NL8403447A - Farmaceutische tabletten met vertraagde afgifte en werkwijze voor de bereiding ervan. - Google Patents
Farmaceutische tabletten met vertraagde afgifte en werkwijze voor de bereiding ervan. Download PDFInfo
- Publication number
- NL8403447A NL8403447A NL8403447A NL8403447A NL8403447A NL 8403447 A NL8403447 A NL 8403447A NL 8403447 A NL8403447 A NL 8403447A NL 8403447 A NL8403447 A NL 8403447A NL 8403447 A NL8403447 A NL 8403447A
- Authority
- NL
- Netherlands
- Prior art keywords
- active ingredient
- tablets
- process according
- granulation
- weight
- Prior art date
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- 229910052749 magnesium Inorganic materials 0.000 description 1
- 229960004815 meprobamate Drugs 0.000 description 1
- 239000002207 metabolite Substances 0.000 description 1
- YLGXILFCIXHCMC-JHGZEJCSSA-N methyl cellulose Chemical compound COC1C(OC)C(OC)C(COC)O[C@H]1O[C@H]1C(OC)C(OC)C(OC)OC1COC YLGXILFCIXHCMC-JHGZEJCSSA-N 0.000 description 1
- IUBSYMUCCVWXPE-UHFFFAOYSA-N metoprolol Chemical compound COCCC1=CC=C(OCC(O)CNC(C)C)C=C1 IUBSYMUCCVWXPE-UHFFFAOYSA-N 0.000 description 1
- 229960002237 metoprolol Drugs 0.000 description 1
- 239000000178 monomer Substances 0.000 description 1
- 229960003057 nialamide Drugs 0.000 description 1
- 229940060184 oil ingredients Drugs 0.000 description 1
- 229960005489 paracetamol Drugs 0.000 description 1
- 229950000688 phenothiazine Drugs 0.000 description 1
- 230000000704 physical effect Effects 0.000 description 1
- 239000006069 physical mixture Substances 0.000 description 1
- 229960002508 pindolol Drugs 0.000 description 1
- 229920000058 polyacrylate Polymers 0.000 description 1
- 229920002959 polymer blend Polymers 0.000 description 1
- 238000006116 polymerization reaction Methods 0.000 description 1
- 229960004482 quinidine sulfate Drugs 0.000 description 1
- 230000009467 reduction Effects 0.000 description 1
- 239000004208 shellac Substances 0.000 description 1
- 235000013874 shellac Nutrition 0.000 description 1
- 229940113147 shellac Drugs 0.000 description 1
- ZLGIYFNHBLSMPS-ATJNOEHPSA-N shellac Chemical compound OCCCCCC(O)C(O)CCCCCCCC(O)=O.C1C23[C@H](C(O)=O)CCC2[C@](C)(CO)[C@@H]1C(C(O)=O)=C[C@@H]3O ZLGIYFNHBLSMPS-ATJNOEHPSA-N 0.000 description 1
- 238000007873 sieving Methods 0.000 description 1
- 239000011734 sodium Substances 0.000 description 1
- 238000002798 spectrophotometry method Methods 0.000 description 1
- 238000005507 spraying Methods 0.000 description 1
- 229910001220 stainless steel Inorganic materials 0.000 description 1
- 239000010935 stainless steel Substances 0.000 description 1
- 239000007858 starting material Substances 0.000 description 1
- 229940114926 stearate Drugs 0.000 description 1
- 239000002344 surface layer Substances 0.000 description 1
- 238000013268 sustained release Methods 0.000 description 1
- 239000012730 sustained-release form Substances 0.000 description 1
- 229960000195 terbutaline Drugs 0.000 description 1
- XCTYLCDETUVOIP-UHFFFAOYSA-N thiethylperazine Chemical compound C12=CC(SCC)=CC=C2SC2=CC=CC=C2N1CCCN1CCN(C)CC1 XCTYLCDETUVOIP-UHFFFAOYSA-N 0.000 description 1
- 229960002784 thioridazine Drugs 0.000 description 1
- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
- 229960001082 trimethoprim Drugs 0.000 description 1
- 235000019154 vitamin C Nutrition 0.000 description 1
- 239000011718 vitamin C Substances 0.000 description 1
- 229920003176 water-insoluble polymer Polymers 0.000 description 1
- 229920003169 water-soluble polymer Polymers 0.000 description 1
- 230000004584 weight gain Effects 0.000 description 1
- 235000019786 weight gain Nutrition 0.000 description 1
- 238000009736 wetting Methods 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU385983 | 1983-11-11 | ||
| HU833859A HU190619B (en) | 1983-11-11 | 1983-11-11 | Process for producing tablets with controlled dissolution of active ingredients |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NL8403447A true NL8403447A (nl) | 1985-06-03 |
Family
ID=10965801
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL8403447A NL8403447A (nl) | 1983-11-11 | 1984-11-09 | Farmaceutische tabletten met vertraagde afgifte en werkwijze voor de bereiding ervan. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4647599A (de) |
| JP (1) | JPH0751497B2 (de) |
| AT (1) | AT391078B (de) |
| BE (1) | BE901007A (de) |
| CH (1) | CH665124A5 (de) |
| DD (1) | DD229030A5 (de) |
| DE (1) | DE3441308C2 (de) |
| FI (1) | FI78614C (de) |
| FR (1) | FR2554717B1 (de) |
| GB (1) | GB2149413B (de) |
| HU (1) | HU190619B (de) |
| NL (1) | NL8403447A (de) |
| SE (1) | SE455571B (de) |
| SU (1) | SU1577684A3 (de) |
| UA (1) | UA5328A1 (de) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2201594B (en) * | 1986-06-24 | 1991-02-13 | Istvan Racz | Production of acid binding pharmaceutical preparations |
| HU196711B (en) * | 1986-06-24 | 1989-01-30 | Istvan Racz | Process for producing long-acting, gastric acid neutralizing pharmaceutics with high acid-binding capacity and increased bioavailability |
| US4844908A (en) * | 1986-11-27 | 1989-07-04 | Duphar International Research B.V. | Method of preparing tablets with clovoxamine fumarate and tablets thus prepared |
| US4853229A (en) * | 1987-10-26 | 1989-08-01 | Alza Corporation | Method for adminstering tiny pills |
| US4961932A (en) * | 1987-10-26 | 1990-10-09 | Alza Corporation | Plurality of tiny pills in liquid dosage form |
| US5030454A (en) * | 1987-10-26 | 1991-07-09 | Alza Corporation | Method for delivering drug in tiny pills in liquid carrier |
| CA1334379C (en) * | 1987-11-24 | 1995-02-14 | James William Mcginity | Method for preparing a solid sustained release form of a functionally active composition |
| US5051261A (en) * | 1987-11-24 | 1991-09-24 | Fmc Corporation | Method for preparing a solid sustained release form of a functionally active composition |
| US4927639A (en) * | 1989-02-02 | 1990-05-22 | Warner-Lambert Company | Modified release gemfibrozil composition |
| US4925676A (en) * | 1989-02-02 | 1990-05-15 | Warner-Lambert Company | Extended release gemfibrozil composition |
| US4971804A (en) * | 1989-02-02 | 1990-11-20 | Warner-Lambert Company | Water dispersible gemfibrozil compositions |
| DE4138513A1 (de) * | 1991-11-23 | 1993-05-27 | Basf Ag | Feste pharmazeutische retardform |
| ES2061394B1 (es) * | 1993-02-05 | 1995-06-16 | Robert S A Lab | Procedimiento de fabricacion de un granulado de citrato potasico con cesion retardada. |
| JP3732557B2 (ja) * | 1995-07-12 | 2006-01-05 | 住友精化株式会社 | カルボキシル基含有重合体組成物 |
| RU2123330C1 (ru) * | 1997-04-02 | 1998-12-20 | Фармацевтическая фирма "Здоровье" | Способ получения таблетированной формы препарата |
| US6492488B1 (en) | 1998-08-02 | 2002-12-10 | Pmd Holdings Corp. | Controlled release polyacrylic acid granules and a process for preparing the same |
| DE19836646A1 (de) * | 1998-08-13 | 2000-02-17 | Basf Ag | Verwendung von N-Vinylpyrrolidon- und Vinylacetat-haltigen Copolymeren als Matrix zur Herstellung von festen, oralen pharmazeutischen und kosmetischen Zubereitungen |
| KR100407519B1 (ko) * | 2001-08-31 | 2003-12-18 | 부광약품 주식회사 | 건조황산제일철과 방출조절제로서 엘-글루타민을 함유하는서방성 정제 및 그의 제조방법 |
| RU2191571C1 (ru) * | 2001-12-05 | 2002-10-27 | Нестерук Владимир Викторович | Способ получения таблеток на основе хлоропирамина |
| CA2534039A1 (en) * | 2003-08-19 | 2005-03-03 | Polybiomed Limited | Polymeric drug release system for medical devices |
| US7846466B2 (en) * | 2004-06-10 | 2010-12-07 | Northwestern University | Biodegradable scaffolds and uses thereof |
| PL2010158T3 (pl) * | 2006-04-26 | 2016-09-30 | Formulacje o kontrolowanym uwalnianiu zawierające niepowlekaną odrębną jednostkę(-i) i macierz o przedłużonym uwalnianiu | |
| GB0707127D0 (en) * | 2007-04-13 | 2007-05-23 | Zysis Ltd | Pharmaceutical compositions |
| CA2798885C (en) | 2010-05-10 | 2014-11-18 | Euro-Celtique S.A. | Combination of active loaded granules with additional actives |
| MX347105B (es) | 2010-05-10 | 2017-04-12 | Euro Celtique Sa | Composiciones farmaceuticas que comprenden hidromorfona y naloxona. |
| CA2798884C (en) * | 2010-05-10 | 2016-09-13 | Euro-Celtique S.A. | Manufacturing of active-free granules and tablets comprising the same |
| AU2013304942A1 (en) * | 2012-08-23 | 2015-03-05 | Cardiolynx Ag | Extended release compositions of an aminoalkyl nitrate |
| EP3068397A1 (de) | 2013-11-13 | 2016-09-21 | Euro-Celtique S.A. | Hydromorphon und naloxon zur behandlung von schmerzen und opioid-reizdarm-dysfunktionssyndrom |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2909462A (en) * | 1955-12-08 | 1959-10-20 | Bristol Myers Co | Acrylic acid polymer laxative compositions |
| DE1467781A1 (de) * | 1963-07-15 | 1968-12-05 | Boehringer Sohn Ingelheim | Verfahren zur Herstellung von Dragees mit verlaengerter Wirkstofffreigabe |
| US3458622A (en) * | 1967-04-07 | 1969-07-29 | Squibb & Sons Inc | Controlled release tablet |
| US3634584A (en) * | 1969-02-13 | 1972-01-11 | American Home Prod | Sustained action dosage form |
| US3590117A (en) * | 1969-03-24 | 1971-06-29 | Richardson Merrell Inc | Long-lasting troche containing guar gum |
| US3870790A (en) * | 1970-01-22 | 1975-03-11 | Forest Laboratories | Solid pharmaceutical formulations containing hydroxypropyl methyl cellulose |
| SE353229B (de) * | 1970-06-04 | 1973-01-29 | Haessle Ab | |
| FR2247206B1 (de) * | 1973-01-24 | 1978-02-03 | Sterwin Ag | |
| US3923974A (en) * | 1973-04-23 | 1975-12-02 | Sterling Drug Inc | Solid fine crystalline paracetamol polymer complex composition |
| US3851032A (en) | 1973-04-23 | 1974-11-26 | Sterling Drug Inc | Process of preparing a solid fine crystalline paracetamol polymer complex composition |
| ZA765931B (en) * | 1975-10-10 | 1977-09-28 | Squibb & Sons Inc | Controlled release tablet |
| FI63335B (fi) * | 1979-02-02 | 1983-02-28 | Orion Yhtymae Oy | Foerfarande foer framstaellning av tabletter med foerdroejd loslighet av effektaemne |
| US4252786A (en) * | 1979-11-16 | 1981-02-24 | E. R. Squibb & Sons, Inc. | Controlled release tablet |
| IL61721A (en) * | 1980-12-16 | 1984-03-30 | Blank Izhak | Nitroglycerin preparations |
| HU183408B (en) * | 1981-04-28 | 1984-05-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing oral ratard pharmaceutical compositions |
| ZA822995B (en) * | 1981-05-21 | 1983-12-28 | Wyeth John & Brother Ltd | Slow release pharmaceutical composition |
| US4557925A (en) * | 1982-07-08 | 1985-12-10 | Ab Ferrosan | Membrane-coated sustained-release tablets and method |
-
1983
- 1983-11-11 HU HU833859A patent/HU190619B/hu unknown
-
1984
- 1984-11-05 CH CH5287/84A patent/CH665124A5/de not_active IP Right Cessation
- 1984-11-08 FR FR8416990A patent/FR2554717B1/fr not_active Expired
- 1984-11-08 BE BE1/011132A patent/BE901007A/fr not_active IP Right Cessation
- 1984-11-09 FI FI844405A patent/FI78614C/fi not_active IP Right Cessation
- 1984-11-09 DD DD84269319A patent/DD229030A5/de not_active IP Right Cessation
- 1984-11-09 AT AT3550/84A patent/AT391078B/de not_active IP Right Cessation
- 1984-11-09 SU SU843814617A patent/SU1577684A3/ru active
- 1984-11-09 US US06/669,945 patent/US4647599A/en not_active Expired - Fee Related
- 1984-11-09 NL NL8403447A patent/NL8403447A/nl active Search and Examination
- 1984-11-09 UA UA3814617A patent/UA5328A1/uk unknown
- 1984-11-09 GB GB08428369A patent/GB2149413B/en not_active Expired
- 1984-11-09 SE SE8405615A patent/SE455571B/sv not_active IP Right Cessation
- 1984-11-09 JP JP59235318A patent/JPH0751497B2/ja not_active Expired - Lifetime
- 1984-11-12 DE DE3441308A patent/DE3441308C2/de not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| SE455571B (sv) | 1988-07-25 |
| JPS60222413A (ja) | 1985-11-07 |
| GB8428369D0 (en) | 1984-12-19 |
| US4647599A (en) | 1987-03-03 |
| HU190619B (en) | 1986-09-29 |
| BE901007A (fr) | 1985-05-08 |
| SU1577684A3 (ru) | 1990-07-07 |
| DE3441308A1 (de) | 1985-05-23 |
| SE8405615L (sv) | 1985-05-12 |
| FI78614B (fi) | 1989-05-31 |
| ATA355084A (de) | 1990-02-15 |
| UA5328A1 (uk) | 1994-12-28 |
| DE3441308C2 (de) | 1994-03-31 |
| CH665124A5 (de) | 1988-04-29 |
| FI78614C (fi) | 1989-09-11 |
| SE8405615D0 (sv) | 1984-11-09 |
| FR2554717B1 (fr) | 1988-05-13 |
| FI844405L (fi) | 1985-05-12 |
| FI844405A0 (fi) | 1984-11-09 |
| GB2149413B (en) | 1987-04-08 |
| AT391078B (de) | 1990-08-10 |
| DD229030A5 (de) | 1985-10-30 |
| FR2554717A1 (fr) | 1985-05-17 |
| HUT34892A (en) | 1985-05-28 |
| JPH0751497B2 (ja) | 1995-06-05 |
| GB2149413A (en) | 1985-06-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BA | A request for search or an international-type search has been filed | ||
| BB | A search report has been drawn up | ||
| BC | A request for examination has been filed | ||
| BN | A decision not to publish the application has become irrevocable |