MX9304676A - Liponucleosidos de seco-nucleosidos, procedimiento para su preparacion y composiciones con actividad antiviral que los contienen. - Google Patents
Liponucleosidos de seco-nucleosidos, procedimiento para su preparacion y composiciones con actividad antiviral que los contienen.Info
- Publication number
- MX9304676A MX9304676A MX9304676A MX9304676A MX9304676A MX 9304676 A MX9304676 A MX 9304676A MX 9304676 A MX9304676 A MX 9304676A MX 9304676 A MX9304676 A MX 9304676A MX 9304676 A MX9304676 A MX 9304676A
- Authority
- MX
- Mexico
- Prior art keywords
- carbon atoms
- amino group
- alkyl
- liponucleotides
- substituted
- Prior art date
Links
- 230000000840 anti-viral effect Effects 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title 1
- 239000002777 nucleoside Substances 0.000 title 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 10
- 125000003277 amino group Chemical group 0.000 abstract 4
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 3
- MYMOFIZGZYHOMD-UHFFFAOYSA-N Dioxygen Chemical compound O=O MYMOFIZGZYHOMD-UHFFFAOYSA-N 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 229920006395 saturated elastomer Polymers 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- 125000004434 sulfur atom Chemical group 0.000 abstract 2
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 150000007529 inorganic bases Chemical class 0.000 abstract 1
- 150000007522 mineralic acids Chemical class 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000000475 sulfinyl group Chemical group [*:2]S([*:1])=O 0.000 abstract 1
- 125000000472 sulfonyl group Chemical group *S(*)(=O)=O 0.000 abstract 1
- 125000004417 unsaturated alkyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
- C07F9/65616—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system having three or more than three double bonds between ring members or between ring members and non-ring members, e.g. purine or analogs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Virology (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biochemistry (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4226279A DE4226279A1 (de) | 1992-08-08 | 1992-08-08 | Liponucleotide von Seco-Nucleosiden, deren Herstellung sowie deren Verwendung als antivirale Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9304676A true MX9304676A (es) | 1994-03-31 |
Family
ID=6465143
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9304676A MX9304676A (es) | 1992-08-08 | 1993-08-03 | Liponucleosidos de seco-nucleosidos, procedimiento para su preparacion y composiciones con actividad antiviral que los contienen. |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP0654036B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP3479299B2 (cg-RX-API-DMAC7.html) |
| KR (1) | KR100243440B1 (cg-RX-API-DMAC7.html) |
| CN (1) | CN1040984C (cg-RX-API-DMAC7.html) |
| AT (1) | ATE152114T1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU672994B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2141030A1 (cg-RX-API-DMAC7.html) |
| DE (2) | DE4226279A1 (cg-RX-API-DMAC7.html) |
| DK (1) | DK0654036T3 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2104163T3 (cg-RX-API-DMAC7.html) |
| FI (1) | FI109699B (cg-RX-API-DMAC7.html) |
| GR (1) | GR3023960T3 (cg-RX-API-DMAC7.html) |
| HU (1) | HUT72605A (cg-RX-API-DMAC7.html) |
| IL (1) | IL106588A (cg-RX-API-DMAC7.html) |
| MX (1) | MX9304676A (cg-RX-API-DMAC7.html) |
| NO (1) | NO304986B1 (cg-RX-API-DMAC7.html) |
| NZ (1) | NZ254813A (cg-RX-API-DMAC7.html) |
| TW (1) | TW306924B (cg-RX-API-DMAC7.html) |
| WO (1) | WO1994003465A1 (cg-RX-API-DMAC7.html) |
| ZA (1) | ZA935718B (cg-RX-API-DMAC7.html) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5817638A (en) * | 1988-07-07 | 1998-10-06 | Nexstar Pharmaceuticals, Inc. | Antiviral liponucleosides: treatment of hepatitis B |
| US6599887B2 (en) | 1988-07-07 | 2003-07-29 | Chimerix, Inc. | Methods of treating viral infections using antiviral liponucleotides |
| US6252060B1 (en) | 1988-07-07 | 2001-06-26 | Nexstar Pharmaceuticals, Inc. | Antiviral liponucleosides: treatment of hepatitis B |
| DE4402492A1 (de) * | 1994-01-28 | 1995-08-03 | Boehringer Mannheim Gmbh | Verfahren zur Herstellung von unsymmetrischen Phosphorsäurediestern |
| US7517858B1 (en) | 1995-06-07 | 2009-04-14 | The Regents Of The University Of California | Prodrugs of pharmaceuticals with improved bioavailability |
| KR100389558B1 (ko) * | 2000-10-11 | 2003-06-27 | 주식회사 한스환경엔지니어링 | 유리섬유 강화플라스틱 성형품의 표면처리용 직물 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5223263A (en) * | 1988-07-07 | 1993-06-29 | Vical, Inc. | Liponucleotide-containing liposomes |
| DE4026265A1 (de) * | 1990-08-20 | 1992-02-27 | Boehringer Mannheim Gmbh | Neue phospholipid-derivate von nucleosiden, deren herstellung sowie deren verwendung als antivirale arzneimittel |
-
1992
- 1992-08-08 DE DE4226279A patent/DE4226279A1/de not_active Withdrawn
-
1993
- 1993-07-07 TW TW082105422A patent/TW306924B/zh active
- 1993-08-03 MX MX9304676A patent/MX9304676A/es not_active IP Right Cessation
- 1993-08-04 IL IL106588A patent/IL106588A/en not_active IP Right Cessation
- 1993-08-06 EP EP93917764A patent/EP0654036B1/de not_active Expired - Lifetime
- 1993-08-06 NZ NZ254813A patent/NZ254813A/en unknown
- 1993-08-06 DE DE59306286T patent/DE59306286D1/de not_active Expired - Fee Related
- 1993-08-06 DK DK93917764.8T patent/DK0654036T3/da active
- 1993-08-06 AT AT93917764T patent/ATE152114T1/de not_active IP Right Cessation
- 1993-08-06 ES ES93917764T patent/ES2104163T3/es not_active Expired - Lifetime
- 1993-08-06 HU HU9500374A patent/HUT72605A/hu unknown
- 1993-08-06 CA CA002141030A patent/CA2141030A1/en not_active Abandoned
- 1993-08-06 WO PCT/EP1993/002101 patent/WO1994003465A1/de not_active Ceased
- 1993-08-06 JP JP50502594A patent/JP3479299B2/ja not_active Expired - Fee Related
- 1993-08-06 AU AU47082/93A patent/AU672994B2/en not_active Ceased
- 1993-08-06 KR KR1019950700463A patent/KR100243440B1/ko not_active Expired - Fee Related
- 1993-08-06 ZA ZA935718A patent/ZA935718B/xx unknown
- 1993-08-07 CN CN93107987A patent/CN1040984C/zh not_active Expired - Fee Related
-
1995
- 1995-02-07 FI FI950533A patent/FI109699B/fi not_active IP Right Cessation
- 1995-02-07 NO NO950445A patent/NO304986B1/no not_active IP Right Cessation
-
1997
- 1997-06-30 GR GR970401610T patent/GR3023960T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI950533L (fi) | 1995-02-07 |
| EP0654036B1 (de) | 1997-04-23 |
| TW306924B (cg-RX-API-DMAC7.html) | 1997-06-01 |
| ATE152114T1 (de) | 1997-05-15 |
| DK0654036T3 (da) | 1997-11-03 |
| ZA935718B (en) | 1995-02-06 |
| GR3023960T3 (en) | 1997-09-30 |
| AU4708293A (en) | 1994-03-03 |
| ES2104163T3 (es) | 1997-10-01 |
| IL106588A0 (en) | 1993-12-08 |
| DE4226279A1 (de) | 1994-02-10 |
| NZ254813A (en) | 1996-05-28 |
| HUT72605A (en) | 1996-05-28 |
| JPH08500345A (ja) | 1996-01-16 |
| CN1085908A (zh) | 1994-04-27 |
| HU9500374D0 (en) | 1995-03-28 |
| CA2141030A1 (en) | 1994-02-09 |
| FI950533A0 (fi) | 1995-02-07 |
| JP3479299B2 (ja) | 2003-12-15 |
| CN1040984C (zh) | 1998-12-02 |
| NO304986B1 (no) | 1999-03-15 |
| KR950702998A (ko) | 1995-08-23 |
| NO950445D0 (no) | 1995-02-07 |
| NO950445L (no) | 1995-02-07 |
| IL106588A (en) | 1998-01-04 |
| AU672994B2 (en) | 1996-10-24 |
| WO1994003465A1 (de) | 1994-02-17 |
| KR100243440B1 (ko) | 2000-03-02 |
| EP0654036A1 (de) | 1995-05-24 |
| DE59306286D1 (de) | 1997-05-28 |
| FI109699B (fi) | 2002-09-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration | ||
| HC | Change of company name or juridical status |
Owner name: CRAYOLA LLC |
|
| PD | Change of proprietorship |
Owner name: HEIDELBERG PHARMA HOLDING GMBH |
|
| MM | Annulment or lapse due to non-payment of fees |