MX338831B - Moduladores selectivos de receptores de androgenos. - Google Patents

Moduladores selectivos de receptores de androgenos.

Info

Publication number
MX338831B
MX338831B MX2012008995A MX2012008995A MX338831B MX 338831 B MX338831 B MX 338831B MX 2012008995 A MX2012008995 A MX 2012008995A MX 2012008995 A MX2012008995 A MX 2012008995A MX 338831 B MX338831 B MX 338831B
Authority
MX
Mexico
Prior art keywords
androgen receptor
iia
iii
formula
receptor modulators
Prior art date
Application number
MX2012008995A
Other languages
English (en)
Spanish (es)
Other versions
MX2012008995A (es
Inventor
Chris P Miller
Original Assignee
Radius Health Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Radius Health Inc filed Critical Radius Health Inc
Publication of MX2012008995A publication Critical patent/MX2012008995A/es
Publication of MX338831B publication Critical patent/MX338831B/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
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    • G—PHYSICS
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    • G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
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    • G—PHYSICS
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    • G01N2333/705—Assays involving receptors, cell surface antigens or cell surface determinants
    • G01N2333/72—Assays involving receptors, cell surface antigens or cell surface determinants for hormones
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    • G01N2500/10—Screening for compounds of potential therapeutic value involving cells

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  • Health & Medical Sciences (AREA)
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  • Medicinal Chemistry (AREA)
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  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
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  • Endocrinology (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
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  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
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MX2012008995A 2010-02-04 2011-02-04 Moduladores selectivos de receptores de androgenos. MX338831B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30149210P 2010-02-04 2010-02-04
PCT/US2011/023768 WO2011097496A1 (en) 2010-02-04 2011-02-04 Selective androgen receptor modulators

Publications (2)

Publication Number Publication Date
MX2012008995A MX2012008995A (es) 2012-11-22
MX338831B true MX338831B (es) 2016-05-03

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Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012008995A MX338831B (es) 2010-02-04 2011-02-04 Moduladores selectivos de receptores de androgenos.

Country Status (8)

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US (3) US8987319B2 (enExample)
EP (1) EP2531029B1 (enExample)
JP (2) JP5964756B2 (enExample)
AU (1) AU2011212813B2 (enExample)
BR (1) BR112012019551A2 (enExample)
CA (1) CA2788907A1 (enExample)
MX (1) MX338831B (enExample)
WO (1) WO2011097496A1 (enExample)

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US9951324B2 (en) 2010-02-25 2018-04-24 Purdue Research Foundation PSMA binding ligand-linker conjugates and methods for using
DK2568806T3 (en) 2010-05-12 2016-08-15 Radius Health Inc therapy Programs
WO2012047617A1 (en) 2010-09-28 2012-04-12 Radius Health, Inc. Selective androgen receptor modulators
CN103172643B (zh) * 2011-12-26 2016-03-02 中国医学科学院药物研究所 黄皮咔唑生物碱及其制备方法和其药物组合物与用途
EP3858341A1 (en) 2012-11-15 2021-08-04 Endocyte, Inc. Psma ligand-containing conjugates for the treatment of prostate cancer
KR101947053B1 (ko) 2013-10-18 2019-02-12 도이체스 크렙스포르슝스첸트룸 전립선 특이적 막 항원（ｐｓｍａ）의 표지된 억제제, 조영제로서의 이의 용도 및 전립선암 치료용 약제
EP3533473A3 (en) 2013-11-14 2019-12-18 Endocyte, Inc. Compounds for positron emission tomography
US9682960B2 (en) 2013-12-19 2017-06-20 Endorecherche, Inc. Non-steroidal antiandrogens and selective androgen receptor modulators with a pyridyl moiety
US9421264B2 (en) 2014-03-28 2016-08-23 Duke University Method of treating cancer using selective estrogen receptor modulators
PL3122426T3 (pl) 2014-03-28 2023-05-15 Duke University Leczenie raka sutka z zastosowaniem selektywnych modulatorów receptora estrogenowego
US10188759B2 (en) 2015-01-07 2019-01-29 Endocyte, Inc. Conjugates for imaging
JP6757037B2 (ja) * 2016-02-15 2020-09-16 学校法人近畿大学 ストレス評価方法
HRP20220619T1 (hr) 2016-06-22 2023-02-03 Ellipses Pharma Ltd Postupci za liječenje ar+ raka dojke
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