NI201700038A - Compuestos de 1-alquil-6-oxo-1,6-dihidropiridin-3-ilo y usos de los mismos - Google Patents

Compuestos de 1-alquil-6-oxo-1,6-dihidropiridin-3-ilo y usos de los mismos

Info

Publication number
NI201700038A
NI201700038A NI201700038A NI201700038A NI201700038A NI 201700038 A NI201700038 A NI 201700038A NI 201700038 A NI201700038 A NI 201700038A NI 201700038 A NI201700038 A NI 201700038A NI 201700038 A NI201700038 A NI 201700038A
Authority
NI
Nicaragua
Prior art keywords
compounds
dihydropyridin
oxo
alkyl
ilo
Prior art date
Application number
NI201700038A
Other languages
English (en)
Inventor
Elisabeth Ripa Lena
Lawitz Karolina
Juhani Lepistö Matti
Hemmerling Martin
Edman Karl
Llinas Antonio
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54252264&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NI201700038(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NI201700038A publication Critical patent/NI201700038A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención se refiere en forma general a los compuestos de 1-alquil-6-oxo-1,6-dihidropiridin-3-ilo (incluyendo sales de los mismos). La presente invención asímismo se refiere a las composiciones farmacéuticas y a los kits que comprenden dichos compuestos, a los usos de dichos compuestos ( incluyendo métodos de tratamiento y preparación de medicamentos), y a los procesos para preparar dichos compuestos.
NI201700038A 2014-09-26 2017-03-24 Compuestos de 1-alquil-6-oxo-1,6-dihidropiridin-3-ilo y usos de los mismos NI201700038A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201462055822P 2014-09-26 2014-09-26

Publications (1)

Publication Number Publication Date
NI201700038A true NI201700038A (es) 2018-01-05

Family

ID=54252264

Family Applications (1)

Application Number Title Priority Date Filing Date
NI201700038A NI201700038A (es) 2014-09-26 2017-03-24 Compuestos de 1-alquil-6-oxo-1,6-dihidropiridin-3-ilo y usos de los mismos

Country Status (30)

Country Link
US (1) US10196374B2 (es)
EP (1) EP3197878B1 (es)
JP (1) JP6430000B2 (es)
KR (1) KR101866706B1 (es)
CN (1) CN107001320B (es)
AP (1) AP2017009819A0 (es)
AR (1) AR105549A1 (es)
AU (1) AU2015323817B2 (es)
BR (1) BR112017006085B1 (es)
CA (1) CA2962312C (es)
CL (1) CL2017000715A1 (es)
CO (1) CO2017003955A2 (es)
CR (1) CR20170106A (es)
DO (1) DOP2017000064A (es)
EA (1) EA031945B1 (es)
ES (1) ES2751640T3 (es)
GT (1) GT201700058A (es)
IL (1) IL250886A0 (es)
MX (1) MX2017003697A (es)
NI (1) NI201700038A (es)
NZ (1) NZ730250A (es)
PE (1) PE20171110A1 (es)
PH (1) PH12017500533A1 (es)
SG (1) SG11201702225VA (es)
SV (1) SV2017005412A (es)
TN (1) TN2017000096A1 (es)
TW (1) TW201619146A (es)
UY (1) UY36327A (es)
WO (1) WO2016046260A1 (es)
ZA (1) ZA201702720B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017161518A1 (en) * 2016-03-23 2017-09-28 Astrazeneca Ab New physical form
US10626106B2 (en) 2017-12-18 2020-04-21 Gruenenthal Gmbh Substituted pyrrolidine amides I
TW201927769A (zh) 2017-12-18 2019-07-16 德商歌林達有限公司 經取代之吡咯啶醯胺ii
EP3908581A1 (en) 2019-01-11 2021-11-17 Grünenthal GmbH Substituted pyrrolidine amides iii
EP3986886A2 (en) 2019-06-19 2022-04-27 Grünenthal GmbH Substituted pyrrolidine amides v
EP3986885B1 (en) 2019-06-19 2023-05-03 Grünenthal GmbH Substituted pyrrolidine amides iv
EP4086247A4 (en) * 2019-12-31 2023-12-06 Medshine Discovery Inc. BENZOPYRAZOLE COMPOUND
US20230265078A1 (en) 2020-07-09 2023-08-24 Gruenenthal Gmbh Substituted pyrrolidine amines and amides vi
CN115667237A (zh) * 2020-07-17 2023-01-31 成都苑东生物制药股份有限公司 作为bet抑制剂的新型杂环化合物
WO2023041695A1 (en) 2021-09-20 2023-03-23 Astrazeneca Ab Methods of treating inflammatory diseases with a selective glucocorticoid receptor modulator

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008506669A (ja) * 2004-07-16 2008-03-06 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 神経変性疾患の処置に適するピペリジン、ピペラジンもしくはモルホリンの二量体化合物またはそれらの7−員同族体
JO2754B1 (en) * 2006-12-21 2014-03-15 استرازينكا ايه بي Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders
US20100080786A1 (en) * 2008-05-20 2010-04-01 Markus Berger Phenyl or Pyridinyl Substituted Indazoles Derivatives

Also Published As

Publication number Publication date
EP3197878A1 (en) 2017-08-02
MX2017003697A (es) 2017-06-26
WO2016046260A8 (en) 2017-04-13
NZ730250A (en) 2018-03-23
JP2017529369A (ja) 2017-10-05
KR101866706B1 (ko) 2018-06-11
AU2015323817A1 (en) 2017-04-06
CA2962312A1 (en) 2016-03-31
DOP2017000064A (es) 2017-03-31
WO2016046260A1 (en) 2016-03-31
US10196374B2 (en) 2019-02-05
US20170298041A1 (en) 2017-10-19
AU2015323817B2 (en) 2018-11-01
CR20170106A (es) 2017-09-01
PE20171110A1 (es) 2017-08-07
CN107001320B (zh) 2019-09-20
CL2017000715A1 (es) 2017-11-10
CN107001320A (zh) 2017-08-01
GT201700058A (es) 2019-08-12
AR105549A1 (es) 2017-10-18
CO2017003955A2 (es) 2017-05-10
TN2017000096A1 (en) 2018-07-04
UY36327A (es) 2016-04-01
EA201790496A1 (ru) 2018-03-30
EA031945B1 (ru) 2019-03-29
JP6430000B2 (ja) 2018-11-28
ZA201702720B (en) 2019-06-26
EP3197878B1 (en) 2019-07-24
SG11201702225VA (en) 2017-04-27
BR112017006085B1 (pt) 2023-03-07
IL250886A0 (en) 2017-04-30
ES2751640T3 (es) 2020-04-01
TW201619146A (zh) 2016-06-01
SV2017005412A (es) 2017-10-23
PH12017500533A1 (en) 2017-08-07
CA2962312C (en) 2019-01-15
KR20170042785A (ko) 2017-04-19
BR112017006085A2 (pt) 2017-12-19
AP2017009819A0 (en) 2017-03-31

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