SE9301830D0 (sv) * 1993-05-28 1993-05-28 Ab Astra New compounds
PL181801B1 (pl) * 1994-06-10 2001-09-28 Byk Gulden Lomberg Chem Fab Podstawione aryloalkilotioalkilotiopirydyny do zwalczania bakterii Helicobacter oraz srodek leczniczy zawierajacy podstawione aryloalkilotioalkilotiopirydyny PL
US5708017A (en) * 1995-04-04 1998-01-13 Merck & Co., Inc. Stable, ready-to-use pharmaceutical paste composition containing proton pump inhibitors
US6093734A (en) * 1998-08-10 2000-07-25 Partnership Of Michael E. Garst, George Sachs, And Jai Moo Shin Prodrugs of proton pump inhibitors
ES2192394T3 (es) * 1998-08-10 2003-10-01 Winston Pharmateuticals Llc Profarmacos de inhibidores de la bomba de protones.
ES2232169T3 (es) * 1998-08-12 2005-05-16 Gilead Sciences, Inc. Procedimiento de fabricacion de nucleosidos de 1,3-oxatiolano.
SE0002476D0 (sv) 2000-06-30 2000-06-30 Astrazeneca Ab New compounds
US6599167B2 (en) * 2000-09-27 2003-07-29 Glenn Waltz Game call holder and amplifying device
WO2002030920A1 (fr) * 2000-10-12 2002-04-18 Takeda Chemical Industries, Ltd. Composes derives de benzimidazole, leur procede de production et leur utilisation

Also Published As

Publication number Publication date
CA2492718A1 (fr) 2004-01-29
KR20050047078A (ko) 2005-05-19
AU2003259154B2 (en) 2006-12-07
JP4463103B2 (ja) 2010-05-12
RU2005105564A (ru) 2005-10-10
TW200502231A (en) 2005-01-16
DE60304726T2 (de) 2007-08-09
HK1079207A1 (en) 2006-03-31
AU2003259154C1 (en) 2004-02-09
PL375255A1 (en) 2005-11-28
DK1556371T3 (da) 2006-08-21
CA2492718C (fr) 2010-12-21
RU2292342C2 (ru) 2007-01-27
US20050143423A1 (en) 2005-06-30
KR100822981B1 (ko) 2008-04-16
AU2003259154A1 (en) 2004-02-09
US20040102484A1 (en) 2004-05-27
ES2263028T3 (es) 2006-12-01
BR0312802A (pt) 2005-04-19
ZA200501116B (en) 2006-11-29
KR20070005029A (ko) 2007-01-09
IL166371A0 (en) 2006-01-16
US6897227B2 (en) 2005-05-24
JP2005536519A (ja) 2005-12-02
EP1556371B1 (fr) 2006-04-19
US20050182101A1 (en) 2005-08-18
KR100788778B1 (ko) 2007-12-27
PT1556371E (pt) 2006-09-29
WO2004009583A3 (fr) 2004-03-18
EP1556371A2 (fr) 2005-07-27
WO2004009583A2 (fr) 2004-01-29
DE60304726D1 (de) 2006-05-24
NZ538221A (en) 2006-11-30
MXPA05000657A (es) 2005-08-19
ATE323695T1 (de) 2006-05-15
CO5690576A2 (es) 2006-10-31

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application