NO20032253L - Piperazinylpyrazinforbindelser som antagonister av serotonin 5-HT2-reseptorer - Google Patents
Piperazinylpyrazinforbindelser som antagonister av serotonin 5-HT2-reseptorerInfo
- Publication number
- NO20032253L NO20032253L NO20032253A NO20032253A NO20032253L NO 20032253 L NO20032253 L NO 20032253L NO 20032253 A NO20032253 A NO 20032253A NO 20032253 A NO20032253 A NO 20032253A NO 20032253 L NO20032253 L NO 20032253L
- Authority
- NO
- Norway
- Prior art keywords
- serotonin
- antagonists
- receptors
- compounds
- piperazinylpyrazine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/20—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0004244A SE0004244D0 (sv) | 2000-11-20 | 2000-11-20 | Novel compounds and their use |
US25370200P | 2000-11-28 | 2000-11-28 | |
PCT/SE2001/002570 WO2002040457A1 (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20032253D0 NO20032253D0 (no) | 2003-05-19 |
NO20032253L true NO20032253L (no) | 2003-07-18 |
NO325321B1 NO325321B1 (no) | 2008-03-31 |
Family
ID=26655310
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20032253A NO325321B1 (no) | 2000-11-20 | 2003-05-19 | Piperazinylpyrazinforbindelser, preparat, fremgangsmate for fremstilling samt anvendelse av slike |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP1337518B1 (no) |
JP (1) | JP4204315B2 (no) |
KR (1) | KR100831909B1 (no) |
CN (1) | CN1227237C (no) |
AT (1) | ATE433962T1 (no) |
AU (1) | AU1529402A (no) |
BR (1) | BR0115436A (no) |
CA (2) | CA2428905A1 (no) |
DE (1) | DE60139021D1 (no) |
DK (1) | DK1337518T3 (no) |
EA (1) | EA005975B1 (no) |
ES (1) | ES2328671T3 (no) |
HK (1) | HK1066810A1 (no) |
IL (2) | IL155875A0 (no) |
MX (1) | MXPA03004391A (no) |
NO (1) | NO325321B1 (no) |
NZ (1) | NZ525699A (no) |
PL (1) | PL360982A1 (no) |
WO (1) | WO2002040457A1 (no) |
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US7105526B2 (en) | 2002-06-28 | 2006-09-12 | Banyu Pharmaceuticals Co., Ltd. | Benzimidazole derivatives |
US7772188B2 (en) | 2003-01-28 | 2010-08-10 | Ironwood Pharmaceuticals, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
CL2004000826A1 (es) * | 2003-04-25 | 2005-03-04 | Pfizer | Uso de un agonista para el receptor 5-ht2c para preparar un medicamento util en el tratamiento de la incontinencia urinaria provocada por estres, con la condicion de que el agonista no sea 1-[6-cloro-5-(trifluorometil)-2-piridinil]piperazina (org-129 |
CN1902177A (zh) | 2003-09-22 | 2007-01-24 | 万有制药株式会社 | 新哌啶衍生物 |
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WO2006020959A2 (en) | 2004-08-13 | 2006-02-23 | Amgen Inc. | Substituted benzofused heterocycles |
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CN101094689B (zh) | 2004-11-01 | 2013-06-12 | 安米林药品有限责任公司 | 治疗肥胖以及肥胖相关疾病和病症的方法 |
US7737155B2 (en) | 2005-05-17 | 2010-06-15 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
US8138206B2 (en) | 2005-05-30 | 2012-03-20 | Msd. K.K. | Piperidine derivative |
EP1916239A4 (en) | 2005-08-10 | 2009-10-21 | Banyu Pharma Co Ltd | PYRIDONE COMPOUND |
EP1922336B1 (en) | 2005-08-11 | 2012-11-21 | Amylin Pharmaceuticals, LLC | Hybrid polypeptides with selectable properties |
BRPI0614649A2 (pt) | 2005-08-11 | 2011-04-12 | Amylin Pharmaceuticals Inc | polipeptìdeos hìbridos com propriedades selecionáveis |
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ES2381205T3 (es) | 2005-11-10 | 2012-05-24 | Msd K.K. | Derivado espiro aza-sustituido |
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WO2016030534A1 (en) | 2014-08-29 | 2016-03-03 | Tes Pharma S.R.L. | INHIBITORS OF α-AMINO-β-CARBOXYMUCONIC ACID SEMIALDEHYDE DECARBOXYLASE |
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2001
- 2001-11-20 ES ES01983901T patent/ES2328671T3/es not_active Expired - Lifetime
- 2001-11-20 IL IL15587501A patent/IL155875A0/xx active IP Right Grant
- 2001-11-20 BR BR0115436-2A patent/BR0115436A/pt not_active IP Right Cessation
- 2001-11-20 EP EP01983901A patent/EP1337518B1/en not_active Expired - Lifetime
- 2001-11-20 AT AT01983901T patent/ATE433962T1/de not_active IP Right Cessation
- 2001-11-20 WO PCT/SE2001/002570 patent/WO2002040457A1/en active IP Right Grant
- 2001-11-20 CA CA002428905A patent/CA2428905A1/en active Pending
- 2001-11-20 CA CA2449899A patent/CA2449899C/en not_active Expired - Fee Related
- 2001-11-20 PL PL36098201A patent/PL360982A1/xx unknown
- 2001-11-20 EA EA200300595A patent/EA005975B1/ru not_active IP Right Cessation
- 2001-11-20 CN CNB018192416A patent/CN1227237C/zh not_active Expired - Fee Related
- 2001-11-20 KR KR1020037006822A patent/KR100831909B1/ko not_active IP Right Cessation
- 2001-11-20 JP JP2002542785A patent/JP4204315B2/ja not_active Expired - Fee Related
- 2001-11-20 DK DK01983901T patent/DK1337518T3/da active
- 2001-11-20 AU AU1529402A patent/AU1529402A/xx not_active Withdrawn
- 2001-11-20 DE DE60139021T patent/DE60139021D1/de not_active Expired - Lifetime
- 2001-11-20 MX MXPA03004391A patent/MXPA03004391A/es active IP Right Grant
- 2001-11-20 NZ NZ525699A patent/NZ525699A/en unknown
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2003
- 2003-05-12 IL IL155875A patent/IL155875A/en not_active IP Right Cessation
- 2003-05-19 NO NO20032253A patent/NO325321B1/no not_active IP Right Cessation
-
2004
- 2004-12-14 HK HK04109907A patent/HK1066810A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
AU1529402A (en) | 2002-05-27 |
EP1337518A1 (en) | 2003-08-27 |
NO20032253D0 (no) | 2003-05-19 |
ATE433962T1 (de) | 2009-07-15 |
BR0115436A (pt) | 2004-01-06 |
NZ525699A (en) | 2005-03-24 |
NO325321B1 (no) | 2008-03-31 |
WO2002040457A1 (en) | 2002-05-23 |
MXPA03004391A (es) | 2004-05-31 |
DE60139021D1 (de) | 2009-07-30 |
DK1337518T3 (da) | 2009-10-19 |
CA2428905A1 (en) | 2002-05-23 |
HK1066810A1 (en) | 2005-04-01 |
IL155875A (en) | 2007-06-17 |
KR20030060946A (ko) | 2003-07-16 |
CN1227237C (zh) | 2005-11-16 |
ES2328671T3 (es) | 2009-11-17 |
EA005975B1 (ru) | 2005-08-25 |
JP2004531465A (ja) | 2004-10-14 |
CA2449899A1 (en) | 2002-05-23 |
KR100831909B1 (ko) | 2008-05-26 |
CN1520404A (zh) | 2004-08-11 |
CA2449899C (en) | 2010-04-06 |
EP1337518B1 (en) | 2009-06-17 |
JP4204315B2 (ja) | 2009-01-07 |
IL155875A0 (en) | 2003-12-23 |
EA200300595A1 (ru) | 2003-10-30 |
PL360982A1 (en) | 2004-09-20 |
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