MXPA04005503A - Derivados de n-aril-n??arilcicloalquilurea como antagonistas de la hormona concentradora de melanina para el tratamiento de la obesidad. - Google Patents

Derivados de n-aril-n??arilcicloalquilurea como antagonistas de la hormona concentradora de melanina para el tratamiento de la obesidad.

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Publication number
MXPA04005503A
MXPA04005503A MXPA04005503A MXPA04005503A MXPA04005503A MX PA04005503 A MXPA04005503 A MX PA04005503A MX PA04005503 A MXPA04005503 A MX PA04005503A MX PA04005503 A MXPA04005503 A MX PA04005503A MX PA04005503 A MXPA04005503 A MX PA04005503A
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Mexico
Prior art keywords
alkyl
compound
substituted
aryl
alkylene
Prior art date
Application number
MXPA04005503A
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English (en)
Spanish (es)
Inventor
Haiqun Tang
Original Assignee
Schering Corp
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Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of MXPA04005503A publication Critical patent/MXPA04005503A/es

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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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MXPA04005503A 2001-12-04 2002-12-03 Derivados de n-aril-n??arilcicloalquilurea como antagonistas de la hormona concentradora de melanina para el tratamiento de la obesidad. MXPA04005503A (es)

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US8394765B2 (en) 2004-11-01 2013-03-12 Amylin Pharmaceuticals Llc Methods of treating obesity with two different anti-obesity agents
AU2005305036B2 (en) * 2004-11-01 2011-03-10 Amylin Pharmaceuticals, Llc Treatment of obesity and related disorders
US20090264650A1 (en) * 2005-03-31 2009-10-22 Nobuo Cho Prophylactic/Therapeutic Agent for Diabetes
US7799943B2 (en) * 2005-06-24 2010-09-21 Rohm And Haas Company Method for promoting Michael addition reactions
RU2008107336A (ru) 2005-07-27 2009-09-10 Дов Фармасьютикал, Инк. (Us) Новые 1-арил-з-азабицикло{3.1.0.} гексаны: получение и применение для лечения психоневрологических расстройств
US20080045725A1 (en) 2006-04-28 2008-02-21 Murry Jerry A Process For The Synthesis of (+) And (-)-1-(3,4-Dichlorophenyl)-3-Azabicyclo[3.1.0]Hexane
US20080269348A1 (en) * 2006-11-07 2008-10-30 Phil Skolnick Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use
US8138377B2 (en) 2006-11-07 2012-03-20 Dov Pharmaceutical, Inc. Arylbicyclo[3.1.0]hexylamines and methods and compositions for their preparation and use
US8030495B2 (en) * 2007-05-23 2011-10-04 Coleman Paul J Cyclopropyl pyrrolidine orexin receptor antagonists
US9133159B2 (en) 2007-06-06 2015-09-15 Neurovance, Inc. 1-heteroaryl-3-azabicyclo[3.1.0]hexanes, methods for their preparation and their use as medicaments
EP2036578A1 (en) * 2007-09-13 2009-03-18 Bayer Schering Pharma Aktiengesellschaft Diagnostic agents for positron emission imaging using F-18 radio labeled amino-alcohols
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WO2018026890A1 (en) 2016-08-03 2018-02-08 Cymabay Therapeutics Oxymethylene aryl compounds for treating inflammatory gastrointestinal diseases or gastrointestinal conditions
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EP1453501A1 (en) 2004-09-08
AR037621A1 (es) 2004-11-17
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US7348328B2 (en) 2008-03-25
CA2468967A1 (en) 2003-06-12
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DE60228317D1 (de) 2008-09-25
JP4330996B2 (ja) 2009-09-16
JP2009235076A (ja) 2009-10-15
ATE404190T1 (de) 2008-08-15
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