MD1743B2 - Derivaţi ai indolului, procedeu de obţinere a lor, compoziţie fungicidă şi procedeu de combatere a fungilor - Google Patents
Derivaţi ai indolului, procedeu de obţinere a lor, compoziţie fungicidă şi procedeu de combatere a fungilorInfo
- Publication number
- MD1743B2 MD1743B2 MD96-0305A MD960305A MD1743B2 MD 1743 B2 MD1743 B2 MD 1743B2 MD 960305 A MD960305 A MD 960305A MD 1743 B2 MD1743 B2 MD 1743B2
- Authority
- MD
- Moldova
- Prior art keywords
- group
- preparation
- fungicidal composition
- indole derivatives
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
- A01N43/38—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings condensed with carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Invenţia se referă la derivaţi ai indolului, procedeu de obţinere a lor, compoziţie fungicidă şi procedeu de combatere a fungilor în focar.Derivatul indolului este prezentat prin formula generală (I),( I )în care R reprezintă o grupă fenil substituită;R3 şi R4, independent, reprezintă atomul de hidrogen sau halogen sau o grupă: alchil, alcoxi, cicloalchil, fenil sau fenoxi, opţional substituită;R5 şi R6, independent, reprezintă atomul de hidrogen sau o grupă: alchil, alcoxi, cicloalchil, fenil sau fenoxi, opţional substituită, sau R5 şi R6 împreună cu atomul de azot intermediar reprezintă grupa eterociclil;R7 reprezintă atomul de hidrogen sau grupa alchil.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP92109525 | 1992-06-05 | ||
PCT/EP1993/001406 WO1993025524A1 (en) | 1992-06-05 | 1993-06-03 | Fungicidal indole derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
MD1743B2 true MD1743B2 (ro) | 2001-09-30 |
Family
ID=8209683
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MD96-0305A MD1743B2 (ro) | 1992-06-05 | 1993-06-03 | Derivaţi ai indolului, procedeu de obţinere a lor, compoziţie fungicidă şi procedeu de combatere a fungilor |
Country Status (17)
Country | Link |
---|---|
US (1) | US5399559A (ro) |
EP (1) | EP0643695B1 (ro) |
JP (1) | JP3296490B2 (ro) |
CN (1) | CN1082318A (ro) |
AT (1) | ATE141260T1 (ro) |
AU (1) | AU666558B2 (ro) |
DE (1) | DE69304057T2 (ro) |
DK (1) | DK0643695T3 (ro) |
ES (1) | ES2091615T3 (ro) |
GE (1) | GEP19981431B (ro) |
GR (1) | GR3020807T3 (ro) |
HU (1) | HU216814B (ro) |
IL (1) | IL105909A (ro) |
MD (1) | MD1743B2 (ro) |
TW (1) | TW229140B (ro) |
WO (1) | WO1993025524A1 (ro) |
ZA (1) | ZA933846B (ro) |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100231956B1 (ko) * | 1995-08-04 | 1999-12-01 | 오쯔까 유우지로 | 인돌-2-카복실산 에스테르 유도체 및 활성 성분으로서 이를 함유하는 농업용 및 원예용 살균제 |
US6353007B1 (en) * | 2000-07-13 | 2002-03-05 | Boehringer Ingelheim Pharmaceuticals, Inc. | Substituted 1-(4-aminophenyl)indoles and their use as anti-inflammatory agents |
EP1314733A1 (en) * | 2001-11-22 | 2003-05-28 | Aventis Pharma Deutschland GmbH | Indole-2-carboxamides as factor Xa inhibitors |
EP1479677A1 (en) | 2003-05-19 | 2004-11-24 | Aventis Pharma Deutschland GmbH | New indole derivatives as factor xa inhibitors |
SE0302035D0 (sv) * | 2003-07-09 | 2003-07-09 | Biolipox Ab | New compound |
CA2570365A1 (en) * | 2004-06-18 | 2005-12-29 | Biolipox Ab | Indoles useful in the treatment of inflammation |
DE602005009209D1 (de) | 2004-06-18 | 2008-10-02 | Biolipox Ab | Zur behandlung von entzündungen geeignete indole |
CA2570531A1 (en) * | 2004-06-18 | 2005-12-29 | Kristofer Olofsson | Indoles useful in the treatment of inflammation |
ATE501119T1 (de) * | 2005-01-19 | 2011-03-15 | Biolipox Ab | Entzündungshemmende indol-derivate |
EP1844051A1 (en) * | 2005-01-19 | 2007-10-17 | Biolipox AB | Thienopyrroles useful in the treatment of inflammation |
WO2006077364A1 (en) * | 2005-01-19 | 2006-07-27 | Biolipox Ab | Indoles useful in the treatment of inflammation |
US20100197687A1 (en) * | 2005-01-19 | 2010-08-05 | Benjamin Pelcman | Indoles Useful in the Treatment of Inflammation |
WO2006077401A1 (en) * | 2005-01-19 | 2006-07-27 | Biolipox Ab | Pyrrolopyridines useful in the treatment of inflammation |
US20090042949A1 (en) * | 2005-01-19 | 2009-02-12 | Benjamin Pelcman | Indoles Useful in the Treatment of Inflammation |
AR056690A1 (es) | 2005-10-14 | 2007-10-17 | Athersys Inc | Derivados de indol como inhibidores de indol como inhibidores del receptor 3 de histamina para el tartamiento de trastornos del sueno y cognitivos obesidad y otros trastornos de snc |
WO2007109178A2 (en) * | 2006-03-16 | 2007-09-27 | Pharmacyclics, Inc. | Indole derivatives as inhibitors of histone deacetylase |
EA020332B1 (ru) * | 2007-08-10 | 2014-10-30 | Х. Лундбекк А/С | Аналоги гетероариламидов |
ME01838B (me) | 2009-06-29 | 2014-12-20 | Lncyte Holdings Corp | Pirimidinoni kao inhibitori pi3k |
US8759359B2 (en) | 2009-12-18 | 2014-06-24 | Incyte Corporation | Substituted heteroaryl fused derivatives as PI3K inhibitors |
EP2558463A1 (en) | 2010-04-14 | 2013-02-20 | Incyte Corporation | Fused derivatives as i3 inhibitors |
US9062055B2 (en) | 2010-06-21 | 2015-06-23 | Incyte Corporation | Fused pyrrole derivatives as PI3K inhibitors |
EP2655374B1 (en) | 2010-12-20 | 2019-10-23 | Incyte Holdings Corporation | N-(1-(substituted-phenyl)ethyl)-9h-purin-6-amines as pi3k inhibitors |
US9108984B2 (en) | 2011-03-14 | 2015-08-18 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors |
WO2012135009A1 (en) | 2011-03-25 | 2012-10-04 | Incyte Corporation | Pyrimidine-4,6-diamine derivatives as pi3k inhibitors |
KR102371532B1 (ko) | 2011-09-02 | 2022-03-07 | 인사이트 홀딩스 코포레이션 | Pi3k 억제제로서 헤테로시클릴아민 |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
NZ734993A (en) | 2015-02-27 | 2024-03-22 | Incyte Holdings Corp | Salts of pi3k inhibitor and processes for their preparation |
US9732097B2 (en) | 2015-05-11 | 2017-08-15 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
WO2024026290A1 (en) * | 2022-07-25 | 2024-02-01 | Cayman Chemical Company Incorporated | NOVEL HETEROCYCLES AS sPLA2-X INHIBITORS |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2008692A1 (de) * | 1969-02-26 | 1970-09-17 | Agence Nationale de Valorisation de La Recherche (ANVAR), Puteaux, Hautsde-Seine (Prankreich) | Verfahren zur Herstellung von Indol-3carbonsäurederivaten und nach dem Verfahren erhältliche, neue Verbindungen |
DE1966206A1 (de) * | 1968-04-26 | 1972-01-20 | Sumitomo Chemical Co | 1,4-Benzodiazepine und Arzneipraeparate |
JPH0570357A (ja) * | 1991-09-12 | 1993-03-23 | Fuso Yakuhin Kogyo Kk | 血液透析用顆粒剤 |
JPH0570358A (ja) * | 1991-09-10 | 1993-03-23 | Kao Corp | 象牙質知覚過敏治療剤 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3634402A (en) * | 1968-04-26 | 1972-01-11 | Sumitomo Chemical Co | Process for producing 1 4-benzodiazepine derivatives and their salts |
DE1935671C3 (de) * | 1968-04-26 | 1975-01-09 | Sumitomo Chemical Co | 2-Aminomethylindole und ihre Salze |
US3582285A (en) * | 1970-03-19 | 1971-06-01 | Xerox Corp | Chemical package |
US4431307A (en) * | 1981-11-19 | 1984-02-14 | Labsystems Oy | Set of cuvettes |
US4599315A (en) * | 1983-09-13 | 1986-07-08 | University Of California Regents | Microdroplet test apparatus |
EP0211698B1 (fr) * | 1985-02-08 | 1991-01-30 | Synthelabo | Dérivés de (dihydro-4,5 1H-imidazolyl-2)-2 dihydro-2,3 indole, leur préparation et leur application en thérapeutique |
US4925629A (en) * | 1988-07-28 | 1990-05-15 | Bioquant, Inc. | Diagnostic device |
US5147529A (en) * | 1988-08-10 | 1992-09-15 | E. I. Du Pont De Nemours And Company | Method for automatically processing magnetic solid phase reagents |
US5041266A (en) * | 1989-12-21 | 1991-08-20 | Hoffmann-La Roche Inc. | Tray for immunometric determinations |
-
1993
- 1993-05-24 TW TW082104079A patent/TW229140B/zh active
- 1993-06-02 ZA ZA933846A patent/ZA933846B/xx unknown
- 1993-06-03 DK DK93912878.1T patent/DK0643695T3/da active
- 1993-06-03 ES ES93912878T patent/ES2091615T3/es not_active Expired - Lifetime
- 1993-06-03 US US08/071,894 patent/US5399559A/en not_active Expired - Lifetime
- 1993-06-03 HU HU9403475A patent/HU216814B/hu not_active IP Right Cessation
- 1993-06-03 EP EP93912878A patent/EP0643695B1/en not_active Expired - Lifetime
- 1993-06-03 AT AT93912878T patent/ATE141260T1/de not_active IP Right Cessation
- 1993-06-03 DE DE69304057T patent/DE69304057T2/de not_active Expired - Fee Related
- 1993-06-03 GE GEAP19932593A patent/GEP19981431B/en unknown
- 1993-06-03 JP JP50108994A patent/JP3296490B2/ja not_active Expired - Fee Related
- 1993-06-03 AU AU43226/93A patent/AU666558B2/en not_active Ceased
- 1993-06-03 MD MD96-0305A patent/MD1743B2/ro unknown
- 1993-06-03 WO PCT/EP1993/001406 patent/WO1993025524A1/en active IP Right Grant
- 1993-06-04 IL IL105909A patent/IL105909A/xx not_active IP Right Cessation
- 1993-06-04 CN CN93108296A patent/CN1082318A/zh active Pending
-
1996
- 1996-08-16 GR GR960401179T patent/GR3020807T3/el unknown
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1966206A1 (de) * | 1968-04-26 | 1972-01-20 | Sumitomo Chemical Co | 1,4-Benzodiazepine und Arzneipraeparate |
DE2008692A1 (de) * | 1969-02-26 | 1970-09-17 | Agence Nationale de Valorisation de La Recherche (ANVAR), Puteaux, Hautsde-Seine (Prankreich) | Verfahren zur Herstellung von Indol-3carbonsäurederivaten und nach dem Verfahren erhältliche, neue Verbindungen |
JPH0570358A (ja) * | 1991-09-10 | 1993-03-23 | Kao Corp | 象牙質知覚過敏治療剤 |
JPH0570357A (ja) * | 1991-09-12 | 1993-03-23 | Fuso Yakuhin Kogyo Kk | 血液透析用顆粒剤 |
Also Published As
Publication number | Publication date |
---|---|
JPH07507323A (ja) | 1995-08-10 |
ES2091615T3 (es) | 1996-11-01 |
HUT69737A (en) | 1995-09-28 |
AU666558B2 (en) | 1996-02-15 |
TW229140B (ro) | 1994-09-01 |
DE69304057T2 (de) | 1997-02-06 |
JP3296490B2 (ja) | 2002-07-02 |
DK0643695T3 (da) | 1996-09-02 |
HU9403475D0 (en) | 1995-03-28 |
EP0643695B1 (en) | 1996-08-14 |
CN1082318A (zh) | 1994-02-23 |
EP0643695A1 (en) | 1995-03-22 |
US5399559A (en) | 1995-03-21 |
IL105909A (en) | 1997-04-15 |
WO1993025524A1 (en) | 1993-12-23 |
IL105909A0 (en) | 1993-10-20 |
ATE141260T1 (de) | 1996-08-15 |
DE69304057D1 (de) | 1996-09-19 |
AU4322693A (en) | 1994-01-04 |
GR3020807T3 (en) | 1996-11-30 |
ZA933846B (en) | 1993-12-28 |
HU216814B (hu) | 1999-08-30 |
GEP19981431B (en) | 1998-10-30 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MD1743B2 (ro) | Derivaţi ai indolului, procedeu de obţinere a lor, compoziţie fungicidă şi procedeu de combatere a fungilor | |
IL111245A0 (en) | Cyclic amides and fungicidal compositions containing them | |
EP0256503A3 (en) | Pyridinecarboxamide derivatives and their use as fungicide | |
GR3021270T3 (en) | Alkoxyiminoacetamide derivatives and their use as fungicides | |
HUT55605A (en) | Herbicide compositions containing diamino-triazine derivatives as active componentsand process for producing the active components | |
EP0324387A3 (en) | Composition for treatment of ischemic disorder in organs | |
IE880772L (en) | Benzoxazines | |
MY109714A (en) | Process for preparing 8-chloroquinolone derivatives | |
EP0555479A4 (ro) | ||
AU572888B2 (en) | 4-(3-alkynyloxy-2-hydroxy-propyl)-piperazin-i-yl-n- phenyl-acetamide derivatives | |
ATE150971T1 (de) | Zusammensetzung zur beschleunigung der wundheilung | |
EP0590681A3 (en) | A process for the preparation of aminothiadiazolylacetyl halide derivatives | |
NO903514D0 (no) | Imidazolderivat og fremgangsmaate til dets fremstilling. | |
NZ333414A (en) | Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity | |
ATE127453T1 (de) | Maleimidderivat, verfahren zu seiner herstellung und dieses maleimidderivat als wirkstoff enthaltende fungizid für den acker- und gartenbau. | |
DK0565059T3 (da) | Indolderivat | |
MX9603762A (es) | N-(arilmetil-sustituidas)-4-[bis-(fenil-sustituidas)metil]piperidina insecticidas. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PD99 | Pending application |