LU78813A1 - Nouvelles imidazo(1,2-a)quinoxalines substituees en position 4,leur procede de preparation et medicament les contenant - Google Patents

Nouvelles imidazo(1,2-a)quinoxalines substituees en position 4,leur procede de preparation et medicament les contenant

Info

Publication number
LU78813A1
LU78813A1 LU78813A LU78813A LU78813A1 LU 78813 A1 LU78813 A1 LU 78813A1 LU 78813 A LU78813 A LU 78813A LU 78813 A LU78813 A LU 78813A LU 78813 A1 LU78813 A1 LU 78813A1
Authority
LU
Luxembourg
Prior art keywords
quinoxalines
substituted
preparation
product containing
medicinal product
Prior art date
Application number
LU78813A
Other languages
English (en)
Inventor
P Warner
E Luber
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of LU78813A1 publication Critical patent/LU78813A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Transplantation (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
LU78813A 1977-01-07 1978-01-05 Nouvelles imidazo(1,2-a)quinoxalines substituees en position 4,leur procede de preparation et medicament les contenant LU78813A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75764077A 1977-01-07 1977-01-07

Publications (1)

Publication Number Publication Date
LU78813A1 true LU78813A1 (fr) 1978-09-18

Family

ID=25048641

Family Applications (1)

Application Number Title Priority Date Filing Date
LU78813A LU78813A1 (fr) 1977-01-07 1978-01-05 Nouvelles imidazo(1,2-a)quinoxalines substituees en position 4,leur procede de preparation et medicament les contenant

Country Status (19)

Country Link
US (1) US4160097A (fr)
JP (2) JPS5387398A (fr)
AU (1) AU521807B2 (fr)
BE (1) BE862608A (fr)
CA (1) CA1149385A (fr)
CH (2) CH636102A5 (fr)
CS (1) CS200232B2 (fr)
DE (2) DE2858766C2 (fr)
DK (1) DK157024C (fr)
FI (1) FI64374C (fr)
FR (1) FR2376858A1 (fr)
GB (2) GB1579499A (fr)
GR (1) GR73168B (fr)
IE (1) IE46191B1 (fr)
LU (1) LU78813A1 (fr)
NL (1) NL7800114A (fr)
SE (2) SE436359B (fr)
YU (1) YU44663B (fr)
ZA (1) ZA7827B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE439308B (sv) * 1978-08-02 1985-06-10 Roussel Uclaf Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav
JPS5569567A (en) * 1978-11-21 1980-05-26 Eisai Co Ltd Novel imidazole compound, and antidepressant containing the same
IT1209431B (it) * 1980-11-28 1989-07-16 Angeli Inst Spa Imidazolilfenil amidine, processi per la loro preparazione e loro impiego farmaceutico, ed intermedi di preparazione.
DE3830054A1 (de) * 1988-09-03 1990-03-15 Boehringer Mannheim Gmbh Phenylamide - verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
JPH0349309U (fr) * 1989-09-21 1991-05-14
US6235740B1 (en) 1997-08-25 2001-05-22 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
US6635626B1 (en) 1997-08-25 2003-10-21 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
AU9651198A (en) 1997-11-11 1999-05-31 Ono Pharmaceutical Co. Ltd. Fused pyrazine compounds
CA2322311C (fr) * 1998-03-04 2009-10-13 Bristol-Myers Squibb Company Inhibiteurs de la proteine tyrosine kinase, a base d'imidazopyrazine a substitution heterocyclo
US6869956B2 (en) * 2000-10-03 2005-03-22 Bristol-Myers Squibb Company Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
ES2260300T3 (es) 2000-10-03 2006-11-01 Bristol-Myers Squibb Company Compuestos tetraciclicos sustituidos con amino utiles como agentes antiinflamatorios y composiciones farmaceuticas que comprenden los mismos.
CZ20032287A3 (cs) * 2001-02-01 2004-02-18 Bristol-Myers Squibb Company Způsoby léčení zánětlivých a imunitních nemocí za použití inhibitorů IkB kinázy (IKK)
US20080076770A1 (en) * 2006-09-25 2008-03-27 Arete Therapeutics, Inc. Soluble epoxide hydrolase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3541109A (en) * 1968-06-25 1970-11-17 Du Pont 1-substituted imidazoles useful in acth reserve assay
US4011236A (en) * 1968-09-09 1977-03-08 Merck & Co., Inc. N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (uv) light absorbers
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
US3994893A (en) 1975-11-03 1976-11-30 E. R. Squibb & Sons, Inc. 4-Amino derivatives of pyrozolo[1,5-a]quinoxaline-3-carboxylic acid and esters

Also Published As

Publication number Publication date
YU2178A (en) 1990-04-30
IE46191B1 (en) 1983-03-23
CH636102A5 (fr) 1983-05-13
CH640229A5 (fr) 1983-12-30
FI64374B (fi) 1983-07-29
FR2376858B1 (fr) 1980-10-24
SE436359B (sv) 1984-12-03
DK4278A (da) 1978-07-08
JPS61171470A (ja) 1986-08-02
CA1149385A (fr) 1983-07-05
GB1579498A (en) 1980-11-19
FR2376858A1 (fr) 1978-08-04
BE862608A (fr) 1978-07-03
CS200232B2 (en) 1980-08-29
NL7800114A (nl) 1978-07-11
DK157024B (da) 1989-10-30
SE8300945D0 (sv) 1983-02-21
AU521807B2 (en) 1982-04-29
US4160097A (en) 1979-07-03
JPH0130825B2 (fr) 1989-06-22
DK157024C (da) 1990-04-02
AU3233178A (en) 1979-07-19
DE2800480C2 (fr) 1990-04-12
IE780037L (en) 1978-07-07
FI64374C (fi) 1983-11-10
FI780023A (fi) 1978-07-08
SE460477B (sv) 1989-10-16
SE8300945L (sv) 1983-02-21
JPS5387398A (en) 1978-08-01
GR73168B (fr) 1984-02-14
JPS6259110B2 (fr) 1987-12-09
DE2858766C2 (fr) 1990-04-05
SE7800138L (sv) 1978-07-08
ZA7827B (en) 1979-01-31
DE2800480A1 (de) 1978-07-13
YU44663B (en) 1990-12-31
GB1579499A (en) 1980-11-19

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