MX2007007188A - Derivados de tetrahidroquinolina sustituidos en 4 con cicloalquilo y su uso como medicamentos. - Google Patents
Derivados de tetrahidroquinolina sustituidos en 4 con cicloalquilo y su uso como medicamentos.Info
- Publication number
- MX2007007188A MX2007007188A MX2007007188A MX2007007188A MX2007007188A MX 2007007188 A MX2007007188 A MX 2007007188A MX 2007007188 A MX2007007188 A MX 2007007188A MX 2007007188 A MX2007007188 A MX 2007007188A MX 2007007188 A MX2007007188 A MX 2007007188A
- Authority
- MX
- Mexico
- Prior art keywords
- compound
- formula
- inhibitors
- salts
- solvates
- Prior art date
Links
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Classifications
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- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
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Landscapes
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- Obesity (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004060997A DE102004060997A1 (de) | 2004-12-18 | 2004-12-18 | Chemische Verbindung und ihre Verwendung |
| DE102004061000A DE102004061000A1 (de) | 2004-12-18 | 2004-12-18 | Chemische Verbindung und ihre Verwendung |
| PCT/EP2005/013490 WO2006063828A1 (de) | 2004-12-18 | 2005-12-15 | 4-cycloalkyl-substituierte tetrahydrochinolinderivate und deren verwendung als medikamente |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007007188A true MX2007007188A (es) | 2007-08-14 |
Family
ID=35841894
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007007188A MX2007007188A (es) | 2004-12-18 | 2005-12-15 | Derivados de tetrahidroquinolina sustituidos en 4 con cicloalquilo y su uso como medicamentos. |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US8124775B2 (https=) |
| EP (1) | EP1828137B1 (https=) |
| JP (1) | JP5132317B2 (https=) |
| KR (1) | KR20070090248A (https=) |
| AR (1) | AR055011A1 (https=) |
| AT (1) | ATE555097T1 (https=) |
| AU (1) | AU2005315770B2 (https=) |
| BR (1) | BRPI0519602A2 (https=) |
| CA (1) | CA2591397A1 (https=) |
| CU (1) | CU23452B7 (https=) |
| CY (1) | CY1112887T1 (https=) |
| DK (1) | DK1828137T3 (https=) |
| DO (1) | DOP2005000259A (https=) |
| ES (1) | ES2384980T3 (https=) |
| GT (1) | GT200500377A (https=) |
| IL (1) | IL184008A (https=) |
| MA (1) | MA29100B1 (https=) |
| MX (1) | MX2007007188A (https=) |
| NO (1) | NO20073146L (https=) |
| PE (1) | PE20060767A1 (https=) |
| PL (1) | PL1828137T3 (https=) |
| PT (1) | PT1828137E (https=) |
| RU (1) | RU2393151C2 (https=) |
| SI (1) | SI1828137T1 (https=) |
| TW (1) | TW200635900A (https=) |
| UY (1) | UY29276A1 (https=) |
| WO (1) | WO2006063828A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0519566A2 (pt) * | 2004-12-18 | 2009-01-27 | Bayer Healthcare Ag | derivados de (5s)-3-[(s)-fléor(4-trifluormetilfenil)metil]-5,6,7,8-tet raidroquinolin-5-ol e seu uso como inibidores de cetp |
| DE102006012548A1 (de) * | 2006-03-18 | 2007-09-20 | Bayer Healthcare Ag | Substituierte Chromanol-Derivate und ihre Verwendung |
| BRPI0909105A2 (pt) * | 2008-03-05 | 2015-08-25 | Boehringer Ingelheim Int | Derivados de piridina tricíclicos, composição farmacêutica e uso dos mesmos, bem como processos para preparar os ditos compostos e a dita composição farmacêutica |
| UY33229A (es) * | 2010-02-19 | 2011-09-30 | Boehringer Ingelheim Int | Derivados de piridina tricíclicos, medicamentos que contienen tales compuestos, su uso y proceso pa ra su preparación |
| CA2804924C (en) * | 2010-07-09 | 2016-06-28 | Daiichi Sankyo Company, Limited | Substituted pyridine compound |
| EP2675811A1 (en) | 2011-02-17 | 2013-12-25 | Boehringer Ingelheim International GmbH | Tricyclic pyridine derivatives, medicaments containing such compounds, their use and process for their preparation |
| EP2760868B1 (en) | 2011-08-17 | 2018-04-25 | Boehringer Ingelheim International GmbH | Furo[3,4-c]quinoline derivatives, medicaments containing such compounds, their use and process for their preparation |
| TWI570118B (zh) | 2012-01-06 | 2017-02-11 | 第一三共股份有限公司 | 經取代之吡啶化合物的酸加成鹽 |
| MX384679B (es) | 2014-07-30 | 2025-03-14 | Hoffmann La Roche | Marcadores genéticos para predecir la reactividad a terapia con agente que eleva la lipoproteína de alta densidad (hdl) o que imita la lipoproteína de alta densidad (hdl). |
| WO2025185022A1 (zh) * | 2024-03-05 | 2025-09-12 | 维康平生(北京)生物科技有限公司 | 一种脂肪体的制备方法 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4128681A1 (de) * | 1991-08-29 | 1993-03-04 | Bayer Ag | Substituierte mandelsaeurederivate, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln |
| DE19610932A1 (de) | 1996-03-20 | 1997-09-25 | Bayer Ag | 2-Aryl-substituierte Pyridine |
| HRP970330B1 (en) * | 1996-07-08 | 2004-06-30 | Bayer Ag | Cycloalkano pyridines |
| DE19627431A1 (de) | 1996-07-08 | 1998-01-15 | Bayer Ag | Heterocyclisch kondensierte Pyridine |
| DE19627430A1 (de) | 1996-07-08 | 1998-01-15 | Bayer Ag | Bicyclisch kondensierte Pyridine |
| US6207671B1 (en) | 1996-07-08 | 2001-03-27 | Bayer Aktiengesellschaft | Cycloalkano-pyridines |
| DE19704244A1 (de) | 1997-02-05 | 1998-08-06 | Bayer Ag | 5-Hydroxy-alkyl substituierte Phenyle |
| DE19709125A1 (de) | 1997-03-06 | 1998-09-10 | Bayer Ag | Substituierte Chinoline |
| MA24643A1 (fr) * | 1997-09-18 | 1999-04-01 | Bayer Ag | Tetrahydro-naphtalenes substitues et composes analogues |
| DE19741051A1 (de) | 1997-09-18 | 1999-03-25 | Bayer Ag | Hetero-Tetrahydrochinoline |
| DE19741399A1 (de) | 1997-09-19 | 1999-03-25 | Bayer Ag | Tetrahydrochinoline |
| DE19935966A1 (de) | 1999-07-30 | 2001-02-01 | Bayer Ag | Verfahren zur Reduktion von Ketoalkoholen |
| DE10148436A1 (de) | 2001-10-01 | 2003-04-17 | Bayer Ag | Tetrahydrochinoline |
| DE10250687A1 (de) | 2002-10-31 | 2004-05-13 | Bayer Ag | 7H-Dibenzo(b,g)(1,5)dioxocin-5-on-Derivate und ihre Verwendung |
| BRPI0519566A2 (pt) * | 2004-12-18 | 2009-01-27 | Bayer Healthcare Ag | derivados de (5s)-3-[(s)-fléor(4-trifluormetilfenil)metil]-5,6,7,8-tet raidroquinolin-5-ol e seu uso como inibidores de cetp |
-
2005
- 2005-12-15 ES ES05820528T patent/ES2384980T3/es not_active Expired - Lifetime
- 2005-12-15 PL PL05820528T patent/PL1828137T3/pl unknown
- 2005-12-15 EP EP05820528A patent/EP1828137B1/de not_active Expired - Lifetime
- 2005-12-15 WO PCT/EP2005/013490 patent/WO2006063828A1/de not_active Ceased
- 2005-12-15 SI SI200531547T patent/SI1828137T1/sl unknown
- 2005-12-15 CA CA002591397A patent/CA2591397A1/en not_active Abandoned
- 2005-12-15 AT AT05820528T patent/ATE555097T1/de active
- 2005-12-15 DK DK05820528.7T patent/DK1828137T3/da active
- 2005-12-15 AU AU2005315770A patent/AU2005315770B2/en not_active Ceased
- 2005-12-15 MX MX2007007188A patent/MX2007007188A/es active IP Right Grant
- 2005-12-15 RU RU2007127127/04A patent/RU2393151C2/ru not_active IP Right Cessation
- 2005-12-15 PT PT05820528T patent/PT1828137E/pt unknown
- 2005-12-15 JP JP2007545948A patent/JP5132317B2/ja not_active Expired - Fee Related
- 2005-12-15 BR BRPI0519602-7A patent/BRPI0519602A2/pt not_active IP Right Cessation
- 2005-12-15 KR KR1020077016219A patent/KR20070090248A/ko not_active Ceased
- 2005-12-15 US US11/793,482 patent/US8124775B2/en not_active Expired - Fee Related
- 2005-12-16 PE PE2005001475A patent/PE20060767A1/es not_active Application Discontinuation
- 2005-12-16 DO DO2005P000259A patent/DOP2005000259A/es unknown
- 2005-12-16 AR ARP050105313A patent/AR055011A1/es not_active Application Discontinuation
- 2005-12-16 TW TW094144588A patent/TW200635900A/zh unknown
- 2005-12-19 GT GT200500377A patent/GT200500377A/es unknown
- 2005-12-20 UY UY29276A patent/UY29276A1/es not_active Application Discontinuation
-
2007
- 2007-06-18 CU CU20070140A patent/CU23452B7/es not_active IP Right Cessation
- 2007-06-18 MA MA30003A patent/MA29100B1/fr unknown
- 2007-06-18 IL IL184008A patent/IL184008A/en not_active IP Right Cessation
- 2007-06-19 NO NO20073146A patent/NO20073146L/no not_active Application Discontinuation
-
2012
- 2012-02-16 US US13/398,290 patent/US20120142728A1/en not_active Abandoned
- 2012-06-29 CY CY20121100588T patent/CY1112887T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20080255068A1 (en) | 2008-10-16 |
| US20120142728A1 (en) | 2012-06-07 |
| AU2005315770B2 (en) | 2011-12-08 |
| US8124775B2 (en) | 2012-02-28 |
| DOP2005000259A (es) | 2006-11-15 |
| IL184008A0 (en) | 2007-10-31 |
| PE20060767A1 (es) | 2006-09-10 |
| CA2591397A1 (en) | 2006-06-22 |
| RU2007127127A (ru) | 2009-01-27 |
| SI1828137T1 (sl) | 2012-08-31 |
| JP5132317B2 (ja) | 2013-01-30 |
| NO20073146L (no) | 2007-09-18 |
| AU2005315770A1 (en) | 2006-06-22 |
| IL184008A (en) | 2012-03-29 |
| ATE555097T1 (de) | 2012-05-15 |
| MA29100B1 (fr) | 2007-12-03 |
| EP1828137A1 (de) | 2007-09-05 |
| KR20070090248A (ko) | 2007-09-05 |
| TW200635900A (en) | 2006-10-16 |
| UY29276A1 (es) | 2006-07-31 |
| PL1828137T3 (pl) | 2012-09-28 |
| DK1828137T3 (da) | 2012-07-23 |
| RU2393151C2 (ru) | 2010-06-27 |
| ES2384980T3 (es) | 2012-07-16 |
| GT200500377A (es) | 2006-11-09 |
| CY1112887T1 (el) | 2016-04-13 |
| EP1828137B1 (de) | 2012-04-25 |
| JP2008524145A (ja) | 2008-07-10 |
| BRPI0519602A2 (pt) | 2009-02-25 |
| CU23452B7 (es) | 2009-12-01 |
| PT1828137E (pt) | 2012-07-04 |
| WO2006063828A1 (de) | 2006-06-22 |
| AR055011A1 (es) | 2007-08-01 |
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