DK72591A - Hidtil ukendt s-timolol-derivat samt fremgangsmaade til fremstilling deraf - Google Patents
Hidtil ukendt s-timolol-derivat samt fremgangsmaade til fremstilling deraf Download PDFInfo
- Publication number
- DK72591A DK72591A DK072591A DK72591A DK72591A DK 72591 A DK72591 A DK 72591A DK 072591 A DK072591 A DK 072591A DK 72591 A DK72591 A DK 72591A DK 72591 A DK72591 A DK 72591A
- Authority
- DK
- Denmark
- Prior art keywords
- procedures
- preparing
- hitherto unknown
- timolol
- derivatives
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008177 pharmaceutical agent Substances 0.000 abstract 1
- 238000011200 topical administration Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Control Of El Displays (AREA)
- Diaphragms For Electromechanical Transducers (AREA)
- Measuring Pulse, Heart Rate, Blood Pressure Or Blood Flow (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FI884838 | 1988-10-20 | ||
| FI884838A FI82240C (fi) | 1988-10-20 | 1988-10-20 | Foerfarande foer framstaellning av farmakologiskt vaerdefullt s-timolol-hemihydrat. |
| PCT/FI1989/000196 WO1990004592A1 (en) | 1988-10-20 | 1989-10-13 | Novel s-timolol derivative and process for its preparation |
| FI8900196 | 1989-10-13 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK72591A true DK72591A (da) | 1991-04-19 |
| DK72591D0 DK72591D0 (da) | 1991-04-19 |
| DK175377B1 DK175377B1 (da) | 2004-09-20 |
Family
ID=8527232
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK199100725A DK175377B1 (da) | 1988-10-20 | 1991-04-19 | Hidtil ukendt S-timolol-derivat samt fremgangsmåde til fremstilling deraf |
Country Status (12)
| Country | Link |
|---|---|
| US (4) | US5231095A (da) |
| EP (1) | EP0440684B1 (da) |
| JP (1) | JP2949508B2 (da) |
| AT (1) | ATE112277T1 (da) |
| AU (1) | AU624431B2 (da) |
| CA (1) | CA2001083C (da) |
| DE (1) | DE68918597T2 (da) |
| DK (1) | DK175377B1 (da) |
| FI (1) | FI82240C (da) |
| NO (1) | NO179838C (da) |
| NZ (1) | NZ231057A (da) |
| WO (1) | WO1990004592A1 (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI82240C (fi) * | 1988-10-20 | 1991-02-11 | Huhtamaeki Oy | Foerfarande foer framstaellning av farmakologiskt vaerdefullt s-timolol-hemihydrat. |
| US5496820A (en) * | 1988-10-20 | 1996-03-05 | Peraelampi; Markku | Ophthalmic use of S-timolol hemihydrate |
| TW208013B (da) * | 1990-03-01 | 1993-06-21 | Daiichi Co Ltd | |
| ATE154513T1 (de) * | 1992-07-08 | 1997-07-15 | Leiras Oy | Augenarzneimittel enthaltend timolol hemihydrat |
| US20060143783A1 (en) * | 2004-12-15 | 2006-07-06 | Berman Paul K | Energy diffusing glove insert |
| US7862552B2 (en) | 2005-05-09 | 2011-01-04 | Boston Scientific Scimed, Inc. | Medical devices for treating urological and uterine conditions |
| CN101622243B (zh) | 2007-02-28 | 2013-12-04 | 旭化成制药株式会社 | 磺酰胺衍生物 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3657237A (en) * | 1968-05-22 | 1972-04-18 | Frosst & Co Charles E | Process for making 1 2 5-thiadiazoles in the sinister configuration |
| US4428883A (en) * | 1981-03-06 | 1984-01-31 | The University Of Kentucky Research Foundation | Novel method of administering β-blockers and novel dosage forms containing same |
| FI71933C (fi) * | 1984-03-30 | 1989-04-06 | Star Oy Ab | Nya l-vinsyra-0-monoestrar av 3-morfolino-4-(3'-tert.-butylamino-2'-hydroxipropoxi)-1,2,5-tiadiazol och deras anvaendning saosom mellanprodukter. |
| JPS60226855A (ja) * | 1984-04-26 | 1985-11-12 | Nippon Kayaku Co Ltd | N−ベンジルオキシカルボニル−l−スレオニンアミド・1/2水和物およびその製造法 |
| US4752478A (en) * | 1984-12-17 | 1988-06-21 | Merck & Co., Inc. | Transdermal system for timolol |
| US4756710A (en) * | 1985-04-05 | 1988-07-12 | Merck & Co., Inc. | pH-Mediated drug delivery system |
| FI82240C (fi) * | 1988-10-20 | 1991-02-11 | Huhtamaeki Oy | Foerfarande foer framstaellning av farmakologiskt vaerdefullt s-timolol-hemihydrat. |
-
1988
- 1988-10-20 FI FI884838A patent/FI82240C/fi not_active IP Right Cessation
-
1989
- 1989-10-13 AT AT89911378T patent/ATE112277T1/de not_active IP Right Cessation
- 1989-10-13 AU AU43473/89A patent/AU624431B2/en not_active Ceased
- 1989-10-13 JP JP1510608A patent/JP2949508B2/ja not_active Expired - Fee Related
- 1989-10-13 US US07/663,853 patent/US5231095A/en not_active Expired - Lifetime
- 1989-10-13 WO PCT/FI1989/000196 patent/WO1990004592A1/en not_active Ceased
- 1989-10-13 EP EP89911378A patent/EP0440684B1/en not_active Expired - Lifetime
- 1989-10-13 DE DE68918597T patent/DE68918597T2/de not_active Expired - Lifetime
- 1989-10-18 NZ NZ231057A patent/NZ231057A/en unknown
- 1989-10-20 CA CA002001083A patent/CA2001083C/en not_active Expired - Fee Related
-
1991
- 1991-04-17 NO NO911508A patent/NO179838C/no unknown
- 1991-04-19 DK DK199100725A patent/DK175377B1/da not_active IP Right Cessation
-
1992
- 1992-07-08 US US07/910,789 patent/US5354860A/en not_active Expired - Lifetime
-
1994
- 1994-10-07 US US08/319,868 patent/US5574035A/en not_active Expired - Lifetime
- 1994-10-11 US US08/320,327 patent/US5541184A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| NZ231057A (en) | 1990-11-27 |
| CA2001083A1 (en) | 1990-04-20 |
| NO179838B (no) | 1996-09-16 |
| JP2949508B2 (ja) | 1999-09-13 |
| FI82240C (fi) | 1991-02-11 |
| AU624431B2 (en) | 1992-06-11 |
| CA2001083C (en) | 1999-06-15 |
| WO1990004592A1 (en) | 1990-05-03 |
| US5231095A (en) | 1993-07-27 |
| NO911508L (no) | 1991-04-17 |
| US5354860A (en) | 1994-10-11 |
| NO179838C (no) | 1996-12-27 |
| AU4347389A (en) | 1990-05-14 |
| EP0440684A1 (en) | 1991-08-14 |
| NO911508D0 (no) | 1991-04-17 |
| JPH04502612A (ja) | 1992-05-14 |
| US5574035A (en) | 1996-11-12 |
| DK175377B1 (da) | 2004-09-20 |
| ATE112277T1 (de) | 1994-10-15 |
| FI82240B (fi) | 1990-10-31 |
| FI884838L (fi) | 1990-04-21 |
| EP0440684B1 (en) | 1994-09-28 |
| DK72591D0 (da) | 1991-04-19 |
| US5541184A (en) | 1996-07-30 |
| FI884838A0 (fi) | 1988-10-20 |
| DE68918597T2 (de) | 1995-05-11 |
| DE68918597D1 (de) | 1994-11-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUP | Patent expired |