MA42409A - Oxystérols et leurs procédés d'utilisation - Google Patents

Oxystérols et leurs procédés d'utilisation

Info

Publication number
MA42409A
MA42409A MA042409A MA42409A MA42409A MA 42409 A MA42409 A MA 42409A MA 042409 A MA042409 A MA 042409A MA 42409 A MA42409 A MA 42409A MA 42409 A MA42409 A MA 42409A
Authority
MA
Morocco
Prior art keywords
oxysterols
methods
Prior art date
Application number
MA042409A
Other languages
English (en)
Inventor
Botella Gabriel Martinez
Albert Jean Robichaud
Francesco G Salituro
Original Assignee
Sage Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sage Therapeutics Inc filed Critical Sage Therapeutics Inc
Publication of MA42409A publication Critical patent/MA42409A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0055—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/582—Recycling of unreacted starting or intermediate materials
MA042409A 2015-07-06 2016-07-06 Oxystérols et leurs procédés d'utilisation MA42409A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562189065P 2015-07-06 2015-07-06

Publications (1)

Publication Number Publication Date
MA42409A true MA42409A (fr) 2018-05-16

Family

ID=57686058

Family Applications (1)

Application Number Title Priority Date Filing Date
MA042409A MA42409A (fr) 2015-07-06 2016-07-06 Oxystérols et leurs procédés d'utilisation

Country Status (8)

Country Link
US (3) US10696712B2 (fr)
EP (2) EP4316591A3 (fr)
JP (2) JP6882996B2 (fr)
AU (2) AU2016289965B2 (fr)
CA (1) CA2991311A1 (fr)
HK (1) HK1255500A1 (fr)
MA (1) MA42409A (fr)
WO (1) WO2017007832A1 (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT2753632T (lt) 2011-09-08 2023-07-10 Sage Therapeutics, Inc. Neuroaktyvieji steroidai, jų kompozicijos ir naudojimas
ES2699445T3 (es) 2013-03-13 2019-02-11 Sage Therapeutics Inc Esteroides neuroactivos y métodos de utilización de los mismos
US10259840B2 (en) 2014-06-18 2019-04-16 Sage Therapeutics, Inc. Oxysterols and methods of use thereof
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IL256710B2 (en) 2015-07-06 2024-01-01 Sage Therapeutics Inc Oxysterols and methods of using them
CA2991311A1 (fr) 2015-07-06 2017-01-12 Sage Therapeutics, Inc. Oxysterols et leurs procedes d'utilisation
MX2020010690A (es) * 2015-07-06 2022-02-25 Sage Therapeutics Inc Oxiesteroles y metodos de uso de los mismos.
PL3436022T3 (pl) 2016-04-01 2022-08-08 Sage Therapeutics, Inc. Oksysterole i sposoby ich stosowania
US10752653B2 (en) 2016-05-06 2020-08-25 Sage Therapeutics, Inc. Oxysterols and methods of use thereof
SI3481846T1 (sl) 2016-07-07 2021-11-30 Sage Therapeutics, Inc. 11-substituirani 24-hidroksisteroli za uporabo pri zdravljenju stanj, povezanih z NMDA
ES2935057T3 (es) 2016-09-30 2023-03-01 Sage Therapeutics Inc C7 oxisteroles sustituidos y estos compuestos para su uso como moduladores de la NMDA
CA3234484A1 (fr) 2016-10-18 2018-04-26 Sage Therapeutics, Inc. Oxysterols et leurs procedes d'utilisation
RU2019115112A (ru) 2016-10-18 2020-11-24 Сейдж Терапьютикс, Инк. Оксистеролы и способы их применения
US10857163B1 (en) 2019-09-30 2020-12-08 Athenen Therapeutics, Inc. Compositions that preferentially potentiate subtypes of GABAA receptors and methods of use thereof
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WO2023114224A1 (fr) 2021-12-13 2023-06-22 Sage Therapeutics, Inc. Combinaison de modulateurs positifs du récepteur muscarinique et de modulateurs allostériques positifs de nmda

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Also Published As

Publication number Publication date
EP3319610A4 (fr) 2019-03-06
CA2991311A1 (fr) 2017-01-12
JP6882996B2 (ja) 2021-06-02
EP4316591A2 (fr) 2024-02-07
US20230047157A1 (en) 2023-02-16
HK1255500A1 (zh) 2019-08-16
AU2016289965B2 (en) 2021-09-09
WO2017007832A1 (fr) 2017-01-12
US20180201643A1 (en) 2018-07-19
JP2021063118A (ja) 2021-04-22
JP2018519329A (ja) 2018-07-19
US20210101925A1 (en) 2021-04-08
JP2022130668A (ja) 2022-09-06
AU2021218227B2 (en) 2023-08-03
US10696712B2 (en) 2020-06-30
EP4316591A3 (fr) 2024-04-24
JP7410062B2 (ja) 2024-01-09
EP3319610A1 (fr) 2018-05-16
AU2021218227A1 (en) 2021-09-09
AU2016289965A1 (en) 2018-01-18

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