MA26867A1 - Ether-dicarboxylates de calcium, procedes pour leur preparation et traitement de maladies vasculaires et du diabete avec ces composés - Google Patents

Ether-dicarboxylates de calcium, procedes pour leur preparation et traitement de maladies vasculaires et du diabete avec ces composés

Info

Publication number
MA26867A1
MA26867A1 MA26735A MA26735A MA26867A1 MA 26867 A1 MA26867 A1 MA 26867A1 MA 26735 A MA26735 A MA 26735A MA 26735 A MA26735 A MA 26735A MA 26867 A1 MA26867 A1 MA 26867A1
Authority
MA
Morocco
Prior art keywords
treatment
dicarboxylates
diabetes
preparation
vascular diseases
Prior art date
Application number
MA26735A
Other languages
English (en)
Inventor
Yoshihisa Ando Howard
Eurgene Butler Donald
Jay Dozeman Gary
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of MA26867A1 publication Critical patent/MA26867A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/125Saturated compounds having only one carboxyl group and containing ether groups, groups, groups, or groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/235Saturated compounds containing more than one carboxyl group
    • C07C59/305Saturated compounds containing more than one carboxyl group containing ether groups, groups, groups, or groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)

Abstract

DEPOSANT Société dite: WARNER-LAMBERTCOMPANY REVENDICATION DE PRIORITES US 25 Janvier 2000 60/177,823 "Ether-dicarboxylates de calcium, procédés pour leur préparation et traitement de maladies vasculaires et du diabète avec ces composés" Les produits de solvatation avec des alcools et l'eau du sel monocalcique d'acide 6-(5-carboxy-5-méthyi-hexyloxy)-2,2-diméthyl-hexanoïque sont cristallins et répondent à la formule (I), dans laquelle R1 représente H ou un groupe alkyle inférieur, et x est un nombre de 0 à 10, et sont utiles pour le traitement de la dyslipidémie.
MA26735A 2000-01-25 2002-07-22 Ether-dicarboxylates de calcium, procedes pour leur preparation et traitement de maladies vasculaires et du diabete avec ces composés MA26867A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17782300P 2000-01-25 2000-01-25

Publications (1)

Publication Number Publication Date
MA26867A1 true MA26867A1 (fr) 2004-12-20

Family

ID=22650106

Family Applications (1)

Application Number Title Priority Date Filing Date
MA26735A MA26867A1 (fr) 2000-01-25 2002-07-22 Ether-dicarboxylates de calcium, procedes pour leur preparation et traitement de maladies vasculaires et du diabete avec ces composés

Country Status (39)

Country Link
EP (1) EP1259474B1 (fr)
JP (1) JP4750995B2 (fr)
KR (1) KR20020073182A (fr)
CN (1) CN1395555A (fr)
AP (1) AP2002002587A0 (fr)
AR (1) AR029436A1 (fr)
AT (1) ATE431326T1 (fr)
AU (1) AU2214001A (fr)
BG (1) BG106851A (fr)
BR (1) BR0107763A (fr)
CA (1) CA2397960C (fr)
CO (1) CO5261537A1 (fr)
CZ (1) CZ20022474A3 (fr)
DE (1) DE60138686D1 (fr)
DK (1) DK1259474T3 (fr)
DZ (1) DZ3239A1 (fr)
EA (1) EA004862B1 (fr)
EE (1) EE200200404A (fr)
ES (1) ES2324281T3 (fr)
GE (1) GEP20053428B (fr)
GT (1) GT200100015A (fr)
HN (1) HN2001000011A (fr)
HU (1) HUP0204422A3 (fr)
IL (1) IL150541A0 (fr)
IS (1) IS6442A (fr)
MA (1) MA26867A1 (fr)
MX (1) MXPA02007223A (fr)
NO (1) NO20023526L (fr)
NZ (1) NZ519550A (fr)
OA (1) OA12166A (fr)
PA (1) PA8510601A1 (fr)
PE (1) PE20011064A1 (fr)
PL (1) PL357076A1 (fr)
SK (1) SK10622002A3 (fr)
SV (1) SV2002000290A (fr)
TN (1) TNSN01013A1 (fr)
UY (1) UY26550A1 (fr)
WO (1) WO2001055078A1 (fr)
ZA (1) ZA200205880B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI1045691T1 (en) * 1997-12-12 2005-04-30 Warner-Lambert Company Llc Statin-carboxyalkylether combinations
MXPA05001254A (es) * 2002-08-22 2005-06-08 Warner Lambert Co Procedimiento para el tratamiento de la osteoartritis.
JPWO2006115130A1 (ja) * 2005-04-19 2008-12-18 エーザイ・アール・アンド・ディー・マネジメント株式会社 ビス[(2s)−3−[3−[(2s)−3−(4−クロロ−2−シアノフェノキシ)−2−フルオロプロポキシ]フェニル]−2−イソプロポキシプロピオン酸]カルシウム及びその中間体
US7816405B2 (en) 2005-04-19 2010-10-19 Eisai R&D Management Co., Ltd. Calcium bis [(2S)-3-[3-[(2S)-3-(4-chloro-2-cyanophenoxy)-2-fluoropropoxy]phenyl ]-2-isopropoxypropionate] and intermediate thereof
US10227285B2 (en) * 2014-11-14 2019-03-12 Gemphire Therapeutics Inc. Processes and intermediates for preparing alpha,omega-dicarboxylic acid-terminated dialkane ethers
US20180297929A1 (en) * 2017-04-18 2018-10-18 Gemphire Therapeutics Inc. Gemcabene, pharmaceutically acceptable salts thereof, compositions thereof and methods of use therefor
KR20210093900A (ko) * 2018-10-18 2021-07-28 젬파이어 세러퓨틱스 인코포레이티드 젬카빈, 이의 약학적으로 허용가능한 염, 이의 조성물 및 이의 사용 방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5648387A (en) 1995-03-24 1997-07-15 Warner-Lambert Company Carboxyalkylethers, formulations, and treatment of vascular diseases
NZ503982A (en) 1997-12-12 2002-03-28 Warner Lambert Co Statin-carboxyalkylether combinations useful for treating vascular disorders and diabetes mellitus

Also Published As

Publication number Publication date
CN1395555A (zh) 2003-02-05
DZ3239A1 (fr) 2001-08-02
CA2397960C (fr) 2008-09-09
AU2214001A (en) 2001-08-07
NO20023526L (no) 2002-08-27
SK10622002A3 (sk) 2003-07-01
CZ20022474A3 (cs) 2003-06-18
NZ519550A (en) 2003-11-28
TNSN01013A1 (fr) 2005-11-10
CA2397960A1 (fr) 2001-08-02
EP1259474B1 (fr) 2009-05-13
JP4750995B2 (ja) 2011-08-17
IL150541A0 (en) 2003-02-12
BR0107763A (pt) 2002-11-12
DK1259474T3 (da) 2009-07-20
PL357076A1 (en) 2004-07-12
EA004862B1 (ru) 2004-08-26
AR029436A1 (es) 2003-06-25
HN2001000011A (es) 2001-06-13
ATE431326T1 (de) 2009-05-15
WO2001055078A1 (fr) 2001-08-02
IS6442A (is) 2002-06-25
DE60138686D1 (de) 2009-06-25
UY26550A1 (es) 2001-08-27
PE20011064A1 (es) 2001-10-22
HUP0204422A3 (en) 2003-08-28
EP1259474A1 (fr) 2002-11-27
AP2002002587A0 (en) 2002-09-30
ZA200205880B (en) 2003-07-23
OA12166A (en) 2003-11-07
NO20023526D0 (no) 2002-07-24
HUP0204422A2 (en) 2003-05-28
MXPA02007223A (es) 2002-11-29
ES2324281T3 (es) 2009-08-04
EE200200404A (et) 2003-10-15
JP2003520835A (ja) 2003-07-08
BG106851A (en) 2003-01-31
KR20020073182A (ko) 2002-09-19
GEP20053428B (en) 2005-01-25
EA200200641A1 (ru) 2002-12-26
GT200100015A (es) 2001-10-19
SV2002000290A (es) 2002-07-16
PA8510601A1 (es) 2002-08-26
CO5261537A1 (es) 2003-03-31

Similar Documents

Publication Publication Date Title
MA27946A1 (fr) Omega-carboxyaryldiphenyluree fluoro-substituee pour le traitement et la prevention de maladies et d'etats pathologiques.
CN101842360B (zh) 抗感染嘧啶及其用途
MA27774A1 (fr) Inhibiteurs de phosphatidylinositol 3-kinase
MA30801B1 (fr) Biaryl-ether-urees
TNSN96172A1 (fr) Composes heterocycliques, procede pour leur preparation et compositions pharmaceutiques les contenant.
TNSN00202A1 (fr) Derives de n-[(purine - 2- yl) methyl]-sulfonamide nouveaux, procede pour leur preparation et compositions les contenant
MA26697A1 (fr) Composes nouveaux inhibiteurs de gsk-3 et compositions pharmaceutiques les contenant
TNSN00203A1 (fr) Derives de purine nouveaux, procede pour leur preparation et des compositions les contenant
TNSN99106A1 (fr) Derives d'isothiazole nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant.
TNSN99156A1 (fr) Derives d'acide hydroxypipecolate-hydroxamique nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant
MA28747B1 (fr) Dérivés de pyridine
UA77454C2 (en) N-substituted hydroxypyrimidinone carboxamide inhibitors of hiv integrase
CN102803223A (zh) 具有取代苯基的环状化合物
MA25035A1 (fr) Derives de 3-azabicyclo [3,1,0] hexane nouveaux, procede pour leur preparation et compositions les contenant
MA28271A1 (fr) Dérivés de benzènesulfonylamino-pyridine -2-yle et composés apparentés servant d'inhibiteurs de la 11-bêta- hydroxystéroïde-déshydrogénase de type 1(11-bêta-HSD-1)pour le traitement du diabète et de l'obésité
MA26864A1 (fr) Antagonistes du facteur de liberation de corticotrophine.
TNSN05250A1 (fr) Pyrimidinones substituees
TNSN99031A1 (fr) Composes heterocycliques nouveaux inhibiteurs de romatases, procede pour leur preparation et compositions pharmaceutiques les contenant
CN101084224A (zh) 具有杀真菌活性的噻吩并-嘧啶化合物
TNSN98024A1 (fr) 2-amino-6-(2-substitue-4-phenoxy)-substitue-pyridines, procede pour leur preparation et compositions pharmaceutiques les contenant.
MA26696A1 (fr) Derives de tetrahydrobenzazepine nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant
TNSN01126A1 (fr) Imidazoles substitues nouveaux, procede pour leur preparation et compositions les contenant
GB2196962A (en) Substituted 2-benzyl-mercapto-imidazoles and analogs useful as anti-inflammatory agents
MA26867A1 (fr) Ether-dicarboxylates de calcium, procedes pour leur preparation et traitement de maladies vasculaires et du diabete avec ces composés
TNSN01094A1 (fr) Derives de 3-azabicyclo [3,1,0] hexane nouveaux, procede pour leur preparation et compositions les contenant