MX2016005482A - Formas de dosificacion granuladas disuasivas del abuso de liberacion inmediata. - Google Patents

Formas de dosificacion granuladas disuasivas del abuso de liberacion inmediata.

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Publication number
MX2016005482A
MX2016005482A MX2016005482A MX2016005482A MX2016005482A MX 2016005482 A MX2016005482 A MX 2016005482A MX 2016005482 A MX2016005482 A MX 2016005482A MX 2016005482 A MX2016005482 A MX 2016005482A MX 2016005482 A MX2016005482 A MX 2016005482A
Authority
MX
Mexico
Prior art keywords
dosage forms
immediate release
disposable
abuse
release abuse
Prior art date
Application number
MX2016005482A
Other languages
English (en)
Other versions
MX384376B (es
Inventor
K Haswani Dinesh
V Moe Derek
a o'neill Victoria
A Vega Zepeda Manuel
Original Assignee
Cima Labs Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51263565&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2016005482(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cima Labs Inc filed Critical Cima Labs Inc
Priority claimed from PCT/US2014/062887 external-priority patent/WO2015066172A1/en
Publication of MX2016005482A publication Critical patent/MX2016005482A/es
Publication of MX384376B publication Critical patent/MX384376B/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
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    • A61K31/60—Salicylic acid; Derivatives thereof
    • A61K31/612—Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid
    • A61K31/616—Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid by carboxylic acids, e.g. acetylsalicylic acid
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
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  • Health & Medical Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Pain & Pain Management (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
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  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se describen formas de dosificación orales de liberación inmediata que contienen características disuasivas del abuso. En particular, las formas de dosificación descritas proporcionan disuasión de abuso por ingestión de múltiples dosis individuales. Además, las formas de dosificación descritas proporcionan protección de sobredosis en el caso de ingestión accidental o intencional de dosis individuales múltiples.
MX2016005482A 2013-10-31 2014-10-29 Formas de dosificación de liberación inmediata disuasivas del abuso, en forma de partículas recubiertas con capas múltiples que comprenden un analgésico narcótico susceptible de abuso o sobredosis. MX384376B (es)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201361898207P 2013-10-31 2013-10-31
PCT/US2014/047014 WO2015065547A1 (en) 2013-10-31 2014-07-17 Immediate release abuse-deterrent granulated dosage forms
US14/333,986 US20150118300A1 (en) 2013-10-31 2014-07-17 Immediate Release Abuse-Deterrent Granulated Dosage Forms
US14/477,354 US20150118301A1 (en) 2013-10-31 2014-09-04 Immediate Release Abuse-Deterrent Granulated Dosage Forms
PCT/US2014/054061 WO2015065586A1 (en) 2013-10-31 2014-09-04 Immediate release abuse-deterrent granulated dosage forms
US14/484,793 US20150118295A1 (en) 2013-10-31 2014-09-12 Immediate Release Abuse-Deterrent Granulated Dosage Forms
PCT/US2014/062887 WO2015066172A1 (en) 2013-10-31 2014-10-29 Immediate release abuse-deterrent granulated dosage forms

Publications (2)

Publication Number Publication Date
MX2016005482A true MX2016005482A (es) 2016-12-16
MX384376B MX384376B (es) 2025-03-14

Family

ID=51263565

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016005482A MX384376B (es) 2013-10-31 2014-10-29 Formas de dosificación de liberación inmediata disuasivas del abuso, en forma de partículas recubiertas con capas múltiples que comprenden un analgésico narcótico susceptible de abuso o sobredosis.

Country Status (11)

Country Link
US (9) US20150118300A1 (es)
JP (1) JP6659925B2 (es)
KR (1) KR102363573B1 (es)
CN (1) CN105682647A (es)
AU (1) AU2014342412B2 (es)
CL (1) CL2016001031A1 (es)
HK (1) HK1223856A1 (es)
MX (1) MX384376B (es)
PE (1) PE20160606A1 (es)
WO (2) WO2015065547A1 (es)
ZA (1) ZA201604451B (es)

Families Citing this family (51)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7776314B2 (en) 2002-06-17 2010-08-17 Grunenthal Gmbh Abuse-proofed dosage system
DE102005005446A1 (de) 2005-02-04 2006-08-10 Grünenthal GmbH Bruchfeste Darreichungsformen mit retardierter Freisetzung
DE10336400A1 (de) 2003-08-06 2005-03-24 Grünenthal GmbH Gegen Missbrauch gesicherte Darreichungsform
US20070048228A1 (en) 2003-08-06 2007-03-01 Elisabeth Arkenau-Maric Abuse-proofed dosage form
DE10361596A1 (de) 2003-12-24 2005-09-29 Grünenthal GmbH Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform
DE102004032049A1 (de) 2004-07-01 2006-01-19 Grünenthal GmbH Gegen Missbrauch gesicherte, orale Darreichungsform
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