MX2009009540A - Inhibidores de metaloproteasa que contienen una porcion heterociclica. - Google Patents

Inhibidores de metaloproteasa que contienen una porcion heterociclica.

Info

Publication number
MX2009009540A
MX2009009540A MX2009009540A MX2009009540A MX2009009540A MX 2009009540 A MX2009009540 A MX 2009009540A MX 2009009540 A MX2009009540 A MX 2009009540A MX 2009009540 A MX2009009540 A MX 2009009540A MX 2009009540 A MX2009009540 A MX 2009009540A
Authority
MX
Mexico
Prior art keywords
mmp
heterocyclic moiety
metalloprotease inhibitors
inhibitors containing
heterocyclic
Prior art date
Application number
MX2009009540A
Other languages
English (en)
Inventor
Christian Gege
Carine Chevrier
Arthur Taveras
Brian M Gallagher Jr
Original Assignee
Alantos Pharm Holding
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alantos Pharm Holding filed Critical Alantos Pharm Holding
Publication of MX2009009540A publication Critical patent/MX2009009540A/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
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Abstract

La presente invención se refiere generalmente a compuestos que inhiben la metaloproteasa heterocíclicos de la fórmula (I). (ver fórmula (I)) Más particularmente, la presente invención proporciona una clase nueva de compuestos que inhiben MMP 3, MMP 8 y/o MMP 13 heterocíclicos con una porción de benzoxazinona o esquearamida, que exhiben una potencia y selectividad incrementada en relación a los inhibidores MMP 13, MMP 8 y MMP 3 actualmente conocidos.
MX2009009540A 2007-03-07 2008-03-07 Inhibidores de metaloproteasa que contienen una porcion heterociclica. MX2009009540A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US90556507P 2007-03-07 2007-03-07
PCT/US2008/003196 WO2008109181A2 (en) 2007-03-07 2008-03-07 Metalloprotease inhibitors containing a heterocyclic moiety

Publications (1)

Publication Number Publication Date
MX2009009540A true MX2009009540A (es) 2009-09-16

Family

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Application Number Title Priority Date Filing Date
MX2009009541A MX2009009541A (es) 2007-03-07 2008-03-07 Inhibidores de metaloproteasa que contienen una porcion heterociclica.
MX2009009552A MX2009009552A (es) 2007-03-07 2008-03-07 Inhibidores de metaloproteasa que contienen una porcion heterociclica.
MX2009009540A MX2009009540A (es) 2007-03-07 2008-03-07 Inhibidores de metaloproteasa que contienen una porcion heterociclica.

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MX2009009541A MX2009009541A (es) 2007-03-07 2008-03-07 Inhibidores de metaloproteasa que contienen una porcion heterociclica.
MX2009009552A MX2009009552A (es) 2007-03-07 2008-03-07 Inhibidores de metaloproteasa que contienen una porcion heterociclica.

Country Status (7)

Country Link
US (5) US20080221093A1 (es)
EP (3) EP2125816A2 (es)
JP (3) JP2010520293A (es)
AU (3) AU2008223348A1 (es)
CA (3) CA2680173A1 (es)
MX (3) MX2009009541A (es)
WO (5) WO2008109178A1 (es)

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