MX2008016519A - Compuestos de pirro[1,2,-b]piridazinona. - Google Patents

Compuestos de pirro[1,2,-b]piridazinona.

Info

Publication number
MX2008016519A
MX2008016519A MX2008016519A MX2008016519A MX2008016519A MX 2008016519 A MX2008016519 A MX 2008016519A MX 2008016519 A MX2008016519 A MX 2008016519A MX 2008016519 A MX2008016519 A MX 2008016519A MX 2008016519 A MX2008016519 A MX 2008016519A
Authority
MX
Mexico
Prior art keywords
alkylene
mmol
alkyl
heterocyclyl
aryl
Prior art date
Application number
MX2008016519A
Other languages
English (en)
Spanish (es)
Inventor
Stephen E Webber
Peter S Dragovich
David John Kucera
Liansheng Li
Frank Ruebsam
Martin T Tran
Douglas E Murphy
Zhongxiang Sun
Chinh Viet Tran
Original Assignee
Anadys Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anadys Pharmaceuticals Inc filed Critical Anadys Pharmaceuticals Inc
Publication of MX2008016519A publication Critical patent/MX2008016519A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2008016519A 2006-06-22 2007-06-21 Compuestos de pirro[1,2,-b]piridazinona. MX2008016519A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81557806P 2006-06-22 2006-06-22
PCT/US2007/071826 WO2007150001A1 (en) 2006-06-22 2007-06-21 Pyrro[1,2-b]pyridazinone compounds

Publications (1)

Publication Number Publication Date
MX2008016519A true MX2008016519A (es) 2009-01-30

Family

ID=38833773

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2008016519A MX2008016519A (es) 2006-06-22 2007-06-21 Compuestos de pirro[1,2,-b]piridazinona.

Country Status (14)

Country Link
US (3) US7462611B2 (de)
EP (1) EP2038286B1 (de)
JP (2) JP5306194B2 (de)
KR (1) KR101384266B1 (de)
CN (2) CN101501039B (de)
AR (1) AR061581A1 (de)
BR (1) BRPI0713684A2 (de)
CA (1) CA2656000C (de)
IL (1) IL196106A0 (de)
MX (1) MX2008016519A (de)
NZ (1) NZ573875A (de)
PA (1) PA8733401A1 (de)
TW (1) TWI395749B (de)
WO (1) WO2007150001A1 (de)

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CA2589527A1 (en) 2004-12-17 2006-06-22 Anadys Pharmaceuticals, Inc. Pyridazinone compounds
EP2038286B1 (de) * 2006-06-22 2017-03-08 Anadys Pharmaceuticals, Inc. Pyrro[1,2-b]pyridazinon-verbindungen
UA100120C2 (en) * 2007-04-03 2012-11-26 Анадис Фармасьютикалз, Инк. 5,6-dihydro-1h-pyridin-2-one compounds
ATE548044T1 (de) 2007-05-04 2012-03-15 Vertex Pharma Kombinationstherapie zur behandlung von hiv- infektionen
AU2009222105B2 (en) * 2008-03-03 2012-05-17 Novartis Ag Compounds and compositions as TLR activity modulators
US20090257979A1 (en) * 2008-04-15 2009-10-15 Intermune, Inc. Novel Inhibitors of Hepatitis C Virus Replication
TWI480272B (zh) 2008-10-09 2015-04-11 Anadys Pharmaceuticals Inc 藉由５，６－二氫－１ｈ－吡啶－２－酮與一或多種其他抗病毒化合物的組合物抑制ｃ型肝炎病毒的方法
WO2011056647A1 (en) * 2009-10-28 2011-05-12 Anadys Pharmaceuticals, Inc. Deuterated 5,6-dihydro-1h-pyridin-2-one compounds
NZ598465A (en) 2009-10-30 2013-10-25 Boehringer Ingelheim Int Dosage regimens for hcv combination therapy comprising bi201335, interferon alpha and ribavirin
TW201121968A (en) * 2009-11-09 2011-07-01 Intermune Inc Novel inhibitors of hepatitis C virus replication
WO2011072370A1 (en) * 2009-12-18 2011-06-23 Boehringer Ingelheim International Gmbh Hcv combination therapy
US20120321590A1 (en) 2011-04-06 2012-12-20 Anadys Pharmaceuticals, Inc. Bridged polycyclic compounds
MY183704A (en) 2011-06-07 2021-03-09 Anadys Pharmaceuticals Inc [1,2,4]thiadiazine 1,1-dioxide compounds for lowering serum uric acid
KR102017867B1 (ko) 2011-06-23 2019-09-03 다이나믹 마이크로시스템즈 세미컨덕터 이큅먼트 게엠베하 반도체 클리너 시스템들 및 방법들
CN102796105B (zh) * 2012-08-15 2014-08-06 苏州施亚生物科技有限公司 2,5,6,7-四氢吡咯并[3,4-c]哒嗪-3-酮及其衍生物以及它们的合成方法
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CN103553986B (zh) * 2013-11-19 2015-04-22 郑州西格玛化工有限公司 一种制备3,4-二氨基苯磺酰胺的方法
WO2021030278A1 (en) * 2019-08-12 2021-02-18 Aligos Therapeutics, Inc. Bicyclic compounds

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Also Published As

Publication number Publication date
CN102584649A (zh) 2012-07-18
NZ573875A (en) 2011-11-25
BRPI0713684A2 (pt) 2012-10-30
JP2013136599A (ja) 2013-07-11
CN101501039B (zh) 2012-02-22
PA8733401A1 (es) 2008-11-19
KR20090063203A (ko) 2009-06-17
US20090312570A1 (en) 2009-12-17
TWI395749B (zh) 2013-05-11
JP2009544575A (ja) 2009-12-17
IL196106A0 (en) 2009-09-01
JP5670487B2 (ja) 2015-02-18
EP2038286B1 (de) 2017-03-08
EP2038286A4 (de) 2010-05-12
CN101501039A (zh) 2009-08-05
WO2007150001A1 (en) 2007-12-27
US20080031852A1 (en) 2008-02-07
TW200817405A (en) 2008-04-16
US20090105473A1 (en) 2009-04-23
KR101384266B1 (ko) 2014-04-24
US7582754B2 (en) 2009-09-01
AR061581A1 (es) 2008-09-03
US7462611B2 (en) 2008-12-09
JP5306194B2 (ja) 2013-10-02
EP2038286A1 (de) 2009-03-25
WO2007150001A8 (en) 2008-02-28
CA2656000C (en) 2016-09-06
AU2007260827A1 (en) 2007-12-27
US7842838B2 (en) 2010-11-30
CA2656000A1 (en) 2007-12-27

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