MX2015005174A - Agente profilactico y/o terapeutico para sintomas conductuales y psicologicos asociados con la enfermedad neurodegenerativa o sintomas impulsivos asociados con enfermedad mental que contiene brexpiprazol o sales del mismo. - Google Patents

Agente profilactico y/o terapeutico para sintomas conductuales y psicologicos asociados con la enfermedad neurodegenerativa o sintomas impulsivos asociados con enfermedad mental que contiene brexpiprazol o sales del mismo.

Info

Publication number
MX2015005174A
MX2015005174A MX2015005174A MX2015005174A MX2015005174A MX 2015005174 A MX2015005174 A MX 2015005174A MX 2015005174 A MX2015005174 A MX 2015005174A MX 2015005174 A MX2015005174 A MX 2015005174A MX 2015005174 A MX2015005174 A MX 2015005174A
Authority
MX
Mexico
Prior art keywords
symptoms associated
behavioral
prophylactic
salt
therapeutic agent
Prior art date
Application number
MX2015005174A
Other languages
English (en)
Other versions
MX371279B (es
Inventor
Kenji Maeda
Mai Nakamura
Shinji Sato
Dai Ishikawa
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of MX2015005174A publication Critical patent/MX2015005174A/es
Publication of MX371279B publication Critical patent/MX371279B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Abstract

La presente invención se refiere a un agente profiláctico y/o terapéutico para los síntomas conductuales y psicológicos asociados con enfermedad neurodegenerativa o síntomas impulsivos asociados con enfermedad mental, que contiene 7-[4-(4--benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1H-quinolin-2 -ona o una de sus sales como un ingrediente activo.
MX2015005174A 2012-10-25 2013-10-24 Agente profiláctico y/o terapéutico para síntomas conductuales y psicológicos asociados con la enfermedad neurodegenerativa o síntomas impulsivos asociados con enfermedad mental que contiene brexpiprazol o sales del mismo. MX371279B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261718305P 2012-10-25 2012-10-25
US201361782467P 2013-03-14 2013-03-14
PCT/JP2013/079480 WO2014065437A1 (en) 2012-10-25 2013-10-24 Prophylactic and/or therapeutic agent for behavioral and psychological symptoms associated with neurodegenerative disease or impulsive symptoms associated with mental disease containing brexpiprazole or salt thereof

Publications (2)

Publication Number Publication Date
MX2015005174A true MX2015005174A (es) 2015-09-04
MX371279B MX371279B (es) 2020-01-24

Family

ID=49585556

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015005174A MX371279B (es) 2012-10-25 2013-10-24 Agente profiláctico y/o terapéutico para síntomas conductuales y psicológicos asociados con la enfermedad neurodegenerativa o síntomas impulsivos asociados con enfermedad mental que contiene brexpiprazol o sales del mismo.

Country Status (22)

Country Link
US (4) US20150272946A1 (es)
EP (2) EP3848033A1 (es)
JP (5) JP6329140B2 (es)
KR (1) KR102245016B1 (es)
CN (4) CN112402421A (es)
AR (1) AR093247A1 (es)
AU (1) AU2013335613B2 (es)
BR (1) BR112015008759A2 (es)
CA (1) CA2889196C (es)
EA (1) EA201590808A1 (es)
HK (1) HK1212609A1 (es)
IL (1) IL238402B (es)
JO (2) JOP20210047A1 (es)
MX (1) MX371279B (es)
MY (1) MY180185A (es)
NZ (1) NZ708321A (es)
PH (1) PH12015500925A1 (es)
SG (2) SG10201702828TA (es)
TW (1) TWI643620B (es)
UA (1) UA116549C2 (es)
WO (1) WO2014065437A1 (es)
ZA (1) ZA201503640B (es)

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TWI415845B (zh) 2006-10-03 2013-11-21 Arena Pharm Inc 用於治療與5-ht2a血清素受體相關聯病症之作為5-ht2a血清素受體之調節劑的吡唑衍生物
WO2009023253A2 (en) 2007-08-15 2009-02-19 Arena Pharmaceuticals Inc. IMIDAZO[L,2-α]PYRIDINE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO
US20110021538A1 (en) 2008-04-02 2011-01-27 Arena Pharmaceuticals, Inc. Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor
CN102264354B (zh) 2008-10-28 2015-03-25 艾尼纳制药公司 用于治疗5-ht2a5-羟色胺受体相关障碍的5-ht2a5-羟色胺受体调节剂组合物
US9126946B2 (en) 2008-10-28 2015-09-08 Arena Pharmaceuticals, Inc. Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto
MX2016013889A (es) 2014-04-22 2017-03-09 Otsuka Pharma Co Ltd Medicamento.
EP3244897A4 (en) * 2015-01-12 2018-08-22 Reviva Pharmaceuticals, Inc. Methods for treating alzheimer's disease
JP2018502158A (ja) * 2015-01-12 2018-01-25 レビバ ファーマシューティカルズ,インコーポレイティド パーキンソン病と関連する精神病の治療方法
JP2018516992A (ja) 2015-06-12 2018-06-28 アクソファント サイエンシーズ ゲーエムベーハーAxovant Sciences Gmbh レム睡眠行動障害の予防および処置のために有用なジアリールおよびアリールヘテロアリール尿素誘導体
BR112018000728A2 (pt) * 2015-07-15 2018-09-04 Axovant Sciences Gmbh resumo método para a profilaxia e/ou tratamento de alucinações visuais em um sujeito com necessidade do mesmo
CN105175401A (zh) * 2015-10-16 2015-12-23 北京康立生医药技术开发有限公司 一种依匹哌唑的制备方法
CN105541819B (zh) * 2016-02-04 2018-09-14 浙江永宁药业股份有限公司 一种依匹唑派的制备方法及其中间体和中间体的制备方法
BR112019010466A2 (pt) 2016-12-20 2019-09-10 Lts Lohmann Therapie Systeme Ag sistema terapêutico transdérmico contendo asenapina
KR102614709B1 (ko) 2016-12-20 2023-12-18 에르테에스 로만 테라피-시스테메 아게 아세나핀 및 폴리실록산 또는 폴리이소부틸렌을 함유하는 경피흡수 치료 시스템
ES2881783T3 (es) 2017-06-26 2021-11-30 Lts Lohmann Therapie Systeme Ag Sistema terapéutico transdérmico que contiene asenapina y polímero de acrílico y silicona
EP3720434A4 (en) 2017-12-05 2021-09-01 Sunovion Pharmaceuticals Inc. NON-RACEMIC MIXTURES AND THEIR USE
MX2020005517A (es) 2017-12-05 2020-11-09 Sunovion Pharmaceuticals Inc Formas cristalinas y metodos de produccion de las mismas.
EP3501506B1 (en) 2017-12-19 2019-10-09 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical tablet composition comprising brexpiprazole
KR20210022656A (ko) 2018-06-20 2021-03-03 에르테에스 로만 테라피-시스테메 아게 아세나핀을 함유하는 경피 치료 시스템
CN114401717A (zh) 2019-06-04 2022-04-26 赛诺维信制药公司 修饰释放配制品及其用途
WO2021029020A1 (ja) * 2019-08-13 2021-02-18 大塚製薬株式会社 経口医薬組成物
EP4173620A1 (en) * 2020-06-24 2023-05-03 National University Corporation Hokkaido University Blood-cerebrospinal fluid barrier protecting agent
CN112137994B (zh) * 2020-09-15 2022-10-14 中山大学 小分子化合物在制备抗丝状病毒药物中的应用
US11229644B1 (en) * 2020-12-31 2022-01-25 Lake O'hara Llc Methods of treating psychiatric disorders in obese patients with brexpiprazole

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JP4315393B2 (ja) * 2005-04-14 2009-08-19 大塚製薬株式会社 複素環化合物
TWI320783B (en) * 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
JP4540700B2 (ja) * 2006-10-13 2010-09-08 大塚製薬株式会社 医薬
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TWI636784B (zh) * 2011-04-05 2018-10-01 大塚製藥股份有限公司 含7-〔4-(4-苯並〔b〕噻吩-4-基-哌-1-基)丁氧基〕-1H-喹啉-2-酮之醫藥組成物與套組,以及彼之用途
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Also Published As

Publication number Publication date
NZ708321A (en) 2019-03-29
CN114712360A (zh) 2022-07-08
WO2014065437A1 (en) 2014-05-01
KR102245016B1 (ko) 2021-04-26
JP2021181448A (ja) 2021-11-25
JOP20210047A1 (ar) 2017-06-16
EP2911670A1 (en) 2015-09-02
CA2889196C (en) 2021-02-16
JP2015535211A (ja) 2015-12-10
KR20150074156A (ko) 2015-07-01
EA201590808A1 (ru) 2015-08-31
JOP20130313B1 (ar) 2021-08-17
SG11201503152TA (en) 2015-05-28
TW201427665A (zh) 2014-07-16
HK1212609A1 (zh) 2016-06-17
CN108578408A (zh) 2018-09-28
US20190314367A1 (en) 2019-10-17
BR112015008759A2 (pt) 2017-07-04
MX371279B (es) 2020-01-24
JP2023123441A (ja) 2023-09-05
AU2013335613B2 (en) 2018-07-12
IL238402A0 (en) 2015-06-30
JP2020045345A (ja) 2020-03-26
AU2013335613A1 (en) 2015-06-04
US20150272946A1 (en) 2015-10-01
CN104755082A (zh) 2015-07-01
CA2889196A1 (en) 2014-05-01
UA116549C2 (uk) 2018-04-10
JP6329140B2 (ja) 2018-05-23
SG10201702828TA (en) 2017-05-30
EP3848033A1 (en) 2021-07-14
US20170258787A1 (en) 2017-09-14
MY180185A (en) 2020-11-24
CN112402421A (zh) 2021-02-26
PH12015500925B1 (en) 2015-06-29
JP2018138555A (ja) 2018-09-06
TWI643620B (zh) 2018-12-11
US20220370442A1 (en) 2022-11-24
ZA201503640B (en) 2016-08-31
PH12015500925A1 (en) 2015-06-29
AR093247A1 (es) 2015-05-27
IL238402B (en) 2018-11-29

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