NO20021803L - Isoksazolkarboksamid-derivater - Google Patents
Isoksazolkarboksamid-derivaterInfo
- Publication number
- NO20021803L NO20021803L NO20021803A NO20021803A NO20021803L NO 20021803 L NO20021803 L NO 20021803L NO 20021803 A NO20021803 A NO 20021803A NO 20021803 A NO20021803 A NO 20021803A NO 20021803 L NO20021803 L NO 20021803L
- Authority
- NO
- Norway
- Prior art keywords
- isoksazolkarboksamid
- derivatives
- isoksazolkarboksamid derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Urology & Nephrology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1999MI002173A IT1314191B1 (it) | 1999-10-18 | 1999-10-18 | Derivati isossazolcarbossamidici |
PCT/EP2000/010144 WO2001029015A2 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20021803D0 NO20021803D0 (no) | 2002-04-17 |
NO20021803L true NO20021803L (no) | 2002-06-17 |
Family
ID=11383797
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20021803A NO20021803L (no) | 1999-10-18 | 2002-04-17 | Isoksazolkarboksamid-derivater |
Country Status (25)
Country | Link |
---|---|
EP (1) | EP1226131B1 (es) |
JP (1) | JP2003512362A (es) |
KR (1) | KR20020038944A (es) |
CN (1) | CN1139579C (es) |
AR (1) | AR029400A1 (es) |
AT (1) | ATE256670T1 (es) |
AU (1) | AU757614B2 (es) |
BR (1) | BR0014851A (es) |
CA (1) | CA2385472A1 (es) |
DE (1) | DE60007347T2 (es) |
DK (1) | DK1226131T3 (es) |
ES (1) | ES2210033T3 (es) |
HK (1) | HK1044940A1 (es) |
HU (1) | HUP0203184A3 (es) |
IL (1) | IL148837A0 (es) |
IT (1) | IT1314191B1 (es) |
MX (1) | MXPA02003432A (es) |
MY (1) | MY120400A (es) |
NO (1) | NO20021803L (es) |
NZ (1) | NZ517884A (es) |
PL (1) | PL356990A1 (es) |
PT (1) | PT1226131E (es) |
RU (1) | RU2002113096A (es) |
WO (1) | WO2001029015A2 (es) |
ZA (1) | ZA200203942B (es) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2006301376A1 (en) | 2005-10-11 | 2007-04-19 | F. Hoffmann-La Roche Ag | Isoxazole derivatives |
ATE466858T1 (de) | 2005-11-09 | 2010-05-15 | Hoffmann La Roche | 3-arylisoxazol-4-carbonylbenzofuranderivative |
WO2007071598A1 (en) | 2005-12-23 | 2007-06-28 | F. Hoffmann-La Roche Ag | Aryl-isoxazolo-4-yl-oxadiazole derivatives |
DK1968973T3 (da) | 2005-12-27 | 2011-10-31 | Hoffmann La Roche | Aryl-isoxazol-4-yl-imidazolderivater |
CA2636112A1 (en) | 2006-01-17 | 2007-07-26 | F.Hoffmann-La Roche Ag | Aryl-isoxazol-4-yl-imidazo[1,2-a]pyridine derivatives useful for the treatment of alzheimer's disease via gaba receptors |
KR101119365B1 (ko) | 2006-05-31 | 2012-03-07 | 에프. 호프만-라 로슈 아게 | 아릴-4-에틴일-아이속사졸 유도체 |
CA2690975A1 (en) | 2007-06-22 | 2008-12-31 | F. Hoffmann-La Roche Ag | Isoxazole-imidazole derivatives |
US7943619B2 (en) | 2007-12-04 | 2011-05-17 | Hoffmann-La Roche Inc. | Isoxazolo-pyridazine derivatives |
US7902201B2 (en) | 2007-12-04 | 2011-03-08 | Hoffmann-La Roche Inc. | Isoxazolo-pyrazine derivatives |
JP5301556B2 (ja) | 2007-12-04 | 2013-09-25 | エフ.ホフマン−ラ ロシュ アーゲー | イソオキサゾロ−ピラジン誘導体 |
WO2010081851A1 (en) | 2009-01-14 | 2010-07-22 | Genoscience Pharma | Piperidin-4-ylpiperazine compounds for the treatment of hcv infection |
TW201033201A (en) | 2009-02-19 | 2010-09-16 | Hoffmann La Roche | Isoxazole-isoxazole and isoxazole-isothiazole derivatives |
US8389550B2 (en) | 2009-02-25 | 2013-03-05 | Hoffmann-La Roche Inc. | Isoxazoles / O-pyridines with ethyl and ethenyl linker |
US8222246B2 (en) | 2009-04-02 | 2012-07-17 | Hoffmann-La Roche Inc. | Substituted isoxazoles |
US8227461B2 (en) | 2009-04-30 | 2012-07-24 | Hoffmann-La Roche Inc. | Isoxazoles |
BRPI1013844A2 (pt) | 2009-05-05 | 2016-04-12 | Hoffmann La Roche | derivados de piridina-isoxazol |
CA2759598C (en) | 2009-05-05 | 2017-09-12 | F. Hoffmann-La Roche Ag | Isoxazole-thiazole derivatives as gaba a receptor inverse agonists for use in the treatment of cognitive disorders |
CA2760746C (en) | 2009-05-05 | 2017-07-11 | F. Hoffmann-La Roche Ag | Isoxazole-pyrazole derivatives |
CA2760597C (en) | 2009-05-05 | 2017-08-22 | F. Hoffmann-La Roche Ag | Isoxazole-pyridazine derivatives |
JP5481555B2 (ja) | 2009-05-07 | 2014-04-23 | エフ.ホフマン−ラ ロシュ アーゲー | Gaba修飾薬としてのイソオキサゾール−ピリジン誘導体 |
US8785435B2 (en) | 2011-10-20 | 2014-07-22 | Hoffmann-La Roche Inc. | Solid forms |
CN113121540B (zh) * | 2020-01-15 | 2024-01-26 | 鲁南制药集团股份有限公司 | 一种西格列汀游离碱的合成方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1254469B (it) * | 1992-02-25 | 1995-09-25 | Recordati Chem Pharm | Derivati benzopiranici e benzotiopiranici |
IT1266582B1 (it) * | 1993-07-30 | 1997-01-09 | Recordati Chem Pharm | Derivati (di)azacicloesanici e diazacicloeptanici |
DE4425146A1 (de) * | 1994-07-15 | 1996-01-18 | Basf Ag | Verwendung heterocyclischer Verbindungen |
-
1999
- 1999-10-18 IT IT1999MI002173A patent/IT1314191B1/it active
-
2000
- 2000-10-10 MY MYPI20004718A patent/MY120400A/en unknown
- 2000-10-16 CN CNB008143226A patent/CN1139579C/zh not_active Expired - Fee Related
- 2000-10-16 EP EP00992436A patent/EP1226131B1/en not_active Expired - Lifetime
- 2000-10-16 CA CA002385472A patent/CA2385472A1/en not_active Abandoned
- 2000-10-16 AU AU28347/01A patent/AU757614B2/en not_active Ceased
- 2000-10-16 DK DK00992436T patent/DK1226131T3/da active
- 2000-10-16 HU HU0203184A patent/HUP0203184A3/hu unknown
- 2000-10-16 NZ NZ517884A patent/NZ517884A/en unknown
- 2000-10-16 IL IL14883700A patent/IL148837A0/xx unknown
- 2000-10-16 MX MXPA02003432A patent/MXPA02003432A/es not_active Application Discontinuation
- 2000-10-16 BR BR0014851-2A patent/BR0014851A/pt not_active IP Right Cessation
- 2000-10-16 KR KR1020027004663A patent/KR20020038944A/ko not_active Application Discontinuation
- 2000-10-16 DE DE60007347T patent/DE60007347T2/de not_active Expired - Fee Related
- 2000-10-16 PT PT00992436T patent/PT1226131E/pt unknown
- 2000-10-16 PL PL00356990A patent/PL356990A1/xx not_active Application Discontinuation
- 2000-10-16 ES ES00992436T patent/ES2210033T3/es not_active Expired - Lifetime
- 2000-10-16 JP JP2001531815A patent/JP2003512362A/ja active Pending
- 2000-10-16 WO PCT/EP2000/010144 patent/WO2001029015A2/en active IP Right Grant
- 2000-10-16 RU RU2002113096/04A patent/RU2002113096A/ru not_active Application Discontinuation
- 2000-10-16 AT AT00992436T patent/ATE256670T1/de not_active IP Right Cessation
- 2000-10-18 AR ARP000105475A patent/AR029400A1/es not_active Application Discontinuation
-
2002
- 2002-04-17 NO NO20021803A patent/NO20021803L/no not_active Application Discontinuation
- 2002-05-17 ZA ZA200203942A patent/ZA200203942B/en unknown
- 2002-08-13 HK HK02105918.6A patent/HK1044940A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
MY120400A (en) | 2005-10-31 |
CN1379767A (zh) | 2002-11-13 |
NZ517884A (en) | 2003-08-29 |
RU2002113096A (ru) | 2003-11-10 |
HUP0203184A3 (en) | 2004-12-28 |
CN1139579C (zh) | 2004-02-25 |
DE60007347T2 (de) | 2004-09-02 |
ATE256670T1 (de) | 2004-01-15 |
IL148837A0 (en) | 2002-09-12 |
AR029400A1 (es) | 2003-06-25 |
EP1226131B1 (en) | 2003-12-17 |
JP2003512362A (ja) | 2003-04-02 |
IT1314191B1 (it) | 2002-12-06 |
HK1044940A1 (zh) | 2002-11-08 |
DK1226131T3 (da) | 2004-04-19 |
HUP0203184A2 (hu) | 2003-01-28 |
ITMI992173A1 (it) | 2001-04-18 |
ES2210033T3 (es) | 2004-07-01 |
AU2834701A (en) | 2001-04-30 |
MXPA02003432A (es) | 2002-08-20 |
PT1226131E (pt) | 2004-05-31 |
ZA200203942B (en) | 2003-01-02 |
WO2001029015A3 (en) | 2001-11-01 |
AU757614B2 (en) | 2003-02-27 |
CA2385472A1 (en) | 2001-04-26 |
KR20020038944A (ko) | 2002-05-24 |
ITMI992173A0 (it) | 1999-10-18 |
BR0014851A (pt) | 2002-06-11 |
DE60007347D1 (de) | 2004-01-29 |
EP1226131A2 (en) | 2002-07-31 |
WO2001029015A2 (en) | 2001-04-26 |
NO20021803D0 (no) | 2002-04-17 |
PL356990A1 (en) | 2004-07-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |