LV12102B - ROTAMASE FUNCTIONS INHIBITORS - Google Patents
ROTAMASE FUNCTIONS INHIBITORS Download PDFInfo
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- LV12102B LV12102B LVP-98-85A LV980085A LV12102B LV 12102 B LV12102 B LV 12102B LV 980085 A LV980085 A LV 980085A LV 12102 B LV12102 B LV 12102B
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- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 description 1
- 239000012049 topical pharmaceutical composition Substances 0.000 description 1
- 206010044652 trigeminal neuralgia Diseases 0.000 description 1
- ZDPHROOEEOARMN-UHFFFAOYSA-N undecanoic acid Chemical compound CCCCCCCCCCC(O)=O ZDPHROOEEOARMN-UHFFFAOYSA-N 0.000 description 1
- 230000002792 vascular Effects 0.000 description 1
- 238000009736 wetting Methods 0.000 description 1
- 239000003871 white petrolatum Substances 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/551,026 US20020013344A1 (en) | 1995-10-31 | 1995-10-31 | Rotamas enzyme activity inhibitors |
| US08/645,149 US5801197A (en) | 1995-10-31 | 1996-05-13 | Rotamase enzyme activity inhibitors |
| PCT/US1996/013624 WO1997016190A1 (en) | 1995-10-31 | 1996-08-26 | Rotamase enzyme activity inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| LV12102A LV12102A (lv) | 1998-08-20 |
| LV12102B true LV12102B (en) | 1998-10-20 |
Family
ID=27069634
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LVP-98-85A LV12102B (en) | 1995-10-31 | 1998-06-25 | ROTAMASE FUNCTIONS INHIBITORS |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5801197A (cs) |
| EP (1) | EP0859614A4 (cs) |
| JP (1) | JPH11514643A (cs) |
| KR (1) | KR19990067257A (cs) |
| BG (1) | BG62596B1 (cs) |
| BR (1) | BRPI9611271A2 (cs) |
| CA (1) | CA2236328A1 (cs) |
| CZ (1) | CZ125198A3 (cs) |
| EA (1) | EA001481B1 (cs) |
| EE (1) | EE9800125A (cs) |
| HU (1) | HUP9901752A3 (cs) |
| LV (1) | LV12102B (cs) |
| NO (1) | NO981903L (cs) |
| NZ (1) | NZ316361A (cs) |
| PL (1) | PL326420A1 (cs) |
| SK (1) | SK55998A3 (cs) |
| WO (1) | WO1997016190A1 (cs) |
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| WO1995012572A1 (en) * | 1993-11-04 | 1995-05-11 | Abbott Laboratories | Cyclobutane derivatives as inhibitors of squalene synthetase and protein farnesyltransferase |
| DE69512220T2 (de) * | 1994-03-07 | 2000-03-16 | Vertex Pharmaceuticals Inc. | Sulfonamidderivate als aspartylprotease-inhibitoren |
| US5744485A (en) * | 1994-03-25 | 1998-04-28 | Vertex Pharmaceuticals Incorporated | Carbamates and ureas as modifiers of multi-drug resistance |
| US5856116A (en) * | 1994-06-17 | 1999-01-05 | Vertex Pharmaceuticals, Incorporated | Crystal structure and mutants of interleukin-1 beta converting enzyme |
| US5716929A (en) * | 1994-06-17 | 1998-02-10 | Vertex Pharmaceuticals, Inc. | Inhibitors of interleukin-1β converting enzyme |
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| IL115685A (en) * | 1994-11-16 | 2000-08-31 | Vertex Pharma | Amino acid derivatives pharmaceutical compositions containing the same and processes for the preparation thereof |
| US5621108A (en) * | 1994-12-05 | 1997-04-15 | Trustees Of The University Of Pennsylvania | Processes and intermediates for preparing macrocycles |
| US5859031A (en) * | 1995-06-07 | 1999-01-12 | Gpi Nil Holdings, Inc. | Small molecule inhibitors of rotamase enzyme activity |
| US5696135A (en) * | 1995-06-07 | 1997-12-09 | Gpi Nil Holdings, Inc. | Inhibitors of rotamase enzyme activity effective at stimulating neuronal growth |
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-
1996
- 1996-05-13 US US08/645,149 patent/US5801197A/en not_active Expired - Lifetime
- 1996-08-26 KR KR1019980703218A patent/KR19990067257A/ko not_active Application Discontinuation
- 1996-08-26 CA CA002236328A patent/CA2236328A1/en not_active Abandoned
- 1996-08-26 JP JP9517308A patent/JPH11514643A/ja active Pending
- 1996-08-26 HU HU9901752A patent/HUP9901752A3/hu unknown
- 1996-08-26 EA EA199800329A patent/EA001481B1/ru not_active IP Right Cessation
- 1996-08-26 CZ CZ981251A patent/CZ125198A3/cs unknown
- 1996-08-26 EP EP96929014A patent/EP0859614A4/en not_active Withdrawn
- 1996-08-26 WO PCT/US1996/013624 patent/WO1997016190A1/en not_active Application Discontinuation
- 1996-08-26 PL PL96326420A patent/PL326420A1/xx unknown
- 1996-08-26 SK SK559-98A patent/SK55998A3/sk unknown
- 1996-08-26 BR BRPI9611271-9A patent/BRPI9611271A2/pt unknown
- 1996-08-26 NZ NZ316361A patent/NZ316361A/xx unknown
- 1996-08-26 EE EE9800125A patent/EE9800125A/xx unknown
-
1998
- 1998-04-27 NO NO981903A patent/NO981903L/no not_active Application Discontinuation
- 1998-04-28 BG BG102410A patent/BG62596B1/bg unknown
- 1998-06-25 LV LVP-98-85A patent/LV12102B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EE9800125A (et) | 1998-10-15 |
| WO1997016190A1 (en) | 1997-05-09 |
| US5801197A (en) | 1998-09-01 |
| MX9803356A (es) | 1998-09-30 |
| BG62596B1 (bg) | 2000-03-31 |
| CZ125198A3 (cs) | 1998-12-16 |
| NO981903L (no) | 1998-06-30 |
| SK55998A3 (en) | 1999-02-11 |
| JPH11514643A (ja) | 1999-12-14 |
| EA001481B1 (ru) | 2001-04-23 |
| EP0859614A4 (en) | 2000-04-26 |
| EA199800329A1 (ru) | 1998-12-24 |
| NO981903D0 (no) | 1998-04-27 |
| EP0859614A1 (en) | 1998-08-26 |
| BRPI9611271A2 (pt) | 2019-04-30 |
| AU6857396A (en) | 1997-05-22 |
| CA2236328A1 (en) | 1997-05-09 |
| NZ316361A (en) | 1999-08-30 |
| KR19990067257A (ko) | 1999-08-16 |
| HUP9901752A3 (en) | 2001-04-28 |
| HUP9901752A2 (hu) | 1999-10-28 |
| BG102410A (en) | 1998-12-30 |
| PL326420A1 (en) | 1998-09-14 |
| AU713302B2 (en) | 1999-11-25 |
| LV12102A (lv) | 1998-08-20 |
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