LV11612B - Novel high enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-beta-amino acids - Google Patents

Novel high enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-beta-amino acids Download PDF

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Publication number
LV11612B
LV11612B LVP-96-233A LV960233A LV11612B LV 11612 B LV11612 B LV 11612B LV 960233 A LV960233 A LV 960233A LV 11612 B LV11612 B LV 11612B
Authority
LV
Latvia
Prior art keywords
carbon atoms
unbranched
phenyl
group
case
Prior art date
Application number
LVP-96-233A
Other languages
English (en)
Latvian (lv)
Other versions
LV11612A (lv
Inventor
Joachim Mittendorf
Hermann Arold
Peter Fey
Michael Matzke
Hans-Christiaan Militzer
Klaus-Helmut Mohr
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of LV11612A publication Critical patent/LV11612A/xx
Publication of LV11612B publication Critical patent/LV11612B/lv

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C07C227/32—Preparation of optical isomers by stereospecific synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/24—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/74—Esters of carboxylic acids having an esterified carboxyl group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
LVP-96-233A 1994-01-13 1996-07-12 Novel high enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-beta-amino acids LV11612B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4400749A DE4400749A1 (de) 1994-01-13 1994-01-13 Neues hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan- und -penten-beta-Aminosäuren
PCT/EP1995/000059 WO1995019337A1 (fr) 1994-01-13 1995-01-09 NOUVEAU PROCEDE HAUTEMENT ENANTIO-SELECTIF POUR LA FABRICATION DE β AMINO-ACIDES DE CYCLOPENTANE ET DE CYCLOPENTENE ENANTIOMERIQUEMENT PURS

Publications (2)

Publication Number Publication Date
LV11612A LV11612A (lv) 1996-12-20
LV11612B true LV11612B (en) 1997-06-20

Family

ID=6507806

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-96-233A LV11612B (en) 1994-01-13 1996-07-12 Novel high enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-beta-amino acids

Country Status (25)

Country Link
US (1) US5962724A (fr)
EP (2) EP0788473B1 (fr)
JP (2) JP4020425B2 (fr)
CN (1) CN1138850A (fr)
AT (1) ATE227259T1 (fr)
AU (1) AU690626B2 (fr)
BR (1) BR9506509A (fr)
CZ (1) CZ192896A3 (fr)
DE (2) DE4400749A1 (fr)
DK (1) DK0788473T3 (fr)
EE (1) EE9600136A (fr)
ES (1) ES2185692T3 (fr)
FI (1) FI962820A (fr)
HU (1) HUT74935A (fr)
LV (1) LV11612B (fr)
MX (1) MX9602756A (fr)
NO (1) NO314451B1 (fr)
NZ (1) NZ278595A (fr)
PL (1) PL315540A1 (fr)
PT (1) PT788473E (fr)
SI (1) SI0788473T1 (fr)
SK (1) SK91296A3 (fr)
TW (1) TW363966B (fr)
WO (1) WO1995019337A1 (fr)
ZA (1) ZA95208B (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19548825C2 (de) * 1995-12-27 1999-03-25 Rolf Dr Hermann Neue, substituierte Cyclopentylaminderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE19617772A1 (de) * 1996-05-03 1997-11-13 Bayer Ag Neues effizientes und hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan-beta-aminosäuren
DE19727517A1 (de) * 1997-06-30 1999-01-07 Basf Ag Racematspaltung von Aminosäureestern durch Enzym-katalysierte Acylierung
CU23048A3 (es) 1997-10-27 2005-06-24 Warner Lambert Co Aminoacidos ciclicos y derivados de los mismos, utiles como agentes farmaceuticos
CA2527632A1 (fr) 2003-06-02 2004-12-09 F. Hoffmann-La Roche Ag Derives de benzamide nitrile
US7084178B2 (en) * 2003-11-26 2006-08-01 Bristol-Myers Squibb Company Antiamyloid phenylsulfonamides: N-cycloalkylcarboxamides derivatives
DE602005026047D1 (de) * 2004-11-03 2011-03-03 Hoffmann La Roche Dicarbonsäureamidderivate und deren verwendung als inhibitoren von faktor xa
CN1332934C (zh) * 2005-01-14 2007-08-22 清华大学 一种用于氨基酸对映体分离的新型试剂
EP2294054A4 (fr) * 2008-06-05 2012-04-18 Dsm Ip Assets Bv Procédé de préparation de (4s,5r)-semi-ester
JP6420106B2 (ja) * 2014-09-30 2018-11-07 富士フイルム株式会社 環構造を有するジカルボン酸モノエステルの製造方法、ジカルボン酸モノエステルアミン塩、ジカルボン酸モノエステルを用いた液晶化合物の製造方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499079A (en) * 1982-11-18 1985-02-12 E. R. Squibb & Sons, Inc. Carboxy and substituted carboxy alkanoyl and cycloalkanoyl peptides
AU673824B2 (en) * 1992-05-29 1996-11-28 Bayer Aktiengesellschaft Cyclopentane- and -pentene-beta-amino acids

Also Published As

Publication number Publication date
ZA95208B (en) 1995-09-08
DE59510446D1 (de) 2002-12-12
DK0788473T3 (da) 2003-03-03
EP0788473A1 (fr) 1997-08-13
NO962912L (no) 1996-07-10
TW363966B (en) 1999-07-11
SI0788473T1 (en) 2003-04-30
CZ192896A3 (en) 1996-10-16
NO314451B1 (no) 2003-03-24
US5962724A (en) 1999-10-05
AU690626B2 (en) 1998-04-30
PT788473E (pt) 2003-02-28
PL315540A1 (en) 1996-11-12
DE4400749A1 (de) 1995-07-20
EP1256568A1 (fr) 2002-11-13
AU1455495A (en) 1995-08-01
NZ278595A (en) 1998-04-27
NO962912D0 (no) 1996-07-10
EE9600136A (et) 1997-04-15
WO1995019337A1 (fr) 1995-07-20
SK91296A3 (en) 1996-12-04
FI962820A0 (fi) 1996-07-11
MX9602756A (es) 1997-05-31
HUT74935A (en) 1997-03-28
BR9506509A (pt) 1997-09-09
CN1138850A (zh) 1996-12-25
ATE227259T1 (de) 2002-11-15
ES2185692T3 (es) 2003-05-01
HU9601913D0 (en) 1996-09-30
FI962820A (fi) 1996-07-11
EP0788473B1 (fr) 2002-11-06
JPH09508107A (ja) 1997-08-19
JP4020425B2 (ja) 2007-12-12
LV11612A (lv) 1996-12-20
JP2005187481A (ja) 2005-07-14

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