NL7800114A - 4-gesubstitueerde imidazo(1,2-a)chinoxalinen en tussenprodukten, en werkwijze om deze te berei- den. - Google Patents

4-gesubstitueerde imidazo(1,2-a)chinoxalinen en tussenprodukten, en werkwijze om deze te berei- den.

Info

Publication number
NL7800114A
NL7800114A NL7800114A NL7800114A NL7800114A NL 7800114 A NL7800114 A NL 7800114A NL 7800114 A NL7800114 A NL 7800114A NL 7800114 A NL7800114 A NL 7800114A NL 7800114 A NL7800114 A NL 7800114A
Authority
NL
Netherlands
Prior art keywords
quinoxalines
intermediates
preparing
substituted imidazo
imidazo
Prior art date
Application number
NL7800114A
Other languages
English (en)
Dutch (nl)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of NL7800114A publication Critical patent/NL7800114A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Transplantation (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NL7800114A 1977-01-07 1978-01-04 4-gesubstitueerde imidazo(1,2-a)chinoxalinen en tussenprodukten, en werkwijze om deze te berei- den. NL7800114A (nl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75764077A 1977-01-07 1977-01-07

Publications (1)

Publication Number Publication Date
NL7800114A true NL7800114A (nl) 1978-07-11

Family

ID=25048641

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7800114A NL7800114A (nl) 1977-01-07 1978-01-04 4-gesubstitueerde imidazo(1,2-a)chinoxalinen en tussenprodukten, en werkwijze om deze te berei- den.

Country Status (19)

Country Link
US (1) US4160097A (US20100223739A1-20100909-C00025.png)
JP (2) JPS5387398A (US20100223739A1-20100909-C00025.png)
AU (1) AU521807B2 (US20100223739A1-20100909-C00025.png)
BE (1) BE862608A (US20100223739A1-20100909-C00025.png)
CA (1) CA1149385A (US20100223739A1-20100909-C00025.png)
CH (2) CH636102A5 (US20100223739A1-20100909-C00025.png)
CS (1) CS200232B2 (US20100223739A1-20100909-C00025.png)
DE (2) DE2858766C2 (US20100223739A1-20100909-C00025.png)
DK (1) DK157024C (US20100223739A1-20100909-C00025.png)
FI (1) FI64374C (US20100223739A1-20100909-C00025.png)
FR (1) FR2376858A1 (US20100223739A1-20100909-C00025.png)
GB (2) GB1579499A (US20100223739A1-20100909-C00025.png)
GR (1) GR73168B (US20100223739A1-20100909-C00025.png)
IE (1) IE46191B1 (US20100223739A1-20100909-C00025.png)
LU (1) LU78813A1 (US20100223739A1-20100909-C00025.png)
NL (1) NL7800114A (US20100223739A1-20100909-C00025.png)
SE (2) SE436359B (US20100223739A1-20100909-C00025.png)
YU (1) YU44663B (US20100223739A1-20100909-C00025.png)
ZA (1) ZA7827B (US20100223739A1-20100909-C00025.png)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE439308B (sv) * 1978-08-02 1985-06-10 Roussel Uclaf Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav
JPS5569567A (en) * 1978-11-21 1980-05-26 Eisai Co Ltd Novel imidazole compound, and antidepressant containing the same
IT1209431B (it) * 1980-11-28 1989-07-16 Angeli Inst Spa Imidazolilfenil amidine, processi per la loro preparazione e loro impiego farmaceutico, ed intermedi di preparazione.
DE3830054A1 (de) * 1988-09-03 1990-03-15 Boehringer Mannheim Gmbh Phenylamide - verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
JPH0349309U (US20100223739A1-20100909-C00025.png) * 1989-09-21 1991-05-14
US6235740B1 (en) 1997-08-25 2001-05-22 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
US6635626B1 (en) 1997-08-25 2003-10-21 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
AU9651198A (en) 1997-11-11 1999-05-31 Ono Pharmaceutical Co. Ltd. Fused pyrazine compounds
WO1999045009A1 (en) * 1998-03-04 1999-09-10 Bristol-Myers Squibb Company Heterocyclo-substituted imidazopyrazine protein tyrosine kinase inhibitors
US6869956B2 (en) * 2000-10-03 2005-03-22 Bristol-Myers Squibb Company Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
DE60117835T2 (de) 2000-10-03 2006-10-19 Bristol-Myers Squibb Co. Amino- substituierte tetracyclische Verbindungen,die als entzündungshemmende Mittel nützlich sind, und diese enthaltende Arzneimittel
WO2002060386A2 (en) * 2001-02-01 2002-08-08 Bristol-Myers Squibb Company METHODS OF TREATING INFLAMMATORY AND IMMUNE DISEASES USING INHIBITORS OF IλB KINASE (IKK)
JP2010504362A (ja) * 2006-09-25 2010-02-12 アレテ セラピューティクス, インコーポレイテッド 可溶性エポキシドヒドロラーゼ阻害剤

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3541109A (en) * 1968-06-25 1970-11-17 Du Pont 1-substituted imidazoles useful in acth reserve assay
US4011236A (en) * 1968-09-09 1977-03-08 Merck & Co., Inc. N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (uv) light absorbers
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
US3994893A (en) 1975-11-03 1976-11-30 E. R. Squibb & Sons, Inc. 4-Amino derivatives of pyrozolo[1,5-a]quinoxaline-3-carboxylic acid and esters

Also Published As

Publication number Publication date
AU521807B2 (en) 1982-04-29
FI64374C (fi) 1983-11-10
SE8300945L (sv) 1983-02-21
FI64374B (fi) 1983-07-29
FR2376858B1 (US20100223739A1-20100909-C00025.png) 1980-10-24
IE780037L (en) 1978-07-07
DE2858766C2 (US20100223739A1-20100909-C00025.png) 1990-04-05
SE8300945D0 (sv) 1983-02-21
BE862608A (fr) 1978-07-03
GR73168B (US20100223739A1-20100909-C00025.png) 1984-02-14
DE2800480A1 (de) 1978-07-13
DK157024B (da) 1989-10-30
DK4278A (da) 1978-07-08
JPH0130825B2 (US20100223739A1-20100909-C00025.png) 1989-06-22
SE7800138L (sv) 1978-07-08
JPS6259110B2 (US20100223739A1-20100909-C00025.png) 1987-12-09
FR2376858A1 (fr) 1978-08-04
IE46191B1 (en) 1983-03-23
JPS61171470A (ja) 1986-08-02
DE2800480C2 (US20100223739A1-20100909-C00025.png) 1990-04-12
ZA7827B (en) 1979-01-31
CA1149385A (en) 1983-07-05
SE460477B (sv) 1989-10-16
SE436359B (sv) 1984-12-03
FI780023A (fi) 1978-07-08
GB1579498A (en) 1980-11-19
YU2178A (en) 1990-04-30
CH636102A5 (fr) 1983-05-13
CS200232B2 (en) 1980-08-29
AU3233178A (en) 1979-07-19
GB1579499A (en) 1980-11-19
US4160097A (en) 1979-07-03
DK157024C (da) 1990-04-02
CH640229A5 (fr) 1983-12-30
JPS5387398A (en) 1978-08-01
LU78813A1 (fr) 1978-09-18
YU44663B (en) 1990-12-31

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
DNT Communications of changes of names of applicants whose applications have been laid open to public inspection

Free format text: BRISTOL-MYERS SQUIBB COMPANY

BV The patent application has lapsed