NO172389C - Analogifremgangsmaate for fremstilling av terapeutisk aktive benzotiazoler - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive benzotiazoler

Info

Publication number
NO172389C
NO172389C NO892059A NO892059A NO172389C NO 172389 C NO172389 C NO 172389C NO 892059 A NO892059 A NO 892059A NO 892059 A NO892059 A NO 892059A NO 172389 C NO172389 C NO 172389C
Authority
NO
Norway
Prior art keywords
benzotiazoles
preparation
therapeutic active
analogue procedure
analogue
Prior art date
Application number
NO892059A
Other languages
English (en)
Norwegian (no)
Other versions
NO892059L (no
NO892059D0 (no
NO172389B (no
Inventor
Anton Franz Josef Fliri
Rodney Caughren Schnur
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO892059D0 publication Critical patent/NO892059D0/no
Publication of NO892059L publication Critical patent/NO892059L/no
Publication of NO172389B publication Critical patent/NO172389B/no
Publication of NO172389C publication Critical patent/NO172389C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
  • Graft Or Block Polymers (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO892059A 1988-05-24 1989-05-23 Analogifremgangsmaate for fremstilling av terapeutisk aktive benzotiazoler NO172389C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19803488A 1988-05-24 1988-05-24

Publications (4)

Publication Number Publication Date
NO892059D0 NO892059D0 (no) 1989-05-23
NO892059L NO892059L (no) 1989-11-27
NO172389B NO172389B (no) 1993-04-05
NO172389C true NO172389C (no) 1993-07-14

Family

ID=22731735

Family Applications (1)

Application Number Title Priority Date Filing Date
NO892059A NO172389C (no) 1988-05-24 1989-05-23 Analogifremgangsmaate for fremstilling av terapeutisk aktive benzotiazoler

Country Status (25)

Country Link
EP (1) EP0343893B1 (de)
JP (1) JPH0678331B2 (de)
KR (1) KR910006864B1 (de)
CN (1) CN1023700C (de)
AT (1) ATE79114T1 (de)
AU (1) AU601905B2 (de)
CA (1) CA1328871C (de)
DD (1) DD283815A5 (de)
DE (1) DE68902358T2 (de)
DK (1) DK249389A (de)
ES (1) ES2043012T3 (de)
FI (1) FI892498A (de)
GR (1) GR3005844T3 (de)
HU (1) HU202507B (de)
IE (1) IE891667L (de)
IL (1) IL90337A0 (de)
MX (1) MX173140B (de)
MY (1) MY106035A (de)
NO (1) NO172389C (de)
NZ (1) NZ229234A (de)
PL (1) PL154875B1 (de)
PT (1) PT90622B (de)
SU (1) SU1681728A3 (de)
YU (1) YU47019B (de)
ZA (1) ZA893862B (de)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2790299B2 (ja) * 1989-02-01 1998-08-27 保土谷化学工業株式会社 ペンゾチアゾール誘導体
US5262400A (en) * 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
US6100423A (en) * 1995-08-30 2000-08-08 G. D. Searle & Co. Amino benzenepropanoic acid compounds and derivatives thereof
AU702487B2 (en) * 1995-08-30 1999-02-25 G.D. Searle & Co. Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
US5716281A (en) * 1995-11-27 1998-02-10 Sega Enterprises, Ltd. Game apparatus using a vehicle with an optical image synthesizing system
TW513418B (en) * 1996-07-31 2002-12-11 Otsuka Pharma Co Ltd Thiazole derivatives, their production and use
AU744281B2 (en) 1997-11-10 2002-02-21 Bristol-Myers Squibb Company Benzothiazole protein tyrosine kinase inhibitors
EP0928793B1 (de) * 1998-01-02 2002-05-15 F. Hoffmann-La Roche Ag Thiazol-Derivate
WO1999052861A1 (de) * 1998-04-09 1999-10-21 Institut für Diagnostikforschung GmbH an der Freien Universität Berlin Neue benzylguanidinderivate für die therapie, in-vivo- und in-vitro-diagnostik
BR0112395A (pt) 2000-06-21 2003-07-08 Hoffmann La Roche Derivados de benzotiazol
US6624163B2 (en) * 2001-11-29 2003-09-23 Hoffman-La Roche Inc. Benzothiazole derivatives
GB0130868D0 (en) 2001-12-24 2002-02-06 Univ Strathclyde New compounds
CN100357283C (zh) * 2002-04-02 2007-12-26 中国科学院上海药物研究所 一类甲硫氨酰氨肽酶抑制剂
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
PT1753760E (pt) 2004-05-24 2008-02-12 Hoffmann La Roche '' - metoxi - 7 - morfolin - 4 - il - benzotiazol - 2 - il) - amida do ácido 4 - hidroxi - 4 - metil - piperidina - 1 - carboxílico''
ES2309814T3 (es) 2004-11-05 2008-12-16 F. Hoffmann-La Roche Ag Proceso para la obtencion de derivados del acido isonicotinico.
RU2412943C2 (ru) 2005-03-23 2011-02-27 Ф. Хоффманн-Ля Рош Аг ПРОИЗВОДНЫЕ АЦЕТИЛЕНИЛ-ПИРАЗОЛО-ПИРИМИДИНА В КАЧЕСТВЕ АНТАГОНИСТОВ mGluR2
JP5048675B2 (ja) 2005-09-27 2012-10-17 エフ.ホフマン−ラ ロシュ アーゲー mGluR2アンタゴニストとしてのオキサジアゾリルピラゾロ−ピリミジン類
CN101405278A (zh) * 2006-03-15 2009-04-08 4Sc股份公司 新颖的杂环NF-κB抑制剂
GB0619325D0 (en) 2006-09-30 2006-11-08 Univ Strathclyde New compounds
US20110178070A1 (en) * 2008-06-24 2011-07-21 Takeda Pharmaceutical Company Limited PI3K/mTOR INHIBITORS
US9499790B2 (en) 2010-08-26 2016-11-22 Kyoto University Method for promoting differentiation of pluripotent stem cells into cardiac muscle cells
KR20140070631A (ko) * 2011-09-30 2014-06-10 키네타, 인크. 항바이러스 화합물
EP2808383B1 (de) 2012-01-27 2018-07-25 Kyoto University Verfahren zur induktion der kardialen differenzierung pluripotenter stammzellen
WO2014136519A1 (ja) 2013-03-08 2014-09-12 国立大学法人京都大学 Egf受容体阻害剤を含む多能性幹細胞の心筋分化促進剤
EP3045451B1 (de) * 2013-09-13 2018-03-28 Kyoto University Verfahren zur induzierung der differenzierung pluripotenter stammzellen in kardiomyozyten
EP3150705B1 (de) 2014-05-30 2019-05-15 Kyoto University Verfahren zur induktion von myokardialer differenzierung von pluripotenten stammzellen mithilfe einer verbindung mit niedrigem molekulargewicht
CN109776486A (zh) * 2019-02-26 2019-05-21 武汉松石科技股份有限公司 一种硫酸亚丙酯的制备方法
CN110590735B (zh) * 2019-09-30 2021-07-23 江苏国泰超威新材料有限公司 一种环状硫酸酯的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61225168A (ja) * 1985-03-30 1986-10-06 Nippon Tokushu Noyaku Seizo Kk 新規ベンズアミド、その製法及び殺虫剤
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법
GB8611606D0 (en) * 1986-05-13 1986-06-18 Fbc Ltd Fungicides

Also Published As

Publication number Publication date
EP0343893A1 (de) 1989-11-29
ES2043012T3 (es) 1993-12-16
MY106035A (en) 1995-03-31
KR910006864B1 (ko) 1991-09-09
EP0343893B1 (de) 1992-08-05
PL154875B1 (en) 1991-09-30
JPH0678331B2 (ja) 1994-10-05
AU601905B2 (en) 1990-09-20
NO892059L (no) 1989-11-27
MX173140B (es) 1994-02-02
NZ229234A (en) 1990-09-26
IE891667L (en) 1989-11-24
HUT51606A (en) 1990-05-28
DK249389D0 (da) 1989-05-23
FI892498A (fi) 1989-11-25
DD283815A5 (de) 1990-10-24
MX16158A (es) 1993-06-01
HU202507B (en) 1991-03-28
YU105989A (en) 1990-08-31
FI892498A0 (fi) 1989-05-23
NO892059D0 (no) 1989-05-23
CN1037898A (zh) 1989-12-13
GR3005844T3 (de) 1993-06-07
DE68902358T2 (de) 1992-12-10
JPH0217181A (ja) 1990-01-22
ZA893862B (en) 1991-01-30
DE68902358D1 (de) 1992-09-10
NO172389B (no) 1993-04-05
PT90622B (pt) 1994-10-31
ATE79114T1 (de) 1992-08-15
SU1681728A3 (ru) 1991-09-30
CA1328871C (en) 1994-04-26
KR890017248A (ko) 1989-12-15
IL90337A0 (en) 1989-12-15
CN1023700C (zh) 1994-02-09
DK249389A (da) 1989-11-27
AU3509889A (en) 1989-11-30
PT90622A (pt) 1989-11-30
YU47019B (sh) 1994-11-15
PL279613A1 (en) 1989-11-27

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