NO180304C - Analogifremgangsmåte for fremstilling av terapeutisk aktivt 2<beta>,19-(ethylen)androst-4-en-3,17-dion - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktivt 2<beta>,19-(ethylen)androst-4-en-3,17-dion

Info

Publication number
NO180304C
NO180304C NO914710A NO914710A NO180304C NO 180304 C NO180304 C NO 180304C NO 914710 A NO914710 A NO 914710A NO 914710 A NO914710 A NO 914710A NO 180304 C NO180304 C NO 180304C
Authority
NO
Norway
Prior art keywords
beta
preparation
therapeutically active
analogous process
compounds
Prior art date
Application number
NO914710A
Other languages
English (en)
Norwegian (no)
Other versions
NO180304B (no
NO914710L (no
NO914710D0 (no
Inventor
John O'neal Johnston
Norton Paul Peet
Joseph Paul Burkhart
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of NO914710D0 publication Critical patent/NO914710D0/no
Publication of NO914710L publication Critical patent/NO914710L/no
Publication of NO180304B publication Critical patent/NO180304B/no
Publication of NO180304C publication Critical patent/NO180304C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Bakery Products And Manufacturing Methods Therefor (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO914710A 1990-11-30 1991-11-29 Analogifremgangsmåte for fremstilling av terapeutisk aktivt 2<beta>,19-(ethylen)androst-4-en-3,17-dion NO180304C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/621,184 US5166201A (en) 1990-11-30 1990-11-30 2β,19-ethylene bridged steroids as aromatase inhibitors

Publications (4)

Publication Number Publication Date
NO914710D0 NO914710D0 (no) 1991-11-29
NO914710L NO914710L (no) 1992-06-01
NO180304B NO180304B (no) 1996-12-16
NO180304C true NO180304C (no) 1997-04-02

Family

ID=24489093

Family Applications (1)

Application Number Title Priority Date Filing Date
NO914710A NO180304C (no) 1990-11-30 1991-11-29 Analogifremgangsmåte for fremstilling av terapeutisk aktivt 2<beta>,19-(ethylen)androst-4-en-3,17-dion

Country Status (20)

Country Link
US (1) US5166201A (ja)
EP (1) EP0488383B1 (ja)
JP (1) JP3143876B2 (ja)
KR (1) KR100190776B1 (ja)
CN (1) CN1033975C (ja)
AT (1) ATE142639T1 (ja)
AU (1) AU635444B2 (ja)
CA (1) CA2056638C (ja)
DE (1) DE69122048T2 (ja)
DK (1) DK0488383T3 (ja)
ES (1) ES2094183T3 (ja)
FI (1) FI102073B1 (ja)
GR (1) GR3021981T3 (ja)
HU (1) HU210830B (ja)
IE (1) IE914168A1 (ja)
IL (1) IL100196A (ja)
NO (1) NO180304C (ja)
NZ (1) NZ240738A (ja)
PT (1) PT99661B (ja)
ZA (1) ZA919296B (ja)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19510862A1 (de) * 1995-03-16 1996-09-19 Schering Ag Verwendung von Antiestrogenen zur männlichen Fertilitätskontrolle
EP1079859B1 (en) 1998-05-22 2010-07-14 The Board Of Trustees Of The Leland Stanford Junior University Bifunctional molecules and therapies based thereon
DK1889198T3 (da) 2005-04-28 2015-02-09 Proteus Digital Health Inc Farma-informatiksystem
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
DK2398500T3 (da) 2009-02-20 2019-05-13 2 Bbb Medicines B V Glutathion-baseret lægemiddelafgivelsessystem
IL255113B (en) 2009-05-06 2022-09-01 Laboratory Skin Care Inc Preparations for administration through the skin that include complexes of an active substance with calcium phosphate and methods of using them

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3627756A (en) * 1970-04-23 1971-12-14 Searle & Co N-dialkylaminoalkyl-n-(2{62 ,19-epoxy-5{60 -androstan-17{62 -yl)amines/formamides and 3{60 -halo derivatives thereof
US4322416A (en) * 1980-06-27 1982-03-30 Merrell Dow Pharmaceuticals Inc. 10-Alkynyl steroids
GB8501035D0 (en) * 1985-01-16 1985-02-20 Senior J Prostaglandins
US4882322A (en) * 1988-10-27 1989-11-21 Merrell Dow Pharmaceuticals Inc. 3β,17β-hydroxy-substituted steroids and related steroidal compounds

Also Published As

Publication number Publication date
HUT59937A (en) 1992-07-28
US5166201A (en) 1992-11-24
PT99661A (pt) 1992-10-30
DK0488383T3 (da) 1996-09-30
AU8812891A (en) 1992-06-04
NO180304B (no) 1996-12-16
FI915623A0 (fi) 1991-11-28
AU635444B2 (en) 1993-03-18
IL100196A0 (en) 1992-08-18
EP0488383B1 (en) 1996-09-11
ZA919296B (en) 1992-08-26
DE69122048T2 (de) 1997-02-20
FI915623A (fi) 1992-05-31
CA2056638A1 (en) 1992-05-31
CN1033975C (zh) 1997-02-05
DE69122048D1 (de) 1996-10-17
HU210830B (en) 1995-08-28
IL100196A (en) 1996-03-31
IE914168A1 (en) 1992-06-03
ATE142639T1 (de) 1996-09-15
HU913739D0 (en) 1992-02-28
EP0488383A1 (en) 1992-06-03
GR3021981T3 (en) 1997-03-31
FI102073B (fi) 1998-10-15
CA2056638C (en) 2002-03-05
PT99661B (pt) 1999-05-31
KR100190776B1 (ko) 1999-06-01
CN1061974A (zh) 1992-06-17
ES2094183T3 (es) 1997-01-16
NZ240738A (en) 1993-11-25
NO914710L (no) 1992-06-01
KR920009842A (ko) 1992-06-25
NO914710D0 (no) 1991-11-29
JP3143876B2 (ja) 2001-03-07
FI102073B1 (fi) 1998-10-15
JPH04290898A (ja) 1992-10-15

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Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees

Free format text: LAPSED IN MAY 2001