MX2009007670A - 1,3-dioxanos sustituidos utiles como moduladores de paar. - Google Patents

1,3-dioxanos sustituidos utiles como moduladores de paar.

Info

Publication number
MX2009007670A
MX2009007670A MX2009007670A MX2009007670A MX2009007670A MX 2009007670 A MX2009007670 A MX 2009007670A MX 2009007670 A MX2009007670 A MX 2009007670A MX 2009007670 A MX2009007670 A MX 2009007670A MX 2009007670 A MX2009007670 A MX 2009007670A
Authority
MX
Mexico
Prior art keywords
compound according
ppar
linear
alkyl
branched
Prior art date
Application number
MX2009007670A
Other languages
English (en)
Spanish (es)
Inventor
Jean-Philippe Meyer
Alexandra Santana Sorensen
Peteris Alberts
Melya Hughes Crameri
Mainkar S Prathama
Original Assignee
Evolva Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/IB2007/002542 external-priority patent/WO2007138485A2/en
Application filed by Evolva Sa filed Critical Evolva Sa
Priority claimed from PCT/US2008/051521 external-priority patent/WO2008089461A1/en
Publication of MX2009007670A publication Critical patent/MX2009007670A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/041,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/061,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
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    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A61K31/36Compounds containing methylenedioxyphenyl groups, e.g. sesamin
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
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    • C07D319/041,3-Dioxanes; Hydrogenated 1,3-dioxanes
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    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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MX2009007670A 2007-01-18 2008-01-18 1,3-dioxanos sustituidos utiles como moduladores de paar. MX2009007670A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
PCT/IB2007/002542 WO2007138485A2 (en) 2006-01-18 2007-01-18 Ppar modulators
US98980507P 2007-11-21 2007-11-21
US98980607P 2007-11-21 2007-11-21
US98980807P 2007-11-21 2007-11-21
PCT/US2008/051521 WO2008089461A1 (en) 2007-01-18 2008-01-18 Substituted 1,3-dioxanes useful as ppar modulators

Publications (1)

Publication Number Publication Date
MX2009007670A true MX2009007670A (es) 2011-11-18

Family

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Family Applications (4)

Application Number Title Priority Date Filing Date
MX2009007670A MX2009007670A (es) 2007-01-18 2008-01-18 1,3-dioxanos sustituidos utiles como moduladores de paar.
MX2009007667A MX2009007667A (es) 2007-01-18 2008-01-18 Profarmacos de 1,3-dioxanos sustituidos y sus usos.
MX2009007669A MX2009007669A (es) 2007-01-18 2008-01-18 1,3,-dioxanos sustituidos y sus usos.
MX2009007668A MX2009007668A (es) 2007-01-18 2008-01-18 1,3-dioxanos sustituidos y sus usos.

Family Applications After (3)

Application Number Title Priority Date Filing Date
MX2009007667A MX2009007667A (es) 2007-01-18 2008-01-18 Profarmacos de 1,3-dioxanos sustituidos y sus usos.
MX2009007669A MX2009007669A (es) 2007-01-18 2008-01-18 1,3,-dioxanos sustituidos y sus usos.
MX2009007668A MX2009007668A (es) 2007-01-18 2008-01-18 1,3-dioxanos sustituidos y sus usos.

Country Status (8)

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US (5) US8536196B2 (enExample)
EP (1) EP2120567A4 (enExample)
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