NO179838C - Fremgangsmåte for fremstilling av S-(-)-3-morfolino-4-(3-tert-butylamino-2-hydroksypropoksy)-1,2,5-tiadiazol-hemihydrat - Google Patents

Fremgangsmåte for fremstilling av S-(-)-3-morfolino-4-(3-tert-butylamino-2-hydroksypropoksy)-1,2,5-tiadiazol-hemihydrat

Info

Publication number
NO179838C
NO179838C NO911508A NO911508A NO179838C NO 179838 C NO179838 C NO 179838C NO 911508 A NO911508 A NO 911508A NO 911508 A NO911508 A NO 911508A NO 179838 C NO179838 C NO 179838C
Authority
NO
Norway
Prior art keywords
hydroxypropoxy
butylamino
morpholino
tert
preparation
Prior art date
Application number
NO911508A
Other languages
English (en)
Norwegian (no)
Other versions
NO911508L (no
NO911508D0 (no
NO179838B (no
Inventor
Markku Peraelampi
Original Assignee
Leiras Oy
Huhtamaeki Yhthymae Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leiras Oy, Huhtamaeki Yhthymae Oy filed Critical Leiras Oy
Publication of NO911508L publication Critical patent/NO911508L/no
Publication of NO911508D0 publication Critical patent/NO911508D0/no
Publication of NO179838B publication Critical patent/NO179838B/no
Publication of NO179838C publication Critical patent/NO179838C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/101,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Measuring Pulse, Heart Rate, Blood Pressure Or Blood Flow (AREA)
  • Control Of El Displays (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO911508A 1988-10-20 1991-04-17 Fremgangsmåte for fremstilling av S-(-)-3-morfolino-4-(3-tert-butylamino-2-hydroksypropoksy)-1,2,5-tiadiazol-hemihydrat NO179838C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FI884838A FI82240C (fi) 1988-10-20 1988-10-20 Foerfarande foer framstaellning av farmakologiskt vaerdefullt s-timolol-hemihydrat.
PCT/FI1989/000196 WO1990004592A1 (en) 1988-10-20 1989-10-13 Novel s-timolol derivative and process for its preparation

Publications (4)

Publication Number Publication Date
NO911508L NO911508L (no) 1991-04-17
NO911508D0 NO911508D0 (no) 1991-04-17
NO179838B NO179838B (no) 1996-09-16
NO179838C true NO179838C (no) 1996-12-27

Family

ID=8527232

Family Applications (1)

Application Number Title Priority Date Filing Date
NO911508A NO179838C (no) 1988-10-20 1991-04-17 Fremgangsmåte for fremstilling av S-(-)-3-morfolino-4-(3-tert-butylamino-2-hydroksypropoksy)-1,2,5-tiadiazol-hemihydrat

Country Status (12)

Country Link
US (4) US5231095A (de)
EP (1) EP0440684B1 (de)
JP (1) JP2949508B2 (de)
AT (1) ATE112277T1 (de)
AU (1) AU624431B2 (de)
CA (1) CA2001083C (de)
DE (1) DE68918597T2 (de)
DK (1) DK175377B1 (de)
FI (1) FI82240C (de)
NO (1) NO179838C (de)
NZ (1) NZ231057A (de)
WO (1) WO1990004592A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5496820A (en) * 1988-10-20 1996-03-05 Peraelampi; Markku Ophthalmic use of S-timolol hemihydrate
FI82240C (fi) * 1988-10-20 1991-02-11 Huhtamaeki Oy Foerfarande foer framstaellning av farmakologiskt vaerdefullt s-timolol-hemihydrat.
TW208013B (de) * 1990-03-01 1993-06-21 Daiichi Co Ltd
ES2106852T3 (es) * 1992-07-08 1997-11-16 Santen Oy Composicion oftalmica que contiene hemihidrato de timolol.
US20060143783A1 (en) * 2004-12-15 2006-07-06 Berman Paul K Energy diffusing glove insert
US7862552B2 (en) 2005-05-09 2011-01-04 Boston Scientific Scimed, Inc. Medical devices for treating urological and uterine conditions
AU2008220104B2 (en) 2007-02-28 2012-09-27 Asahi Kasei Pharma Corporation Sulfonamide derivative

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3657237A (en) * 1968-05-22 1972-04-18 Frosst & Co Charles E Process for making 1 2 5-thiadiazoles in the sinister configuration
US4428883A (en) * 1981-03-06 1984-01-31 The University Of Kentucky Research Foundation Novel method of administering β-blockers and novel dosage forms containing same
FI71933C (fi) * 1984-03-30 1989-04-06 Star Oy Ab Nya l-vinsyra-0-monoestrar av 3-morfolino-4-(3'-tert.-butylamino-2'-hydroxipropoxi)-1,2,5-tiadiazol och deras anvaendning saosom mellanprodukter.
JPS60226855A (ja) * 1984-04-26 1985-11-12 Nippon Kayaku Co Ltd N−ベンジルオキシカルボニル−l−スレオニンアミド・1/2水和物およびその製造法
US4752478A (en) * 1984-12-17 1988-06-21 Merck & Co., Inc. Transdermal system for timolol
US4756710A (en) * 1985-04-05 1988-07-12 Merck & Co., Inc. pH-Mediated drug delivery system
FI82240C (fi) * 1988-10-20 1991-02-11 Huhtamaeki Oy Foerfarande foer framstaellning av farmakologiskt vaerdefullt s-timolol-hemihydrat.

Also Published As

Publication number Publication date
FI82240B (fi) 1990-10-31
AU624431B2 (en) 1992-06-11
DK72591A (da) 1991-04-19
NO911508L (no) 1991-04-17
DE68918597D1 (de) 1994-11-03
US5354860A (en) 1994-10-11
CA2001083C (en) 1999-06-15
DK72591D0 (da) 1991-04-19
JPH04502612A (ja) 1992-05-14
NO911508D0 (no) 1991-04-17
JP2949508B2 (ja) 1999-09-13
NZ231057A (en) 1990-11-27
FI884838A0 (fi) 1988-10-20
EP0440684A1 (de) 1991-08-14
EP0440684B1 (de) 1994-09-28
CA2001083A1 (en) 1990-04-20
FI884838A (fi) 1990-04-21
DE68918597T2 (de) 1995-05-11
WO1990004592A1 (en) 1990-05-03
ATE112277T1 (de) 1994-10-15
DK175377B1 (da) 2004-09-20
AU4347389A (en) 1990-05-14
US5574035A (en) 1996-11-12
FI82240C (fi) 1991-02-11
NO179838B (no) 1996-09-16
US5231095A (en) 1993-07-27
US5541184A (en) 1996-07-30

Similar Documents

Publication Publication Date Title
MY103850A (en) Phenol substituted gem-diphosphonate derivatives, process for their preparation and pharmaceutical compositions containing them.
MY102038A (en) 4-substituted androstendione derivatives and process for their preparation
IE45256L (en) Quinazolone derivatives
EP0279149A3 (en) Benzimidazole derivatives, process for their production and a pharmaceutical composition containing the same
EP0614913A3 (de) Dynorphin Derivate.
ES8606282A1 (es) Un procedimiento de preparar derivados de acidos quinolin- ynaftiridin-carboxilicos
MY108601A (en) Drug solutions of increased stability and without- tissuedamaging effect and process for preparing same
IL84409A0 (en) Imidazolidinone derivatives,their preparation and pharmaceutical compositions containing them
NO179838C (no) Fremgangsmåte for fremstilling av S-(-)-3-morfolino-4-(3-tert-butylamino-2-hydroksypropoksy)-1,2,5-tiadiazol-hemihydrat
MY102003A (en) Novel derivatives of 4, 5-dihydrooxazoles, a process for their preparation, and their use.
HUT45537A (en) Process for producing delta-22 derivatives of ll-f 28249 compounds and pharmaceutical compositions containing them as active components, and insecticide compositions
DE3565104D1 (en) Thiadiazine compound, process for its preparation and pharmaceutical compositions containing it
EP0270046A3 (en) Pharmaceutical composition for treatment of cataract
IL77051A (en) Crystalline form of the monoethanolamine salt of n-(2-pyridyl)-2-methyl-4-hydroxy-2h-1,2-benzothiazine-3-carboxamide 1,1-dioxide and pharmaceutical compositions containing it
HUT41025A (en) Process for preparing octahydro-indolizine derivatives and pharmaceutical compositions containing such compounds as active ingredients
HUT39439A (en) Process for producing new thiazolidinedione derivatives and pharmaceutical compositions containing them as active agents
GR3000512T3 (en) Pharmaceutical compositions containing 5-phenyl-1,3-dioxoalkenyl compounds
ES8800198A1 (es) Procedimiento para preparar derivados de acidos aziridin-2- carboxilicos substituidos en n
ES8501378A1 (es) Procedimiento de preparar derivados de n-cicloalcoilmetil-2 oxo-3 diaril 5-6 as triacina
HUT45059A (en) Process for producing abeoergoline derivatives
ES8601200A1 (es) Un procedimiento para preparar compuestos de 3-(2-haloetil)-4-oxopirazolo-(5, 1-d)-1, 2, 3, 5-tetrazin-8-carboxamida
ES2000614A6 (es) Procedimiento de obtencion de nuevos complejos de platino (ii) derivados del 2,3-dimercapto-2-butene-dinitrilato (2-)-s,s'"
ES8606375A1 (es) Un procedimiento para preparar un derivado de aminoprpilaminobleomicina