MY156536A - Inhibitors of protein tyrosine kinase activity - Google Patents

Inhibitors of protein tyrosine kinase activity

Info

Publication number
MY156536A
MY156536A MYPI2010000797A MYPI20100797A MY156536A MY 156536 A MY156536 A MY 156536A MY PI2010000797 A MYPI2010000797 A MY PI2010000797A MY PI20100797 A MYPI20100797 A MY PI20100797A MY 156536 A MY156536 A MY 156536A
Authority
MY
Malaysia
Prior art keywords
tyrosine kinase
kinase activity
protein tyrosine
receptor signalling
inhibitors
Prior art date
Application number
MYPI2010000797A
Other languages
English (en)
Inventor
Claridge Stephen William
Vaisburg Arkadii
Uno Tetsuyuki
Raeppel Stéphane
Isakovic Ljubomir
Mannion Michael
Saavedra Oscar Mario
Gaudette Frédéric
Zhan Lijie
Nancy Z Zhou
Raeppel Franck
Déziel Robert
Original Assignee
Methylgene Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Methylgene Inc filed Critical Methylgene Inc
Publication of MY156536A publication Critical patent/MY156536A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
MYPI2010000797A 2007-08-29 2008-08-28 Inhibitors of protein tyrosine kinase activity MY156536A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US96867307P 2007-08-29 2007-08-29

Publications (1)

Publication Number Publication Date
MY156536A true MY156536A (en) 2016-02-26

Family

ID=40386626

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI2010000797A MY156536A (en) 2007-08-29 2008-08-28 Inhibitors of protein tyrosine kinase activity

Country Status (19)

Country Link
US (3) US8404846B2 (enExample)
EP (1) EP2183254B1 (enExample)
JP (1) JP5656634B2 (enExample)
KR (1) KR101556269B1 (enExample)
CN (3) CN101932586A (enExample)
AR (1) AR068066A1 (enExample)
AU (1) AU2008293038B2 (enExample)
BR (1) BRPI0816064B8 (enExample)
CA (1) CA2697795C (enExample)
DK (1) DK2183254T3 (enExample)
ES (1) ES2635131T3 (enExample)
IL (1) IL204192A (enExample)
MX (1) MX2010002427A (enExample)
MY (1) MY156536A (enExample)
PL (1) PL2183254T3 (enExample)
RU (1) RU2495044C2 (enExample)
TW (1) TWI571468B (enExample)
WO (1) WO2009026717A1 (enExample)
ZA (1) ZA201001512B (enExample)

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WO2019018570A1 (en) 2017-07-19 2019-01-24 Ignyta, Inc. PHARMACEUTICAL COMPOSITIONS CONTAINING ENTRECTINIB
US10180422B1 (en) 2017-08-22 2019-01-15 Scripps Health Methods of treating a neuroendocrine tumor
WO2019077506A1 (en) 2017-10-17 2019-04-25 Ignyta, Inc. PHARMACEUTICAL COMPOSITIONS AND SOLID GALENIC FORMS
EP3762392B1 (en) 2018-03-08 2024-05-15 Wellmarker Bio Co., Ltd. Thienopyridine derivatives and pharmaceutical composition comprising same
CN112566935B (zh) 2018-05-23 2024-12-13 百济神州有限公司 抗ox40抗体和使用方法
CN109384799B (zh) * 2018-11-12 2020-07-14 深圳海王医药科技研究院有限公司 一种多靶点激酶抑制剂化合物的晶型a及制备方法和含有其的药物组合物
JP2022554042A (ja) 2019-09-06 2022-12-28 ウェルマーカー・バイオ・カンパニー・リミテッド バイオマーカー型治療用組成物
WO2021050580A1 (en) * 2019-09-10 2021-03-18 Mirati Therapeutics, Inc. Crystalline form of a multi-tyrosine kinase inhibitor, method of preparation, and use thereof
WO2021098769A1 (en) * 2019-11-21 2021-05-27 Beigene, Ltd. Treatment of cancer with anti-ox40 antibodies and multi-kinase inhibitors
EP4089095A4 (en) * 2020-01-07 2024-03-27 Medshine Discovery Inc. DEUTERATED THIENOPYRIDINE COMPOUND
EP4213844A4 (en) 2020-09-17 2024-11-20 Mirati Therapeutics, Inc. POLYTHERAPIES
TW202302597A (zh) * 2021-03-10 2023-01-16 美商米拉蒂醫療公司 多重酪胺酸激酶抑制劑之結晶鹽、其製備方法及用途
WO2022240802A1 (en) 2021-05-10 2022-11-17 Teva Pharmaceuticals International Gmbh Solid state forms of sitravatinib salts and processes for preparation thereof
TW202342426A (zh) * 2022-02-15 2023-11-01 大陸商百濟神州（蘇州）生物科技有限公司 N-[(6-溴吡啶-3-基)甲基]-2-甲氧基乙烷-1-胺鹽及其製備方法
CN118846073B (zh) * 2024-06-25 2026-01-30 深圳海王医药科技研究院有限公司 一种酪氨酸激酶抑制剂的新应用
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Also Published As

Publication number Publication date
EP2183254A1 (en) 2010-05-12
PL2183254T3 (pl) 2017-10-31
CA2697795A1 (en) 2009-03-05
JP2010536887A (ja) 2010-12-02
IL204192A (en) 2016-08-31
CN105777776A (zh) 2016-07-20
RU2010111729A (ru) 2011-10-10
CN101932586A (zh) 2010-12-29
MX2010002427A (es) 2010-03-30
CN109970759B (zh) 2026-08-04
US8389541B2 (en) 2013-03-05
AR068066A1 (es) 2009-11-04
BRPI0816064B1 (pt) 2020-01-28
BRPI0816064B8 (pt) 2021-05-25
US20130165477A1 (en) 2013-06-27
DK2183254T3 (en) 2017-09-11
KR20100075873A (ko) 2010-07-05
AU2008293038A1 (en) 2009-03-05
RU2495044C2 (ru) 2013-10-10
ZA201001512B (en) 2010-11-24
US8846927B2 (en) 2014-09-30
TW200914458A (en) 2009-04-01
ES2635131T3 (es) 2017-10-02
CN105777776B (zh) 2021-06-08
US20090264440A1 (en) 2009-10-22
US20120108628A1 (en) 2012-05-03
BRPI0816064A2 (pt) 2015-03-31
CA2697795C (en) 2016-08-16
WO2009026717A1 (en) 2009-03-05
EP2183254A4 (en) 2011-09-28
TWI571468B (zh) 2017-02-21
US8404846B2 (en) 2013-03-26
JP5656634B2 (ja) 2015-01-21
EP2183254B1 (en) 2017-06-21
AU2008293038B2 (en) 2013-08-29
KR101556269B1 (ko) 2015-09-30
CN109970759A (zh) 2019-07-05

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