MX9203366A - Esteres del acido androstadien-17-carboxilico y composiciones farmaceuticas que los contienen. - Google Patents

Esteres del acido androstadien-17-carboxilico y composiciones farmaceuticas que los contienen.

Info

Publication number
MX9203366A
MX9203366A MX9203366A MX9203366A MX9203366A MX 9203366 A MX9203366 A MX 9203366A MX 9203366 A MX9203366 A MX 9203366A MX 9203366 A MX9203366 A MX 9203366A MX 9203366 A MX9203366 A MX 9203366A
Authority
MX
Mexico
Prior art keywords
androstadien
esters
carboxylic acid
pharmaceutical compositions
compositions containing
Prior art date
Application number
MX9203366A
Other languages
English (en)
Inventor
Jaroslav Kalvoda
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of MX9203366A publication Critical patent/MX9203366A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX9203366A 1976-02-24 1992-06-25 Esteres del acido androstadien-17-carboxilico y composiciones farmaceuticas que los contienen. MX9203366A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH225376A CH628355A5 (de) 1976-02-24 1976-02-24 Verfahren zur herstellung neuer androstadien-17beta-carbonsaeuren und ihrer ester und salze.

Publications (1)

Publication Number Publication Date
MX9203366A true MX9203366A (es) 1992-09-01

Family

ID=4229445

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9203366A MX9203366A (es) 1976-02-24 1992-06-25 Esteres del acido androstadien-17-carboxilico y composiciones farmaceuticas que los contienen.

Country Status (26)

Country Link
US (1) US4285937A (es)
JP (1) JPS52102264A (es)
AT (1) AT361141B (es)
AU (1) AU513559B2 (es)
BE (1) BE851725A (es)
CA (1) CA1084483A (es)
CH (4) CH628355A5 (es)
CY (1) CY1198A (es)
DD (1) DD145918A5 (es)
DE (1) DE2707336A1 (es)
DK (1) DK153493C (es)
ES (5) ES456134A1 (es)
FR (2) FR2342302A1 (es)
GB (1) GB1578243A (es)
HK (1) HK57483A (es)
HU (1) HU176762B (es)
IE (1) IE45023B1 (es)
IL (2) IL51519A (es)
KE (1) KE3300A (es)
MX (1) MX9203366A (es)
MY (1) MY8500017A (es)
NL (1) NL7701886A (es)
NZ (1) NZ183418A (es)
SE (1) SE436572B (es)
SG (1) SG37383G (es)
ZA (1) ZA771087B (es)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4188385A (en) * 1978-04-05 1980-02-12 Syntex (U.S.A.) Inc. Thioetianic acid derivatives
US4198403A (en) * 1978-04-05 1980-04-15 Syntex (U.S.A.) Inc. 17 Beta-thiocarboxylic acid esters of 4-halo-3-oxoandrost-4-enes
PT69411A (en) * 1978-04-05 1979-04-01 Syntex Inc 4-halo etianic acids and derivatives thereof
DE3024008C2 (de) * 1980-06-24 1982-04-15 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 17α-Hydroxy-etiocarbonsäuren
US4607028A (en) * 1983-08-18 1986-08-19 Ciba-Geigy Corporation Novel carboxylic acid esters
SE8306370D0 (sv) * 1983-11-18 1983-11-18 Draco Ab Novel androstane-17beta-carboxylic acid esters, a process and intermediates for their preparation, compositions and method for the treatment of inflammatory conditions
SE8501693D0 (sv) * 1985-04-04 1985-04-04 Draco Ab Novel 16,17-acetalsubstituted androstane-17beta-carboxylic acid esters
IL78144A0 (en) * 1985-04-04 1986-07-31 Draco Ab Novel androstane-17beta-carboxylic acid esters
WO1990015816A1 (en) * 1989-06-16 1990-12-27 The Upjohn Company Suramin type compounds and angiostatic steroids to inhibit angiogenesis
US6596260B1 (en) * 1993-08-27 2003-07-22 Novartis Corporation Aerosol container and a method for storage and administration of a predetermined amount of a pharmaceutically active aerosol
US5646136A (en) * 1994-01-04 1997-07-08 Duke University Methods of inhibiting angiogenesis and tumor growth, and treating ophthalmologic conditions with angiostatic and therapeutic steroids
US5981517A (en) * 1996-05-09 1999-11-09 Soft Drugs, Inc. Androstene derivatives
GB0015876D0 (en) * 2000-06-28 2000-08-23 Novartis Ag Organic compounds
US6858593B2 (en) * 2000-08-05 2005-02-22 Smithkline Beecham Corporation Anti-inflammatory androstane derivative compositions
US6777400B2 (en) * 2000-08-05 2004-08-17 Smithkline Beecham Corporation Anti-inflammatory androstane derivative compositions
US6858596B2 (en) * 2000-08-05 2005-02-22 Smithkline Beecham Corporation Formulation containing anti-inflammatory androstane derivative
US6759398B2 (en) * 2000-08-05 2004-07-06 Smithkline Beecham Corporation Anti-inflammatory androstane derivative
US6777399B2 (en) * 2000-08-05 2004-08-17 Smithkline Beecham Corporation Anti-inflammatory androstane derivative compositions
US6750210B2 (en) * 2000-08-05 2004-06-15 Smithkline Beecham Corporation Formulation containing novel anti-inflammatory androstane derivative
US6787532B2 (en) * 2000-08-05 2004-09-07 Smithkline Beecham Corporation Formulation containing anti-inflammatory androstane derivatives
EP1305329B2 (en) * 2000-08-05 2015-03-18 Glaxo Group Limited 6.alpha.,9.alpha.-difluoro-17.alpha.-(2-furanylcarboxyl)oxy-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent
GB0019172D0 (en) 2000-08-05 2000-09-27 Glaxo Group Ltd Novel compounds
UA77656C2 (en) * 2001-04-07 2007-01-15 Glaxo Group Ltd S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent
BR0209271A (pt) * 2001-04-30 2004-06-15 Glaxo Group Ltd Composto, uso de um composto composição farmacêutica, formulação em aerossol farmacêutica, método para o tratamento de um paciente humano ou animal com uma condição inflamatória e/ou alérgica, e, processo para a preparação de um composto
US20050175545A1 (en) * 2002-02-04 2005-08-11 Keith Biggadike Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist
GB0202635D0 (en) * 2002-02-05 2002-03-20 Glaxo Wellcome Mfg Pte Ltd Formulation containing novel anti-inflammatory androstane derivative
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
EP1653974B1 (en) * 2003-06-19 2010-01-06 BODOR, Nicholas S. Enhancement of activity and/or duration of action of soft anti-inflammatory steroids for topical or other local application
WO2004112800A1 (en) * 2003-06-19 2004-12-29 Bodor Nicholas S Enhancement of activity and/or duration of action of selected anti-inflammatory steroids
GB0507165D0 (en) * 2005-04-08 2005-05-18 Glaxo Group Ltd Novel crystalline pharmaceutical product
BRPI0617673C1 (pt) * 2005-10-19 2012-05-22 Ranbaxy Lab Ltd composições de inibidores de fosfodiesterase do tipo iv
US7691811B2 (en) * 2006-05-25 2010-04-06 Bodor Nicholas S Transporter-enhanced corticosteroid activity and methods and compositions for treating dry eye
US7687484B2 (en) * 2006-05-25 2010-03-30 Bodor Nicholas S Transporter enhanced corticosteroid activity
GB0615108D0 (en) * 2006-07-28 2006-09-06 Glaxo Group Ltd Novel formulations
US8227027B2 (en) 2007-12-07 2012-07-24 Presspart Gmbh & Co. Kg Method for applying a polymer coating to an internal surface of a container
EP2111861A1 (en) 2008-04-21 2009-10-28 Ranbaxy Laboratories Limited Compositions of phosphodiesterase type IV inhibitors
US8835410B2 (en) 2011-05-10 2014-09-16 Bodor Laboratories, Inc. Treatment of eyelid dermatitis
CN111100176A (zh) * 2019-12-20 2020-05-05 重庆华邦胜凯制药有限公司 一种化合物的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3636010A (en) * 1968-12-23 1972-01-18 Ciba Geigy Corp Esters of steroid-17-carboxylic acids
GB1384372A (en) * 1971-01-20 1975-02-19 Glaxo Lab Ltd Dereivatives of 17alpha-hydroxyandrost-4-ene-17beta-carboxylic acids
GB1438940A (en) * 1972-07-19 1976-06-09 Glaxo Lab Ltd 17beta-haloalkoxycarbonyl-17alpha-oxysteroids
US4093721A (en) * 1974-08-30 1978-06-06 Glaxo Laboratories Limited Pharmaceutical compositions of 6α,9α-difluoro-androst-4-ene-17β-carboxylates and derivatives thereof
GB1514476A (en) * 1974-08-30 1978-06-14 Glaxo Lab Ltd Alkyl and haloalkyl androst-4-ene and androsta-1,4-diene-17beta-carboxylates

Also Published As

Publication number Publication date
AU2257277A (en) 1978-08-31
ATA119477A (de) 1980-07-15
FR2369297A1 (fr) 1978-05-26
AT361141B (de) 1981-02-25
DK153493B (da) 1988-07-18
DD145918A5 (de) 1981-01-14
JPS6139959B2 (es) 1986-09-06
JPS52102264A (en) 1977-08-27
ES467433A1 (es) 1979-10-16
IL51519A0 (en) 1977-04-29
CH628641A5 (de) 1982-03-15
HK57483A (en) 1983-11-25
KE3300A (en) 1983-08-05
IE45023L (en) 1977-08-24
ES467434A1 (es) 1979-08-16
AU513559B2 (en) 1980-12-11
SE7701999L (sv) 1977-08-25
DK79077A (da) 1977-08-25
CA1084483A (en) 1980-08-26
SE436572B (sv) 1985-01-07
CH629824A5 (de) 1982-05-14
MY8500017A (en) 1985-12-31
DE2707336A1 (de) 1977-08-25
FR2342302A1 (fr) 1977-09-23
DK153493C (da) 1988-11-28
NZ183418A (en) 1980-02-21
ES456134A1 (es) 1978-05-01
ES467430A1 (es) 1979-08-16
CH628355A5 (de) 1982-02-26
US4285937A (en) 1981-08-25
NL7701886A (nl) 1977-08-26
SG37383G (en) 1984-02-17
GB1578243A (en) 1980-11-05
FR2369297B1 (es) 1981-03-06
CY1198A (en) 1983-12-31
ES467432A1 (es) 1979-08-16
HU176762B (en) 1981-05-28
IL51519A (en) 1983-03-31
CH628356A5 (de) 1982-02-26
IE45023B1 (en) 1982-06-02
DE2707336C2 (es) 1988-09-01
IL61512A0 (en) 1980-12-31
FR2342302B1 (es) 1981-01-09
ZA771087B (en) 1978-01-25
BE851725A (fr) 1977-08-23

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