NO20011417L - [1,2,4]triazolo[1,5-c]pyrimidin-derivater - Google Patents

[1,2,4]triazolo[1,5-c]pyrimidin-derivater

Info

Publication number
NO20011417L
NO20011417L NO20011417A NO20011417A NO20011417L NO 20011417 L NO20011417 L NO 20011417L NO 20011417 A NO20011417 A NO 20011417A NO 20011417 A NO20011417 A NO 20011417A NO 20011417 L NO20011417 L NO 20011417L
Authority
NO
Norway
Prior art keywords
represent
triazolo
aryl
pyrimidine derivatives
lower alkyl
Prior art date
Application number
NO20011417A
Other languages
English (en)
Other versions
NO20011417D0 (no
Inventor
Junichi Shimada
Hironori Imma
Naoto Osakada
Shizuo Shiozaki
Tomoyuki Kanda
Yoshihisa Kuwana
Original Assignee
Kyowa Hakko Kogyo Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyowa Hakko Kogyo Kk filed Critical Kyowa Hakko Kogyo Kk
Publication of NO20011417D0 publication Critical patent/NO20011417D0/no
Publication of NO20011417L publication Critical patent/NO20011417L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20011417A 1998-09-22 2001-03-20 [1,2,4]triazolo[1,5-c]pyrimidin-derivater NO20011417L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP26717898 1998-09-22
PCT/JP1999/005176 WO2000017201A1 (fr) 1998-09-22 1999-09-22 DERIVES DE [1,2,4]TRIAZOLO[1,5-c]PYRIMIDINE

Publications (2)

Publication Number Publication Date
NO20011417D0 NO20011417D0 (no) 2001-03-20
NO20011417L true NO20011417L (no) 2001-05-21

Family

ID=17441200

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20011417A NO20011417L (no) 1998-09-22 2001-03-20 [1,2,4]triazolo[1,5-c]pyrimidin-derivater

Country Status (15)

Country Link
US (1) US6545000B1 (no)
EP (1) EP1116722B1 (no)
KR (1) KR20010087361A (no)
CN (1) CN1328560A (no)
AT (1) ATE286900T1 (no)
AU (1) AU756144B2 (no)
BR (1) BR9914040A (no)
CA (1) CA2344828A1 (no)
DE (1) DE69923197T2 (no)
EA (1) EA200100265A1 (no)
HU (1) HUP0103921A3 (no)
IL (1) IL142128A0 (no)
NO (1) NO20011417L (no)
NZ (1) NZ510629A (no)
WO (1) WO2000017201A1 (no)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002079204A1 (fr) * 2001-03-28 2002-10-10 Kyowa Hakko Kogyo Co., Ltd. Derive 8-thiazolyl[1,2,4]triazolo[1,5-c]pyrimidine
JP5280597B2 (ja) 2001-03-30 2013-09-04 サンスター技研株式会社 一液加熱硬化型エポキシ樹脂組成物および半導体実装用アンダーフィル材
JP2005516891A (ja) * 2001-09-13 2005-06-09 シェーリング　コーポレイション アデノシンＡ２ａレセプタアンタゴニストと抗鬱薬または抗不安薬との組合せ
AU2002352933A1 (en) * 2001-11-30 2003-06-17 Schering Corporation [1,2,4]-triazole bicylic adenosine A2a receptor antagonists
TW200300686A (en) 2001-11-30 2003-06-16 Schering Corp Adenosine A2a receptor antagonists
US6734179B2 (en) * 2001-12-12 2004-05-11 Hoffmann-La Roche Inc. Benzothiazoles
PL370980A1 (en) * 2001-12-12 2005-06-13 F.Hoffmann-La Roche Ag Benzothiophenes as adenosine receptor modulators
MXPA04007299A (es) 2002-01-28 2004-10-29 Kyowa Hakko Kogyo Kk Metodos de tratamiento de pacientes que sufren de trastornos de movimiento.
AU2003211993A1 (en) * 2002-02-15 2003-09-04 Kyowa Hakko Kogyo Co., Ltd. (1,2,4)TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVES
US20060058320A1 (en) * 2002-09-24 2006-03-16 Kyowa Hakko Kogyo Co., Ltd. [1,2,4] Triazolo[1,5-c]pyrimidine derivatives
US20070010522A1 (en) * 2003-04-09 2007-01-11 Chi Vu Triazolo[1,5-c]pyrimidines and pyrazolo[1,5-c]pyrimidines useful as a2a adenosine receptor antagonists
WO2004092170A2 (en) 2003-04-09 2004-10-28 Biogen Idec Ma Inc. Triazolotriazines and pyrazolotriazines useful as a2a adenosine receptor antagon ists
US7674791B2 (en) 2003-04-09 2010-03-09 Biogen Idec Ma Inc. Triazolopyrazines and methods of making and using the same
EP1633756B1 (en) 2003-04-09 2008-12-24 Biogen Idec MA Inc. A2a adenosine receptor antagonists
BRPI0411120A (pt) 2003-06-10 2006-07-18 Kyowa Hakko Kogyo Kk método para tratar de um distúrbio de ansiedade, composição, agente para tratar de um distúrbio de ansiedade, e, usos de um composto e de um derivado de xantina
US7851478B2 (en) * 2005-06-07 2010-12-14 Kyowa Hakko Kirin Co., Ltd. Agent for preventing and/or treating movement disorder
EP2089389A2 (en) 2006-11-01 2009-08-19 Bristol-Myers Squibb Company Heterocyclic compounds as modulators of glucocorticoid receptor, ap-1, and/or nf-kappa-b activity
TWI473614B (zh) 2008-05-29 2015-02-21 Kyowa Hakko Kirin Co Ltd Anti-analgesic inhibitors
EP2322223A4 (en) * 2008-07-23 2012-08-22 Kyowa Hakko Kirin Co Ltd THERAPEUTIC AGENT AGAINST MIGRAINE
JP5730281B2 (ja) * 2009-03-27 2015-06-10 武田薬品工業株式会社 ポリ（ａｄｐ−リボース）ポリメラーゼ（ｐａｒｐ）阻害剤
WO2018166493A1 (zh) 2017-03-16 2018-09-20 江苏恒瑞医药股份有限公司 杂芳基并[4，3-c]嘧啶-5-胺类衍生物、其制备方法及其在医药上的应用
US20190292188A1 (en) 2018-02-27 2019-09-26 Incyte Corporation Imidazopyrimidines and triazolopyrimidines as a2a / a2b inhibitors
CA3100731A1 (en) 2018-05-18 2019-11-21 Incyte Corporation Fused pyrimidine derivatives as a2a / a2b inhibitors
CA3105721A1 (en) 2018-07-05 2020-01-09 Incyte Corporation Fused pyrazine derivatives as a2a / a2b inhibitors
CN110903291B (zh) * 2018-09-14 2021-09-03 江苏恒瑞医药股份有限公司 一种杂芳基并[4,3-c]嘧啶-5-胺类衍生物的盐、盐的晶型及制备方法
TWI829857B (zh) 2019-01-29 2024-01-21 美商英塞特公司 作為a2a / a2b抑制劑之吡唑并吡啶及三唑并吡啶

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4477450A (en) 1983-03-03 1984-10-16 Riker Laboratories, Inc. Triazolo [4,3-c]pyrimidines substituted by nitrogen-containing heterocyclic rings
US4572910A (en) 1983-03-03 1986-02-25 Riker Laboratories, Inc. Triazolo[1,5-c]pyrimidines substituted by nitrogen-containing heterocyclic rings
US4483987A (en) 1983-06-20 1984-11-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines and amides
NZ208996A (en) 1983-07-28 1989-08-29 American Cyanamid Co 5-substituted(1,2,4 triazpyrimidin-2-amine derivatives and pharmaceutical compositions
EP0459702A1 (en) * 1990-05-29 1991-12-04 Zeneca Limited Azole Derivatives
US5356894A (en) 1990-05-29 1994-10-18 Rodney Peter W Morpholinyl substituted [1,2,4]-triazolo[1,5-a]triazine as antagonist
ATE198890T1 (de) * 1993-09-06 2001-02-15 Kyowa Hakko Kogyo Kk Antidepressiva
DE69820866T2 (de) 1997-03-24 2004-12-30 Kyowa Hakko Kogyo Co., Ltd. [1,2,4]TRIAZOLO[1,5-c]PYRIMIDIN-DERIVATE

Also Published As

Publication number Publication date
DE69923197D1 (de) 2005-02-17
EP1116722A4 (en) 2002-05-29
AU5757999A (en) 2000-04-10
BR9914040A (pt) 2002-01-15
US6545000B1 (en) 2003-04-08
EA200100265A1 (ru) 2001-10-22
EP1116722A1 (en) 2001-07-18
AU756144B2 (en) 2003-01-02
WO2000017201A1 (fr) 2000-03-30
KR20010087361A (ko) 2001-09-15
NO20011417D0 (no) 2001-03-20
ATE286900T1 (de) 2005-01-15
EP1116722B1 (en) 2005-01-12
HUP0103921A2 (hu) 2002-04-29
CA2344828A1 (en) 2000-03-30
CN1328560A (zh) 2001-12-26
IL142128A0 (en) 2002-03-10
DE69923197T2 (de) 2005-12-29
HUP0103921A3 (en) 2002-12-28
NZ510629A (en) 2003-04-29

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application