MX2019012757A - Composicion farmaceutica para administracion oral que comprende enzalutamida. - Google Patents
Composicion farmaceutica para administracion oral que comprende enzalutamida.Info
- Publication number
- MX2019012757A MX2019012757A MX2019012757A MX2019012757A MX2019012757A MX 2019012757 A MX2019012757 A MX 2019012757A MX 2019012757 A MX2019012757 A MX 2019012757A MX 2019012757 A MX2019012757 A MX 2019012757A MX 2019012757 A MX2019012757 A MX 2019012757A
- Authority
- MX
- Mexico
- Prior art keywords
- enzalutamide
- pharmaceutical composition
- orally administrable
- containing pharmaceutical
- administrable pharmaceutical
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
Se proporciona una composición farmacéutica para administración oral en donde se mejoran las propiedades de solubilidad y/o disolución de enzalutamida y se mantiene la sobresaturación. También se proporciona una composición farmacéutica para administración oral en donde se mejora la capacidad de absorción oral de enzalutamida. La composición farmacéutica para administración oral comprende enzalutamida y alcohol polivinílico.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2017090300 | 2017-04-28 | ||
PCT/JP2018/017159 WO2018199282A1 (ja) | 2017-04-28 | 2018-04-27 | エンザルタミドを含有する経口投与用医薬組成物 |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2019012757A true MX2019012757A (es) | 2019-12-16 |
Family
ID=63920425
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2019012757A MX2019012757A (es) | 2017-04-28 | 2018-04-27 | Composicion farmaceutica para administracion oral que comprende enzalutamida. |
Country Status (10)
Country | Link |
---|---|
US (1) | US20200146977A1 (es) |
EP (1) | EP3616696A4 (es) |
JP (1) | JP7172997B2 (es) |
KR (1) | KR20190137920A (es) |
CN (1) | CN110573153B (es) |
AU (1) | AU2018256998B2 (es) |
CA (1) | CA3060366A1 (es) |
MX (1) | MX2019012757A (es) |
RU (1) | RU2019138248A (es) |
WO (1) | WO2018199282A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA201991484A1 (ru) | 2012-09-11 | 2019-11-29 | Лекарственные формы энзалутамида | |
JP7238509B2 (ja) * | 2019-03-19 | 2023-03-14 | 三菱ケミカル株式会社 | 医薬錠剤 |
WO2021240206A1 (en) * | 2020-05-24 | 2021-12-02 | Lotus International Pte. Ltd. | Enzalutamide formulation |
JP7414668B2 (ja) | 2020-08-28 | 2024-01-16 | 信越化学工業株式会社 | ポリビニルアルコール含有造粒物及び固形製剤 |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP4072597B2 (ja) * | 1994-12-27 | 2008-04-09 | ナムローゼ・フェンノートシャップ・オルガノン | 持続性製剤 |
JPH10316576A (ja) * | 1997-05-13 | 1998-12-02 | Nissui Pharm Co Ltd | キトサン含有錠剤 |
ME01992B (me) | 2005-05-13 | 2012-10-30 | Univ California | Jedinjenje diarilhidantoina |
WO2010029930A1 (ja) * | 2008-09-12 | 2010-03-18 | 第一三共ヘルスケア株式会社 | 変色が抑制された安定な医薬製剤 |
MX2012009782A (es) | 2010-02-24 | 2012-11-29 | Medivation Prostate Therapeutics Inc | Procesos para la sintesis de diariltiohidantoina y compuestos de diarilhidantoina. |
MX357551B (es) * | 2011-03-23 | 2018-07-13 | Ironshore Pharmaceuticals & Dev Inc | Metodos y composiciones para el tratamiento de trastorno por deficit de atencion. |
EP2674149B1 (en) * | 2012-06-15 | 2017-10-04 | Shin-Etsu Chemical Co., Ltd. | Method of preparing composite granule comprising low-substituted hydroxypropyl cellulose and rapid release preparation |
JP2015534550A (ja) | 2012-09-11 | 2015-12-03 | ドクター レディズ ラボラトリーズ リミテッド | エンザルタミドの多形形態およびその調製 |
EA201991484A1 (ru) * | 2012-09-11 | 2019-11-29 | Лекарственные формы энзалутамида | |
WO2014167428A2 (en) * | 2013-04-10 | 2014-10-16 | Shilpa Medicare Limited | Amorphous 4-(3-(4-cyano-3-(trifluoromethyl)phenyl)-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl)-2-fluoro-n-methylbenzamide |
JP6133445B2 (ja) * | 2014-01-30 | 2017-05-24 | テイカ製薬株式会社 | 口腔内速崩壊性固形製剤用組成物 |
CN112402360A (zh) * | 2014-02-05 | 2021-02-26 | 斯洛文尼亚莱柯制药股份有限公司 | 雄激素受体拮抗剂的固体药物组合物 |
WO2015120014A1 (en) * | 2014-02-05 | 2015-08-13 | Merck Sharp & Dohme Corp. | Novel disintegration systems for pharmaceutical dosage forms |
SG11201607623XA (en) * | 2014-04-25 | 2016-11-29 | Chugai Pharmaceutical Co Ltd | Preparation containing tetracyclic compound at high dose |
US20180280302A1 (en) * | 2015-01-20 | 2018-10-04 | Merck Patent Gmbh | Solid dispersions of compounds using polyvinyl alcohol as a carrier polymer |
JP6403615B2 (ja) * | 2015-03-18 | 2018-10-10 | 日本酢ビ・ポバール株式会社 | フィルムコーティング組成物並びに経口固形製剤及びその製造方法 |
JP2016056208A (ja) * | 2016-01-15 | 2016-04-21 | 日本酢ビ・ポバール株式会社 | フィルムコーティング組成物並びに経口固形製剤及びその製造方法 |
-
2018
- 2018-04-27 WO PCT/JP2018/017159 patent/WO2018199282A1/ja unknown
- 2018-04-27 CA CA3060366A patent/CA3060366A1/en active Pending
- 2018-04-27 US US16/609,062 patent/US20200146977A1/en active Pending
- 2018-04-27 MX MX2019012757A patent/MX2019012757A/es unknown
- 2018-04-27 EP EP18791486.6A patent/EP3616696A4/en active Pending
- 2018-04-27 CN CN201880028051.1A patent/CN110573153B/zh active Active
- 2018-04-27 JP JP2019514651A patent/JP7172997B2/ja active Active
- 2018-04-27 RU RU2019138248A patent/RU2019138248A/ru unknown
- 2018-04-27 AU AU2018256998A patent/AU2018256998B2/en active Active
- 2018-04-27 KR KR1020197034702A patent/KR20190137920A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JPWO2018199282A1 (ja) | 2020-03-12 |
RU2019138248A3 (es) | 2021-07-21 |
US20200146977A1 (en) | 2020-05-14 |
CN110573153B (zh) | 2023-04-04 |
JP7172997B2 (ja) | 2022-11-16 |
EP3616696A4 (en) | 2021-01-27 |
WO2018199282A1 (ja) | 2018-11-01 |
KR20190137920A (ko) | 2019-12-11 |
CN110573153A (zh) | 2019-12-13 |
RU2019138248A (ru) | 2021-05-28 |
CA3060366A1 (en) | 2018-11-01 |
AU2018256998A1 (en) | 2019-12-05 |
EP3616696A1 (en) | 2020-03-04 |
AU2018256998B2 (en) | 2023-11-09 |
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