NO20003069D0 - 5-[4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl]tiazolidin- 2,4-dion-maleinsyre-salt-hydrat som farmasøytikum - Google Patents

5-[4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl]tiazolidin- 2,4-dion-maleinsyre-salt-hydrat som farmasøytikum

Info

Publication number
NO20003069D0
NO20003069D0 NO20003069A NO20003069A NO20003069D0 NO 20003069 D0 NO20003069 D0 NO 20003069D0 NO 20003069 A NO20003069 A NO 20003069A NO 20003069 A NO20003069 A NO 20003069A NO 20003069 D0 NO20003069 D0 NO 20003069D0
Authority
NO
Norway
Prior art keywords
thiazolidine
dione
pyridyl
ethoxy
benzyl
Prior art date
Application number
NO20003069A
Other languages
English (en)
Other versions
NO20003069L (no
NO317254B1 (no
Inventor
Paul David James Blackler
Michael John Sasse
David C Lee
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of NO20003069L publication Critical patent/NO20003069L/no
Publication of NO20003069D0 publication Critical patent/NO20003069D0/no
Publication of NO317254B1 publication Critical patent/NO317254B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
NO20003069A 1997-12-16 2000-06-15 5-[4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl]tiazolidin-2,4-dion-maleinsyre-salt-hydrat som farmasoytikum NO317254B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9726566.4A GB9726566D0 (en) 1997-12-16 1997-12-16 Novel pharmaceutical
PCT/EP1998/008155 WO1999031095A1 (en) 1997-12-16 1998-12-14 5-[4-[2- (n-methyl-n- (2-pyridyl)amino) ethoxy]benzyl] thiazolidine-2, 4-dione, maleic acid salt, hydrate as pharmaceutical

Publications (3)

Publication Number Publication Date
NO20003069L NO20003069L (no) 2000-06-15
NO20003069D0 true NO20003069D0 (no) 2000-06-15
NO317254B1 NO317254B1 (no) 2004-09-27

Family

ID=10823692

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20003069A NO317254B1 (no) 1997-12-16 2000-06-15 5-[4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl]tiazolidin-2,4-dion-maleinsyre-salt-hydrat som farmasoytikum

Country Status (35)

Country Link
EP (2) EP1661895A1 (no)
JP (1) JP2002508373A (no)
KR (1) KR100549142B1 (no)
CN (3) CN101381367A (no)
AP (1) AP1365A (no)
AR (1) AR017214A1 (no)
AU (1) AU1967999A (no)
BG (1) BG64988B1 (no)
BR (1) BR9813600A (no)
CA (1) CA2314107A1 (no)
CO (1) CO4980880A1 (no)
CZ (1) CZ299965B6 (no)
DZ (1) DZ2681A1 (no)
EA (1) EA004260B1 (no)
EG (1) EG22337A (no)
GB (1) GB9726566D0 (no)
HR (1) HRP20000408B1 (no)
HU (1) HUP0100509A3 (no)
IL (1) IL136424A (no)
IN (1) IN192487B (no)
MA (1) MA26580A1 (no)
MY (1) MY135612A (no)
NO (1) NO317254B1 (no)
OA (1) OA11766A (no)
PE (1) PE20000058A1 (no)
PL (1) PL341146A1 (no)
RS (1) RS50126B (no)
SA (1) SA99191115B1 (no)
SK (1) SK286618B6 (no)
TR (2) TR200001799T2 (no)
TW (1) TW509690B (no)
UA (1) UA72198C2 (no)
UY (2) UY25304A1 (no)
WO (1) WO1999031095A1 (no)
ZA (1) ZA9811506B (no)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6664278B2 (en) 1997-12-16 2003-12-16 Smithkline Beecham P.L.C. Hydrate of 5-[4-[2-(N-methyl-N-(2-pyridil)amino)ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt
GB9726568D0 (en) 1997-12-16 1998-02-11 Smithkline Beecham Plc Novel pharmaceutical
GB9909041D0 (en) * 1999-04-20 1999-06-16 Smithkline Beecham Plc Novel pharmaceutical
WO2000064892A2 (en) * 1999-04-23 2000-11-02 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
PL351684A1 (en) * 1999-04-23 2003-06-02 Smithkline Beecham Plc Polymorph of 5−[4−[2− (n−methyl−n−( 2−pyridyl)amino) ethoxy]benzyl] thiazolidine−2,4−dione, maleic acid salt
EP1175418A2 (en) * 1999-04-23 2002-01-30 Smithkline Beecham Plc Thiazolidinedione derivative and its use as antidiabetic
EA004244B1 (ru) 2000-04-25 2004-02-26 Киорин Фармасьютикал Ко., Лтд. Новый стабильный кристалл производного тиазолидиндиона и способ его получения
GB0014005D0 (en) * 2000-06-08 2000-08-02 Smithkline Beecham Plc Novel pharmaceutical
GB0021784D0 (en) * 2000-09-05 2000-10-18 Smithkline Beecham Plc Novel pharmaceutical
GB0021978D0 (en) * 2000-09-07 2000-10-25 Smithkline Beecham Plc Novel pharmaceutical
BR0114196A (pt) * 2000-09-26 2003-07-22 Reddy S Res Foundation Formas polimórficas de maleato de 5-[4-[2-[n-metil-n-(2-piridil) amino]etóxi]benzil]tiazolidina-2,4-diona e processo para a preparação das mesmas.
GB0129872D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
AU2002350965A1 (en) * 2001-12-13 2003-06-23 Smithkline Beecham Plc Toluenesulfonate hydrates of a thiazolidinedione derivative
GB0129876D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB2405403A (en) * 2003-08-29 2005-03-02 Cipla Ltd Rosiglitazone maleate of particular polymorphic forms and methods of preparing rosiglitazone free base
ITMI20041537A1 (it) * 2004-07-28 2004-10-28 Chemi Spa Nuova forma polimorfa del rosiglitazone maleato
CZ298424B6 (cs) * 2005-05-24 2007-09-26 Zentiva, A. S. Zpusob krystalizace rosiglitazonu a jeho derivátuze smesných rozpouštedel
EP2184055A1 (en) 2008-11-07 2010-05-12 LEK Pharmaceuticals d.d. Process for preparing solid dosage forms of rosiglitazone maleate

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3856378T2 (de) * 1987-09-04 2000-05-11 Beecham Group Plc Substituierte Thiazolidindionderivate
GB8820389D0 (en) * 1988-08-26 1988-09-28 Beecham Group Plc Novel compounds
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
WO1995021608A1 (en) * 1994-02-10 1995-08-17 Smithkline Beecham Plc Use of insulin sensitisers for treating renal diseases

Also Published As

Publication number Publication date
UA72198C2 (en) 2005-02-15
EA200000654A1 (ru) 2000-12-25
UY25308A1 (es) 1999-07-19
WO1999031095A1 (en) 1999-06-24
UY25304A1 (es) 2000-12-29
KR100549142B1 (ko) 2006-02-03
RS50126B (sr) 2009-03-25
BR9813600A (pt) 2000-10-10
IN192487B (no) 2004-04-24
CN101302215A (zh) 2008-11-12
YU36300A (sh) 2004-03-12
ZA9811506B (en) 2000-11-06
SA99191115B1 (ar) 2006-10-11
AU1967999A (en) 1999-07-05
JP2002508373A (ja) 2002-03-19
HUP0100509A2 (hu) 2002-05-29
NO20003069L (no) 2000-06-15
HRP20000408A2 (en) 2000-08-31
DZ2681A1 (fr) 2004-06-20
TR199802625A3 (tr) 1999-10-21
EP1661895A1 (en) 2006-05-31
NO317254B1 (no) 2004-09-27
MY135612A (en) 2008-05-30
BG64988B1 (bg) 2006-11-30
PE20000058A1 (es) 2000-02-26
OA11766A (en) 2005-07-19
CZ20002204A3 (cs) 2000-11-15
HRP20000408B1 (en) 2008-04-30
AP1365A (en) 2005-01-26
EA004260B1 (ru) 2004-02-26
EG22337A (en) 2002-12-31
SK9172000A3 (en) 2001-01-18
MA26580A1 (fr) 2004-12-20
AP2000001831A0 (en) 2000-06-30
EP1040110A1 (en) 2000-10-04
IL136424A (en) 2003-12-10
CN101381367A (zh) 2009-03-11
CN1281453A (zh) 2001-01-24
KR20010033141A (ko) 2001-04-25
PL341146A1 (en) 2001-03-26
AR017214A1 (es) 2001-08-22
GB9726566D0 (en) 1998-02-11
IL136424A0 (en) 2001-06-14
CA2314107A1 (en) 1999-06-24
CO4980880A1 (es) 2000-11-27
TR199802625A2 (xx) 1999-10-21
TR200001799T2 (tr) 2001-01-22
HUP0100509A3 (en) 2002-06-28
CZ299965B6 (cs) 2009-01-07
BG104603A (en) 2001-03-30
SK286618B6 (sk) 2009-02-05
TW509690B (en) 2002-11-11

Similar Documents

Publication Publication Date Title
NO20003069D0 (no) 5-[4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl]tiazolidin- 2,4-dion-maleinsyre-salt-hydrat som farmasøytikum
HUP0300158A3 (en) Hydrochloride salts of-5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione, method for their production and pharmaceutical compositions containing them
IL146111A0 (en) 5-[4-[2-(n-methyl-n-(2-pyridyl) amino)ethoxy]benzyl] thiazolidine-2,4-dione, maleic acid salt
NO2009002I1 (no) 5-{4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl}tiazolidin-2,4-dionmaleat(salter/solvater)+glimepirid
NO20003068L (no) Hydrat av 5-[-4-[2-(N-metyl-N-(2- pyridyl)amino)etoksy]benzyl]tiazolidin-2,4-dion-maleinsyre-salt
MXPA03001956A (es) La sal de clorhidrato de 5-[4-[2-(n-metil, -n-metil-n -(2-piridil) amino) etoxi] bencil] tiazolidin-2, 4-diona.
IL188116A0 (en) Sodium salts of 5-[4-[2-(n-methyl-n-(2-pyridyl) amino) ethoxy] benzyl] thiazolidine-2,4-dione
DK1446404T3 (da) Rosiglitazonedisylater og deres anvendelse som antidiabetika
NO20025882L (no) 5-(4-(2-(N-metyl-N-(2-pyridyl)amino)etoksy)benzyl)-tiazolidin- 2,4-dion hydriodid som farmasöytisk middel
SI1265893T1 (sl) Hidrokloridne soli 5-(4-(2-(n-metil-n-(2-piridil)amino)etoksi)benzil)tiazolidin-2,4-diona
HU0700069D0 (en) Acid addition salts of 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione different from malei acid salt
AU2002222305A1 (en) 5-'4-'2-(n-methyl-n- (2-pyridyl)amino)ethoxy!benzyl!thiazolidine-2, 4-dione mesylate salt

Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees